Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50028457
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50257066(1-(6-(4-chlorophenoxy)hexyl)-2-ethynyl-3-(pyridin-...)
Affinity DataIC50: 8nMAssay Description:Inhibition of IKK-beta by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50135482(1-(5-Methoxy-2-thiophen-2-yl-quinazolin-4-ylamino)...)
Affinity DataIC50: 8nMAssay Description:Inhibition of IKK-beta by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50230828([5-(p-fluorophenyl)-2-ureido]thiophene-3-carboxami...)
Affinity DataIC50: 18nMAssay Description:Inhibition of IKK-beta by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50257010(5-(2-(2-(benzyl(methyl)amino)ethoxy)phenyl)-2-urei...)
Affinity DataIC50: 40nMAssay Description:Inhibition of IKK-beta by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50257065((S)-3-(ethyl(phenyl)amino)-2-(2-(pyridin-4-yl)-1H-...)
Affinity DataIC50: 70nMAssay Description:Inhibition of IKK-beta by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50257012(4-amino-2-(2,5-dihydroxyphenyl)-6-(piperidin-3-yl)...)
Affinity DataIC50: 316nMAssay Description:Inhibition of IKK-beta by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM7166(CHEMBL361862 | 3-(4-sulfamoylphenyl)-3,4,10,11-tet...)
Affinity DataIC50: 670nMAssay Description:Inhibition of IKK-beta by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50256912((Z)-5-(3,4-dihydroxybenzylidene)-2-iminothiazolidi...)
Affinity DataIC50: 1.76E+3nMAssay Description:Inhibition of IKK-beta by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50257011((S)-7-(2-(cyclopropylmethoxy)-6-hydroxyphenyl)-5-(...)
Affinity DataKi:  2nMAssay Description:Inhibition of IKK-beta by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed