Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50028365
TargetMitogen-activated protein kinase 14(Human)
Eberhard-Karls-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50241111(3-(2-amino-4-fluoro-phenylamino)-6,11-dihydro-dibe...)
Affinity DataIC50: 40nMAssay Description:Inhibition of p38alpha MAPK by cell-free enzyme immunosorbent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Eberhard-Karls-UniversitäT

Curated by ChEMBL
LigandPNGBDBM13336(4-{4-(4-fluorophenyl)-2-[4-(methylsulfinyl)phenyl]...)
Affinity DataIC50: 50nMAssay Description:Inhibition of p38alpha MAPK by cell-free enzyme immunosorbent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Eberhard-Karls-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50241112(2-(2-Amino-phenylamino)-10,11-dihydro-dibenzo[a,d]...)
Affinity DataIC50: 100nMAssay Description:Inhibition of p38alpha MAPK by cell-free enzyme immunosorbent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMitogen-activated protein kinase 14(Human)
Eberhard-Karls-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50248858(2-(2-Amino-4-fluoro-phenylamino)-10,11-dihydro-dib...)
Affinity DataIC50: 130nMAssay Description:Inhibition of p38alpha MAPK by cell-free enzyme immunosorbent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Eberhard-Karls-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50248859(2-(2,4-Difluoro-phenylamino)-10,11-dihydro-dibenzo...)
Affinity DataIC50: 130nMAssay Description:Inhibition of p38alpha MAPK by cell-free enzyme immunosorbent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Eberhard-Karls-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50248941(8-(2,4-Difluoro-phenylamino)-11H-10-oxa-1-aza-dibe...)
Affinity DataIC50: 180nMAssay Description:Inhibition of p38alpha MAPK by cell-free enzyme immunosorbent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Eberhard-Karls-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50248913(8-(2,4-Difluoro-phenylamino)-10,11-dihydro-benzo[4...)
Affinity DataIC50: 240nMAssay Description:Inhibition of p38alpha MAPK by cell-free enzyme immunosorbent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Eberhard-Karls-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50241114(3-(2,4-difluoro-phenylamino)-6,11-dihydro-dibenzo[...)
Affinity DataIC50: 240nMAssay Description:Inhibition of p38alpha MAPK by cell-free enzyme immunosorbent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Eberhard-Karls-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50241115(3-(2-amino-phenylamino)-6,11-dihydro-dibenzo[b,e]o...)
Affinity DataIC50: 300nMAssay Description:Inhibition of p38alpha MAPK by cell-free enzyme immunosorbent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Eberhard-Karls-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50248890(8-(2-Amino-phenylamino)-10,11-dihydro-benzo[4,5]cy...)
Affinity DataIC50: 310nMAssay Description:Inhibition of p38alpha MAPK by cell-free enzyme immunosorbent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Eberhard-Karls-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50248889(8-(2,4-Difluoro-phenylamino)-benzo[4,5]cyclohepta[...)
Affinity DataIC50: 330nMAssay Description:Inhibition of p38alpha MAPK by cell-free enzyme immunosorbent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Eberhard-Karls-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50248915(8-(2-Amino-phenylamino)-5,6-dihydro-benzo[5,6]cycl...)
Affinity DataIC50: 440nMAssay Description:Inhibition of p38alpha MAPK by cell-free enzyme immunosorbent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Eberhard-Karls-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50241113(2-(2-amino-phenylamino)-dibenzo[a,d]cyclohepten-5-...)
Affinity DataIC50: 1.06E+3nMAssay Description:Inhibition of p38alpha MAPK by cell-free enzyme immunosorbent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Eberhard-Karls-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50248888(8-(2-Amino-phenylamino)-benzo[4,5]cyclohepta[1,2-b...)
Affinity DataIC50: 1.08E+3nMAssay Description:Inhibition of p38alpha MAPK by cell-free enzyme immunosorbent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Eberhard-Karls-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50248891(8-(2-Amino-4-fluoro-phenylamino)-10,11-dihydro-ben...)
Affinity DataIC50: 1.19E+3nMAssay Description:Inhibition of p38alpha MAPK by cell-free enzyme immunosorbent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Eberhard-Karls-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50248914(8-(2-Amino-phenylamino)-benzo[5,6]cyclohepta[1,2-c...)
Affinity DataIC50: 1.95E+3nMAssay Description:Inhibition of p38alpha MAPK by cell-free enzyme immunosorbent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Eberhard-Karls-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50248887(2-(2,4-Difluoro-phenylamino)-dibenzo[a,d]cyclohept...)
Affinity DataIC50: 2.53E+3nMAssay Description:Inhibition of p38alpha MAPK by cell-free enzyme immunosorbent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Eberhard-Karls-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50248939(8-(2-Amino-phenylamino)-11H-10-oxa-1-aza-dibenzo[a...)
Affinity DataIC50: 2.68E+3nMAssay Description:Inhibition of p38alpha MAPK by cell-free enzyme immunosorbent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Eberhard-Karls-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50248940(8-(2-Amino-4-fluoro-phenylamino)-11H-10-oxa-1-aza-...)
Affinity DataIC50: 2.73E+3nMAssay Description:Inhibition of p38alpha MAPK by cell-free enzyme immunosorbent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed