Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50028209
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50182369(4-(2-(4-fluorophenyl)-7-(1-methylpiperidin-4-yl)H-...)
Affinity DataIC50: 0.0440nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50248496(2-(4-(2-(4-fluorophenyl)-3-(pyridin-4-yl)-1H-indol...)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50248451(2-(4-fluorophenyl)-6-(1-methylpiperidin-4-yl)-3-(p...)
Affinity DataIC50: 0.150nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50248450(2-(4-fluorophenyl)-6-(piperidin-4-yl)-3-(pyridin-4...)
Affinity DataIC50: 0.150nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50248452(6-(1-ethylpiperidin-4-yl)-2-(4-fluorophenyl)-3-(py...)
Affinity DataIC50: 0.160nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50248396(4-(2-(4-fluorophenyl)-6-(piperidin-4-yl)-1H-indol-...)
Affinity DataIC50: 0.210nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50248543(4-(2-(4-fluorophenyl)-6-(1-methylpiperidin-4-yl)-1...)
Affinity DataIC50: 0.220nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50248397(2-(4-(3-(2-aminopyrimidin-4-yl)-2-(4-fluorophenyl)...)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50248399(2-(4-fluorophenyl)-6-(1-methylpiperidin-4-yl)-3-(p...)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50248498(2-(4-fluorophenyl)-6-(1-methylazetidin-3-yl)-3-(py...)
Affinity DataIC50: 0.620nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50248398(2-(4-fluorophenyl)-6-(piperidin-4-yl)-3-(pyrimidin...)
Affinity DataIC50: 0.650nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50248449(2-(4-(2-(4-fluorophenyl)-3-(pyrimidin-4-yl)-1H-ind...)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50248499(2-(4-fluorophenyl)-6-((1-methylpiperidin-4-yl)meth...)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50248542(2-(4-fluorophenyl)-6-((4-methylpiperazin-1-yl)meth...)
Affinity DataIC50: 8.90nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50248497(4-(2-(4-fluorophenyl)-3-(pyridin-4-yl)-1H-indol-6-...)
Affinity DataIC50: 9.20nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50248541((2-(4-fluorophenyl)-3-(pyridin-4-yl)-1H-indol-6-yl...)
Affinity DataIC50: 12.7nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed