Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 3040
LigandPNGBDBM19992(2-{3-[3-({[2-chloro-3-(trifluoromethyl)phenyl]meth...)
Affinity DataEC50:  25nMpH: 7.5 T: 2°CAssay Description:The LXR LiSA measures the ligand-dependent recruitment of a 25 amino acid fragment of the steroid receptor coactivator 1 (SRC1) to the ligand-binding...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM27174(2-{4-[3-({[2-chloro-3-(trifluoromethyl)phenyl]meth...)
Affinity DataEC50:  4nMpH: 7.5 T: 2°CAssay Description:The LXR LiSA measures the ligand-dependent recruitment of a 25 amino acid fragment of the steroid receptor coactivator 1 (SRC1) to the ligand-binding...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2009
Entry Details Article
PubMed
LigandPNGBDBM27173({[2-chloro-3-(trifluoromethyl)phenyl]methyl}(2,2-d...)
Affinity DataEC50:  7nMpH: 7.5 T: 2°CAssay Description:The LXR LiSA measures the ligand-dependent recruitment of a 25 amino acid fragment of the steroid receptor coactivator 1 (SRC1) to the ligand-binding...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2009
Entry Details Article
PubMed
LigandPNGBDBM27172({[2-chloro-3-(trifluoromethyl)phenyl]methyl}(2,2-d...)
Affinity DataEC50:  12nMpH: 7.5 T: 2°CAssay Description:The LXR LiSA measures the ligand-dependent recruitment of a 25 amino acid fragment of the steroid receptor coactivator 1 (SRC1) to the ligand-binding...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2009
Entry Details Article
PubMed
LigandPNGBDBM27171({[2-chloro-3-(trifluoromethyl)phenyl]methyl}(2,2-d...)
Affinity DataEC50:  15nMpH: 7.5 T: 2°CAssay Description:The LXR LiSA measures the ligand-dependent recruitment of a 25 amino acid fragment of the steroid receptor coactivator 1 (SRC1) to the ligand-binding...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2009
Entry Details Article
PubMed
LigandPNGBDBM27170({[2-chloro-3-(trifluoromethyl)phenyl]methyl}(2,2-d...)
Affinity DataEC50:  23nMpH: 7.5 T: 2°CAssay Description:The LXR LiSA measures the ligand-dependent recruitment of a 25 amino acid fragment of the steroid receptor coactivator 1 (SRC1) to the ligand-binding...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2009
Entry Details Article
PubMed
LigandPNGBDBM27169(methyl 2-{5-[3-({[2-chloro-3-(trifluoromethyl)phen...)
Affinity DataEC50:  288nMpH: 7.5 T: 2°CAssay Description:The LXR LiSA measures the ligand-dependent recruitment of a 25 amino acid fragment of the steroid receptor coactivator 1 (SRC1) to the ligand-binding...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2009
Entry Details Article
PubMed
LigandPNGBDBM27168({[2-chloro-3-(trifluoromethyl)phenyl]methyl}(2,2-d...)
Affinity DataEC50:  560nMpH: 7.5 T: 2°CAssay Description:The LXR LiSA measures the ligand-dependent recruitment of a 25 amino acid fragment of the steroid receptor coactivator 1 (SRC1) to the ligand-binding...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2009
Entry Details Article
PubMed
LigandPNGBDBM27167({[2-chloro-3-(trifluoromethyl)phenyl]methyl}[3-({4...)
Affinity DataEC50:  510nMpH: 7.5 T: 2°CAssay Description:The LXR LiSA measures the ligand-dependent recruitment of a 25 amino acid fragment of the steroid receptor coactivator 1 (SRC1) to the ligand-binding...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2009
Entry Details Article
PubMed
LigandPNGBDBM27166({[2-chloro-3-(trifluoromethyl)phenyl]methyl}(2,2-d...)
Affinity DataEC50:  60nMpH: 7.5 T: 2°CAssay Description:The LXR LiSA measures the ligand-dependent recruitment of a 25 amino acid fragment of the steroid receptor coactivator 1 (SRC1) to the ligand-binding...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2009
Entry Details Article
PubMed
LigandPNGBDBM27165(methyl 3-[3-({[2-chloro-3-(trifluoromethyl)phenyl]...)
Affinity DataEC50:  26nMpH: 7.5 T: 2°CAssay Description:The LXR LiSA measures the ligand-dependent recruitment of a 25 amino acid fragment of the steroid receptor coactivator 1 (SRC1) to the ligand-binding...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2009
Entry Details Article
PubMed
LigandPNGBDBM27164({[2-chloro-3-(trifluoromethyl)phenyl]methyl}(2,2-d...)
Affinity DataEC50:  15nMpH: 7.5 T: 2°CAssay Description:The LXR LiSA measures the ligand-dependent recruitment of a 25 amino acid fragment of the steroid receptor coactivator 1 (SRC1) to the ligand-binding...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2009
Entry Details Article
PubMed
LigandPNGBDBM19992(2-{3-[3-({[2-chloro-3-(trifluoromethyl)phenyl]meth...)
Affinity DataEC50:  175nMpH: 7.5 T: 2°CAssay Description:The LXR LiSA measures the ligand-dependent recruitment of a 25 amino acid fragment of the steroid receptor coactivator 1 (SRC1) to the ligand-binding...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM27174(2-{4-[3-({[2-chloro-3-(trifluoromethyl)phenyl]meth...)
Affinity DataEC50:  14nMpH: 7.5 T: 2°CAssay Description:The LXR LiSA measures the ligand-dependent recruitment of a 25 amino acid fragment of the steroid receptor coactivator 1 (SRC1) to the ligand-binding...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM27173({[2-chloro-3-(trifluoromethyl)phenyl]methyl}(2,2-d...)
Affinity DataEC50:  20nMpH: 7.5 T: 2°CAssay Description:The LXR LiSA measures the ligand-dependent recruitment of a 25 amino acid fragment of the steroid receptor coactivator 1 (SRC1) to the ligand-binding...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2009
Entry Details Article
PubMed
LigandPNGBDBM27172({[2-chloro-3-(trifluoromethyl)phenyl]methyl}(2,2-d...)
Affinity DataEC50:  39nMpH: 7.5 T: 2°CAssay Description:The LXR LiSA measures the ligand-dependent recruitment of a 25 amino acid fragment of the steroid receptor coactivator 1 (SRC1) to the ligand-binding...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2009
Entry Details Article
PubMed
LigandPNGBDBM27171({[2-chloro-3-(trifluoromethyl)phenyl]methyl}(2,2-d...)
Affinity DataEC50:  60nMpH: 7.5 T: 2°CAssay Description:The LXR LiSA measures the ligand-dependent recruitment of a 25 amino acid fragment of the steroid receptor coactivator 1 (SRC1) to the ligand-binding...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2009
Entry Details Article
PubMed
LigandPNGBDBM27170({[2-chloro-3-(trifluoromethyl)phenyl]methyl}(2,2-d...)
Affinity DataEC50:  226nMpH: 7.5 T: 2°CAssay Description:The LXR LiSA measures the ligand-dependent recruitment of a 25 amino acid fragment of the steroid receptor coactivator 1 (SRC1) to the ligand-binding...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2009
Entry Details Article
PubMed
LigandPNGBDBM27169(methyl 2-{5-[3-({[2-chloro-3-(trifluoromethyl)phen...)
Affinity DataEC50:  630nMpH: 7.5 T: 2°CAssay Description:The LXR LiSA measures the ligand-dependent recruitment of a 25 amino acid fragment of the steroid receptor coactivator 1 (SRC1) to the ligand-binding...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2009
Entry Details Article
PubMed
LigandPNGBDBM27168({[2-chloro-3-(trifluoromethyl)phenyl]methyl}(2,2-d...)
Affinity DataEC50:  790nMpH: 7.5 T: 2°CAssay Description:The LXR LiSA measures the ligand-dependent recruitment of a 25 amino acid fragment of the steroid receptor coactivator 1 (SRC1) to the ligand-binding...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2009
Entry Details Article
PubMed
LigandPNGBDBM27167({[2-chloro-3-(trifluoromethyl)phenyl]methyl}[3-({4...)
Affinity DataEC50: >3.00E+3nMpH: 7.5 T: 2°CAssay Description:The LXR LiSA measures the ligand-dependent recruitment of a 25 amino acid fragment of the steroid receptor coactivator 1 (SRC1) to the ligand-binding...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2009
Entry Details Article
PubMed
LigandPNGBDBM27166({[2-chloro-3-(trifluoromethyl)phenyl]methyl}(2,2-d...)
Affinity DataEC50:  110nMpH: 7.5 T: 2°CAssay Description:The LXR LiSA measures the ligand-dependent recruitment of a 25 amino acid fragment of the steroid receptor coactivator 1 (SRC1) to the ligand-binding...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2009
Entry Details Article
PubMed
LigandPNGBDBM27165(methyl 3-[3-({[2-chloro-3-(trifluoromethyl)phenyl]...)
Affinity DataEC50:  63nMpH: 7.5 T: 2°CAssay Description:The LXR LiSA measures the ligand-dependent recruitment of a 25 amino acid fragment of the steroid receptor coactivator 1 (SRC1) to the ligand-binding...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2009
Entry Details Article
PubMed
LigandPNGBDBM27164({[2-chloro-3-(trifluoromethyl)phenyl]methyl}(2,2-d...)
Affinity DataEC50:  23nMpH: 7.5 T: 2°CAssay Description:The LXR LiSA measures the ligand-dependent recruitment of a 25 amino acid fragment of the steroid receptor coactivator 1 (SRC1) to the ligand-binding...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2009
Entry Details Article
PubMed