Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50004163
TargetAurora kinase A(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479526(CHEMBL515560)
Affinity DataIC50: 33nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479524(CHEMBL474344)
Affinity DataIC50: 449nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479510(CHEMBL515112)
Affinity DataIC50: 460nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479520(CHEMBL473334)
Affinity DataIC50: 719nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479527(CHEMBL461954)
Affinity DataIC50: 804nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479521(CHEMBL461785)
Affinity DataIC50: 838nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479522(CHEMBL473131)
Affinity DataIC50: 960nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479528(CHEMBL518032)
Affinity DataIC50: 1.07E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479511(CHEMBL474540)
Affinity DataIC50: 1.09E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479517(CHEMBL461599)
Affinity DataIC50: 1.35E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479525(CHEMBL473333)
Affinity DataIC50: 1.45E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479531(CHEMBL517573)
Affinity DataIC50: 1.48E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479512(CHEMBL516353)
Affinity DataIC50: 1.57E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479516(CHEMBL460720)
Affinity DataIC50: 1.58E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479529(CHEMBL514951)
Affinity DataIC50: 1.58E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479519(CHEMBL461784)
Affinity DataIC50: 1.62E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479513(CHEMBL460905)
Affinity DataIC50: 1.75E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479533(CHEMBL460728)
Affinity DataIC50: 1.94E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479518(CHEMBL461972)
Affinity DataIC50: 1.94E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479509(CHEMBL473948)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479530(CHEMBL517571)
Affinity DataIC50: 5.25E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479514(CHEMBL454390)
Affinity DataIC50: 1.15E+4nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479515(CHEMBL455180)
Affinity DataIC50: 1.37E+4nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479534(CHEMBL455177)
Affinity DataIC50: 1.51E+4nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479523(CHEMBL461955)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetAurora kinase A(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479532(CHEMBL451034)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed