Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50038764
TargetTranslocator protein(Rat)
Brain and Mind Research Institute

Curated by ChEMBL
LigandPNGBDBM22040(Ro5-4864 | 4' Cl-diazepam | 4 -chlorodiazepam ...)
Affinity DataKd:  1.10nMAssay Description:Displacement of [3H]Ro5-4864 from TSPO in rat kainate lesioned striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Brain and Mind Research Institute

Curated by ChEMBL
LigandPNGBDBM22032(PK 11195 | PK11195 | RP 52028 | N-(butan-2-yl)-1-(...)
Affinity DataKd:  0.600nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTranslocator protein(Rat)
Brain and Mind Research Institute

Curated by ChEMBL
LigandPNGBDBM50255226(SR-180575 | (7-chloro-N,N,5-trimethyl-4-oxo-3-phen...)
Affinity DataKd:  3nMAssay Description:Displacement of [3H]SSR180575 from TSPO in rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Brain and Mind Research Institute

Curated by ChEMBL
LigandPNGBDBM50185957(N-(4-chloro-2-phenoxyphenyl)-N-(2-isopropoxybenzyl...)
Affinity DataKi:  0.920nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Brain and Mind Research Institute

Curated by ChEMBL
LigandPNGBDBM50253713(N-benzyl-2-(5-chloro-2-(4-chlorophenyl)-1H-indol-3...)
Affinity DataKi:  3.33nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat kidney membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Brain and Mind Research Institute

Curated by ChEMBL
LigandPNGBDBM50045877(2-(2-(4-fluorophenyl)-1H-indol-3-yl)-N,N-dihexylac...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Brain and Mind Research Institute

Curated by ChEMBL
LigandPNGBDBM50243007(N,N-diethyl-2-(2-(4-(2-fluoroethoxy)phenyl)-5,7-di...)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed