Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50028018
TargetIntegrin alpha-V(Human)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50265535(2-((2R,8R,11R,14S)-11-((5R,8S,11R,17R,20S,23R,26S)...)
Affinity DataIC50: 10.8nMAssay Description:Displacement of [125I]c(RGDyK) form integrin alphaVbeta3 receptor in human U87MG cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50265534(2-((2R,8R,11R,14S)-11-(4-aminobutyl)-8-(3-guanidin...)
Affinity DataIC50: 11.2nMAssay Description:Displacement of [125I]c(RGDyK) form integrin alphaVbeta3 receptor in human U87MG cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50265536(2-((2R,8R,11R,14S)-11-((5R,8S,11R,17R,20S,23R,26S)...)
Affinity DataIC50: 13.8nMAssay Description:Displacement of [125I]c(RGDyK) form integrin alphaVbeta3 receptor in human U87MG cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50265536(2-((2R,8R,11R,14S)-11-((5R,8S,11R,17R,20S,23R,26S)...)
Affinity DataIC50: 73.3nMAssay Description:Displacement of [125I][Tyr4]BBN form integrin alphaVbeta3 receptor in human PC3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50265537((S)-N1-((5R,8S,11R,17R,20S,23R)-11-((1H-imidazol-4...)
Affinity DataIC50: 79.0nMAssay Description:Displacement of [125I][Tyr4]BBN form integrin alphaVbeta3 receptor in human PC3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50265535(2-((2R,8R,11R,14S)-11-((5R,8S,11R,17R,20S,23R,26S)...)
Affinity DataIC50: 85.5nMAssay Description:Displacement of [125I][Tyr4]BBN form integrin alphaVbeta3 receptor in human PC3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed