Compile Data Set for Download or QSAR
Report error Found 44 Enz. Inhib. hit(s) with all data for entry = 3470
TargetProtein kinase C zeta type(Human)
Pfizer

LigandPNGBDBM35167(indazole-benzimidazole, 3)
Affinity DataIC50: 2.26nMpH: 7.5 T: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
LigandPNGBDBM35167(indazole-benzimidazole, 3)
Affinity DataIC50: 4.10nMT: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
LigandPNGBDBM35190(pyrazolo[3,4-b]-pyridine, 2)
Affinity DataIC50: 5nMT: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
Pfizer

LigandPNGBDBM35173(indazole-benzimidazole, 9)
Affinity DataIC50: 5.18nMpH: 7.5 T: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
Pfizer

LigandPNGBDBM35168(indazole-benzimidazole, 4)
Affinity DataIC50: 5.60nMpH: 7.5 T: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
LigandPNGBDBM35168(indazole-benzimidazole, 4)
Affinity DataIC50: 13.3nMT: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
Pfizer

LigandPNGBDBM35166(indazole-benzimidazole, 1)
Affinity DataIC50: 22nMpH: 7.5 T: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
Pfizer

LigandPNGBDBM35181(indazole-benzimidazole, 17)
Affinity DataIC50: 23.3nMpH: 7.5 T: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
Pfizer

LigandPNGBDBM35176(indazole-benzimidazole, 12)
Affinity DataIC50: 51.3nMpH: 7.5 T: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
Pfizer

LigandPNGBDBM35175(indazole-benzimidazole, 11)
Affinity DataIC50: 55.5nMpH: 7.5 T: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
LigandPNGBDBM35166(indazole-benzimidazole, 1)
Affinity DataIC50: 102nMT: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
LigandPNGBDBM35176(indazole-benzimidazole, 12)
Affinity DataIC50: 247nMT: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
Pfizer

LigandPNGBDBM35169(indazole-benzimidazole, 5)
Affinity DataIC50: 290nMpH: 7.5 T: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
Pfizer

LigandPNGBDBM35179(indazole-benzimidazole, 15)
Affinity DataIC50: 585nMpH: 7.5 T: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
LigandPNGBDBM35173(indazole-benzimidazole, 9)
Affinity DataIC50: 1.04E+3nMT: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
Pfizer

LigandPNGBDBM35188(indazole-benzimidazole, 24)
Affinity DataIC50: 1.07E+3nMpH: 7.5 T: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
Pfizer

LigandPNGBDBM35180(indazole-benzimidazole, 16)
Affinity DataIC50: 1.31E+3nMpH: 7.5 T: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
Pfizer

LigandPNGBDBM35174(indazole-benzimidazole, 10)
Affinity DataIC50: 1.51E+3nMpH: 7.5 T: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
LigandPNGBDBM35175(indazole-benzimidazole, 11)
Affinity DataIC50: 1.73E+3nMT: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
Pfizer

LigandPNGBDBM35189(indazole-benzimidazole, 25)
Affinity DataIC50: 3.02E+3nMpH: 7.5 T: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
Pfizer

LigandPNGBDBM35186(indazole-benzimidazole, 22)
Affinity DataIC50: 4.08E+3nMpH: 7.5 T: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
Pfizer

LigandPNGBDBM35171(indazole-benzimidazole, 7)
Affinity DataIC50: 5.52E+3nMpH: 7.5 T: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
LigandPNGBDBM35174(indazole-benzimidazole, 10)
Affinity DataIC50: 6.10E+3nMT: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
Pfizer

LigandPNGBDBM35187(indazole-benzimidazole, 23)
Affinity DataIC50: 6.84E+3nMpH: 7.5 T: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
Pfizer

LigandPNGBDBM35178(indazole-benzimidazole, 14)
Affinity DataIC50: 8.80E+3nMpH: 7.5 T: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
Pfizer

LigandPNGBDBM35185(indazole-benzimidazole, 21)
Affinity DataIC50: 8.93E+3nMpH: 7.5 T: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
LigandPNGBDBM35187(indazole-benzimidazole, 23)
Affinity DataIC50: 1.00E+4nMT: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
LigandPNGBDBM35186(indazole-benzimidazole, 22)
Affinity DataIC50: 1.00E+4nMT: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
LigandPNGBDBM35170(indazole-benzimidazole, 6)
Affinity DataIC50: 1.00E+4nMT: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
LigandPNGBDBM35171(indazole-benzimidazole, 7)
Affinity DataIC50: 1.00E+4nMT: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
LigandPNGBDBM35172(indazole-benzimidazole, 8)
Affinity DataIC50: 1.00E+4nMT: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
LigandPNGBDBM35183(indazole-benzimidazole, 19)
Affinity DataIC50: 1.00E+4nMT: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
LigandPNGBDBM35182(indazole-benzimidazole, 18)
Affinity DataIC50: 1.00E+4nMT: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
LigandPNGBDBM35177(indazole-benzimidazole, 13)
Affinity DataIC50: 1.00E+4nMT: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
LigandPNGBDBM35178(indazole-benzimidazole, 14)
Affinity DataIC50: 1.00E+4nMT: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
LigandPNGBDBM35181(indazole-benzimidazole, 17)
Affinity DataIC50: 1.00E+4nMT: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
Pfizer

LigandPNGBDBM35184(indazole-benzimidazole, 20)
Affinity DataIC50: 1.18E+4nMpH: 7.5 T: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
Pfizer

LigandPNGBDBM35170(indazole-benzimidazole, 6)
Affinity DataIC50: 1.24E+4nMpH: 7.5 T: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
Pfizer

LigandPNGBDBM35183(indazole-benzimidazole, 19)
Affinity DataIC50: 1.36E+4nMpH: 7.5 T: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
Pfizer

LigandPNGBDBM35172(indazole-benzimidazole, 8)
Affinity DataIC50: 1.90E+4nMpH: 7.5 T: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
LigandPNGBDBM35169(indazole-benzimidazole, 5)
Affinity DataIC50: 2.15E+4nMT: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
Pfizer

LigandPNGBDBM35182(indazole-benzimidazole, 18)
Affinity DataIC50: 2.73E+4nMpH: 7.5 T: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
Pfizer

LigandPNGBDBM35177(indazole-benzimidazole, 13)
Affinity DataIC50: 3.11E+4nMpH: 7.5 T: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed
LigandPNGBDBM35179(indazole-benzimidazole, 15)
Affinity DataIC50: 1.09E+5nMT: 2°CAssay Description:Protein kinase C (PKC), zeta activity was measured by following the phosphorylation of a biotinylated peptide substrate in the presence of ATP using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2009
Entry Details Article
PubMed