Compile Data Set for Download or QSAR
Report error Found 106 Enz. Inhib. hit(s) with all data for entry = 50035973
TargetSerotonin 2 (5-HT2) receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010041(CHEMBL84087 | {1-[3-(1,1-Dioxo-1H-1lambda*6*-napht...)
Affinity DataIC50: 0.100nMAssay Description:The concentration required to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010048(CHEMBL418929 | 2-[3-(4-Phenyl-piperidin-1-yl)-prop...)
Affinity DataIC50: 0.200nMAssay Description:The concentration required to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010049(CHEMBL79375 | 4-{4-[3-(1,1-Dioxo-1H-1lambda*6*-nap...)
Affinity DataIC50: 0.300nMAssay Description:The concentration required to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010038(CHEMBL79927 | 2-[3-(4-Benzo[d]isothiazol-3-yl-pipe...)
Affinity DataIC50: 0.400nMAssay Description:The concentration required to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010044(FANANSERIN | ChEMBL_131689 | 2-{3-[4-(4-Fluoro-phe...)
Affinity DataIC50: 0.5nMAssay Description:The concentration required to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50229423(CHEMBL82229)
Affinity DataIC50: 1nMAssay Description:The concentration required to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010040(CHEMBL83787 | 2-[3-(4-Phenyl-3,6-dihydro-2H-pyridi...)
Affinity DataIC50: 1nMAssay Description:The concentration required to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50001775(cid_5074 | Ritanserine | 6-(2-{4-[Bis-(4-fluoro-ph...)
Affinity DataIC50: 1.70nMAssay Description:The concentration required to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010052(CHEMBL440134 | 2-[4-(4-Phenyl-3,6-dihydro-2H-pyrid...)
Affinity DataIC50: 2.10nMAssay Description:The concentration required to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010033(CHEMBL418911 | 2-[3-(4-Benzo[d]isoxazol-3-yl-piper...)
Affinity DataIC50: 2.30nMAssay Description:The concentration required to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010057(CHEMBL82651 | 2-[3-(4-Phenyl-piperazin-1-yl)-propy...)
Affinity DataIC50: 2.60nMAssay Description:The concentration required to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010047(CHEMBL83975 | 2-{3-[4-(2-Fluoro-phenyl)-piperazin-...)
Affinity DataIC50: 3nMAssay Description:The concentration required to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010061(CHEMBL82826 | 2-{4-[4-(4-Fluoro-phenyl)-piperazin-...)
Affinity DataIC50: 3.70nMAssay Description:The concentration required to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010034(CHEMBL84465 | 2-[3-(4-p-Tolyl-piperazin-1-yl)-prop...)
Affinity DataIC50: 4nMAssay Description:The concentration required to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010042(CHEMBL83035 | 2-{3-[4-(4-Chloro-phenyl)-piperazin-...)
Affinity DataIC50: 5nMAssay Description:The concentration required to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010037(CHEMBL79598 | N-Naphthalen-1-yl-N-[3-(4-phenyl-3,6...)
Affinity DataIC50: 5.10nMAssay Description:The concentration required to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010055(CHEMBL316227 | 2-[3-(4-Pyridin-2-yl-piperazin-1-yl...)
Affinity DataIC50: 6.30nMAssay Description:The concentration required to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010043(CHEMBL310105 | 2-[2-(4-Phenyl-3,6-dihydro-2H-pyrid...)
Affinity DataIC50: 6.30nMAssay Description:The concentration required to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010054(CHEMBL81813 | 1-{1-[3-(1,1-Dioxo-1H-1lambda*6*-nap...)
Affinity DataIC50: 7nMAssay Description:The concentration required to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010045(CHEMBL83780 | 2-{3-[4-(4-Bromo-phenyl)-piperazin-1...)
Affinity DataIC50: 7nMAssay Description:The concentration required to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010052(CHEMBL440134 | 2-[4-(4-Phenyl-3,6-dihydro-2H-pyrid...)
Affinity DataIC50: 7.80nMAssay Description:The concentration required to inhibit [3H]prazosin binding to Alpha-1 adrenergic receptor in rat brain membranes was measured (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010041(CHEMBL84087 | {1-[3-(1,1-Dioxo-1H-1lambda*6*-napht...)
Affinity DataIC50: 7.90nMAssay Description:The concentration required to inhibit [3H]prazosin binding to Alpha-1 adrenergic receptor in rat brain membranes was measured (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010032(CHEMBL442185 | 1-[3-(4-Phenyl-3,6-dihydro-2H-pyrid...)
Affinity DataIC50: 9.80nMAssay Description:The concentration required to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010050(CHEMBL309660 | N-Phenyl-N-[3-(4-phenyl-3,6-dihydro...)
Affinity DataIC50: 10nMAssay Description:The concentration required to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010036(CHEMBL83664 | 10-[3-(4-Phenyl-3,6-dihydro-2H-pyrid...)
Affinity DataIC50: 10nMAssay Description:The concentration required to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010036(CHEMBL83664 | 10-[3-(4-Phenyl-3,6-dihydro-2H-pyrid...)
Affinity DataIC50: 10nMAssay Description:The concentration required to inhibit [3H]prazosin binding to Alpha-1 adrenergic receptor in rat brain membranes was measured (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010054(CHEMBL81813 | 1-{1-[3-(1,1-Dioxo-1H-1lambda*6*-nap...)
Affinity DataIC50: 10nMAssay Description:The concentration required to inhibit [3H]prazosin binding to Alpha-1 adrenergic receptor in rat brain membranes was measured (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010031(CHEMBL84346 | 2-(3-{4-[Bis-(4-fluoro-phenyl)-methy...)
Affinity DataIC50: 11nMAssay Description:The concentration required to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010061(CHEMBL82826 | 2-{4-[4-(4-Fluoro-phenyl)-piperazin-...)
Affinity DataIC50: 11nMAssay Description:The concentration required to inhibit 3[H]prazosin binding to Alpha-1 adrenergic receptor in rat brain membranes was measured (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010039(CHEMBL415272 | 2-{3-[4-(3-Fluoro-phenyl)-piperazin...)
Affinity DataIC50: 18nMAssay Description:The concentration required to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50001775(cid_5074 | Ritanserine | 6-(2-{4-[Bis-(4-fluoro-ph...)
Affinity DataIC50: 23nMAssay Description:The concentration required to inhibit [3H]spiperone binding to dopamine receptor D2 in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010051(CHEMBL79420 | 2-{3-[4-(4-Methoxy-phenyl)-piperazin...)
Affinity DataIC50: 25nMAssay Description:The concentration required to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010053(CHEMBL84077 | 2-{3-[4-(4-Nitro-phenyl)-piperazin-1...)
Affinity DataIC50: 25nMAssay Description:The concentration required to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010048(CHEMBL418929 | 2-[3-(4-Phenyl-piperidin-1-yl)-prop...)
Affinity DataIC50: 27nMAssay Description:The concentration required to inhibit [3H]prazosin binding to Alpha-1 adrenergic receptor in rat brain membranes was measured (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010060(CHEMBL312043 | 2-[3-(4-Pyrimidin-2-yl-piperazin-1-...)
Affinity DataIC50: 32nMAssay Description:The concentration required to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010050(CHEMBL309660 | N-Phenyl-N-[3-(4-phenyl-3,6-dihydro...)
Affinity DataIC50: 35nMAssay Description:The concentration required to inhibit [3H]prazosin binding to Alpha-1 adrenergic receptor in rat brain membranes was measured (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50001775(cid_5074 | Ritanserine | 6-(2-{4-[Bis-(4-fluoro-ph...)
Affinity DataIC50: 37nMAssay Description:The concentration required to inhibit [3H]prazosin binding to Alpha-1 adrenergic receptor in rat brain membranes was measured (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010041(CHEMBL84087 | {1-[3-(1,1-Dioxo-1H-1lambda*6*-napht...)
Affinity DataIC50: 41nMAssay Description:The concentration required to inhibit [3H]spiperone binding to dopamine receptor D2 in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010054(CHEMBL81813 | 1-{1-[3-(1,1-Dioxo-1H-1lambda*6*-nap...)
Affinity DataIC50: 46nMAssay Description:The concentration required to inhibit [3H]spiperone binding to dopamine receptor D2 in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010031(CHEMBL84346 | 2-(3-{4-[Bis-(4-fluoro-phenyl)-methy...)
Affinity DataIC50: 50nMAssay Description:The concentration required to inhibit [3H]prazosin binding to Alpha-1 adrenergic receptor in rat brain membranes was measured (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010047(CHEMBL83975 | 2-{3-[4-(2-Fluoro-phenyl)-piperazin-...)
Affinity DataIC50: 52nMAssay Description:The concentration required to inhibit [3H]prazosin binding to Alpha-1 adrenergic receptor in rat brain membranes was measured (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010052(CHEMBL440134 | 2-[4-(4-Phenyl-3,6-dihydro-2H-pyrid...)
Affinity DataIC50: 55nMAssay Description:The concentration required to inhibit [3H]spiperone binding to dopamine receptor D2 in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50229423(CHEMBL82229)
Affinity DataIC50: 64nMAssay Description:The concentration required to inhibit [3H]prazosin binding to Alpha-1 adrenergic receptor in rat brain membranes was measured (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010038(CHEMBL79927 | 2-[3-(4-Benzo[d]isothiazol-3-yl-pipe...)
Affinity DataIC50: 75nMAssay Description:The concentration required to inhibit [3H]prazosin binding to Alpha-1 adrenergic receptor in rat brain membranes was measured (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
Centre De Recherches De Vitry Alfortville Rh£Ne-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50010037(CHEMBL79598 | N-Naphthalen-1-yl-N-[3-(4-phenyl-3,6...)
Affinity DataIC50: 75nMAssay Description:The concentration required to inhibit [3H]prazosin binding to Alpha-1 adrenergic receptor in rat brain membranes was measured (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherches De Vitry Alfortville Rh£Ne-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50010050(CHEMBL309660 | N-Phenyl-N-[3-(4-phenyl-3,6-dihydro...)
Affinity DataIC50: 80nMAssay Description:The concentration required to inhibit [3H]spiperone binding to dopamine receptor D2 in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50010043(CHEMBL310105 | 2-[2-(4-Phenyl-3,6-dihydro-2H-pyrid...)
Affinity DataIC50: 98nMAssay Description:The concentration required to inhibit [3H]prazosin binding to Alpha-1 adrenergic receptor in rat brain membranes was measured (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Centre De Recherches De Vitry Alfortville Rh£Ne-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50229428(CHEMBL310902)
Affinity DataIC50: 100nMAssay Description:The concentration required to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherches De Vitry Alfortville Rh£Ne-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50010032(CHEMBL442185 | 1-[3-(4-Phenyl-3,6-dihydro-2H-pyrid...)
Affinity DataIC50: 100nMAssay Description:The concentration required to inhibit [3H]spiperone binding to dopamine receptor D2 in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherches De Vitry Alfortville Rh£Ne-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50010043(CHEMBL310105 | 2-[2-(4-Phenyl-3,6-dihydro-2H-pyrid...)
Affinity DataIC50: 100nMAssay Description:The concentration required to inhibit [3H]spiperone binding to dopamine receptor D2 in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
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