Report error Found 114 Enz. Inhib. hit(s) with all data for entry = 50027806
Affinity DataIC50: 80nMAssay Description:Inhibition of ABCB1-mediated [3H]vinblastine transportation in human Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibition of ABCB1 transfected in MDCK cells assessed as increase in calcein-AM accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of ABCB1 transfected in MDCK cells assessed as increase in calcein-AM accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Inhibition of ABCB1-mediated [3H]vinblastine transportation in human Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibition of ABCB1-mediated [3H]vinblastine transportation in human Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibition of ABCB1 transfected in MDCK cells assessed as increase in calcein-AM accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Inhibition of ABCB1-mediated [3H]vinblastine transportation in human Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of ABCB1-mediated [3H]vinblastine transportation in human Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 350nMAssay Description:Inhibition of ABCB1-mediated [3H]vinblastine transportation in human Caco-2 cellsMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Universita Degli Studi Di Bari
Curated by ChEMBL
Universita Degli Studi Di Bari
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of ABCB1-mediated [3H]vinblastine transportation in human Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 750nMAssay Description:Inhibition of ABCB1-mediated [3H]vinblastine transportation in human Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 750nMAssay Description:Inhibition of ABCB1-mediated [3H]vinblastine transportation in human Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 780nMAssay Description:Inhibition of ABCB1 transfected in MDCK cells assessed as increase in calcein-AM accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Inhibition of ABCB1-mediated [3H]vinblastine transportation in human Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.14E+3nMAssay Description:Inhibition of ABCB1 transfected in MDCK cells assessed as increase in calcein-AM accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.17E+3nMAssay Description:Inhibition of ABCB1 transfected in MDCK cells assessed as increase in calcein-AM accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of ABCB1-mediated [3H]vinblastine transportation in human Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of ABCB1-mediated [3H]vinblastine transportation in human Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.27E+3nMAssay Description:Inhibition of ABCB1-mediated [3H]vinblastine transportation in human Caco-2 cellsMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Universita Degli Studi Di Bari
Curated by ChEMBL
Universita Degli Studi Di Bari
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of ABCG2More data for this Ligand-Target Pair
Affinity DataIC50: 1.72E+3nMAssay Description:Inhibition of ABCB1-mediated [3H]vinblastine transportation in human Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.78E+3nMAssay Description:Inhibition of ABCB1 transfected in MDCK cells assessed as increase in calcein-AM accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.79E+3nMAssay Description:Inhibition of ABCB1 transfected in MDCK cells assessed as increase in calcein-AM accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of ABCB1-mediated [3H]vinblastine transportation in human Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of ABCB1-mediated [3H]vinblastine transportation in human Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of ABCB1-mediated [3H]vinblastine transportation in human Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.12E+3nMAssay Description:Inhibition of ABCB1-mediated [3H]vinblastine transportation in human Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of ABCB1-mediated [3H]vinblastine transportation in human Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of ABCB1-mediated [3H]vinblastine transportation in human Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.65E+3nMAssay Description:Inhibition of ABCB1-mediated [3H]vinblastine transportation in human Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.17E+3nMAssay Description:Inhibition of ABCB1-mediated [3H]vinblastine transportation in human Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of ABCB1-mediated [3H]vinblastine transportation in human Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 4.78E+3nMAssay Description:Inhibition of ABCB1 transfected in MDCK cells assessed as increase in calcein-AM accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of ABCB1-mediated [3H]vinblastine transportation in human Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of ABCB1-mediated [3H]vinblastine transportation in human Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of ABCB1-mediated [3H]vinblastine transportation in human Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 6.82E+3nMAssay Description:Inhibition of ABCB1-mediated [3H]vinblastine transportation in human Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 7.76E+3nMAssay Description:Inhibition of ABCB1 transfected in MDCK cells assessed as increase in calcein-AM accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of ABCB1-mediated [3H]vinblastine transportation in human Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of ABCB1-mediated [3H]vinblastine transportation in human Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of ABCB1-mediated [3H]vinblastine transportation in human Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of ABCB1-mediated [3H]vinblastine transportation in human Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of ABCB1-mediated [3H]vinblastine transportation in human Caco-2 cellsMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Universita Degli Studi Di Bari
Curated by ChEMBL
Universita Degli Studi Di Bari
Curated by ChEMBL
Affinity DataIC50: 1.20E+5nMAssay Description:Inhibition of ABCG2More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Universita Degli Studi Di Bari
Curated by ChEMBL
Universita Degli Studi Di Bari
Curated by ChEMBL
Affinity DataIC50: 1.50E+5nMAssay Description:Inhibition of ABCG2More data for this Ligand-Target Pair





















3D Structure (crystal)













