Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50027802
TargetSecreted frizzled-related protein 1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50247135(2-methyl-N-phenethyl-5-(phenylsulfonyl)benzenesulf...)
Affinity DataEC50:  3.88E+3nMAssay Description:Inhibition of human sFRP1 expressed in human U2OS assessed as luciferase activity by TCF-luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSecreted frizzled-related protein 1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50246651(N-[2-(3,4-Dimethoxyphenyl)ethyl]-2-ethyl-5-(phenyl...)
Affinity DataEC50:  6.97E+3nMAssay Description:Inhibition of human sFRP1 expressed in human U2OS assessed as luciferase activity by TCF-luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSecreted frizzled-related protein 1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50246617(2-Ethyl-5-(phenylsulfonyl)-N-(3-pyrrolidin-1-ylpro...)
Affinity DataEC50:  9.00E+3nMAssay Description:Inhibition of human sFRP1 expressed in human U2OS assessed as luciferase activity by TCF-luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSecreted frizzled-related protein 1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50246616(N-[3-(Dimethylamino)propyl]-2-ethyl-5-(phenylsulfo...)
Affinity DataEC50:  1.27E+3nMAssay Description:Inhibition of human sFRP1 expressed in human U2OS assessed as luciferase activity by TCF-luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSecreted frizzled-related protein 1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50247135(2-methyl-N-phenethyl-5-(phenylsulfonyl)benzenesulf...)
Affinity DataKd:  350nMAssay Description:Binding affinity to human sFRP1 by fluorescence spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed