Compile Data Set for Download or QSAR
Report error Found 128 Enz. Inhib. hit(s) with all data for entry = 50027725
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50253952(3-{(S)-3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-[3-(...)
Affinity DataKi:  0.0800nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM104908(CHEMBL468270 | US8569313, Inhibitor 16)
Affinity DataKi:  1nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254410(3-{(S)-3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-[3-(...)
Affinity DataKi:  1.60nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254368((+/-)-3-[3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-(4...)
Affinity DataKi:  2.5nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254219(US8569313, 71 | CHEMBL461870 | Azetidine-3-carboxy...)
Affinity DataKi:  3nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM23917(3-amino-N-(3-{[(2S)-1-[4-(2-aminoethyl)piperidin-1...)
Affinity DataKi:  3.80nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254367((+/-)-3-[3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-(3...)
Affinity DataKi:  5.40nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254365((+/-)-3-[3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-(4...)
Affinity DataKi:  6nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254218(3-{(S)-3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-[3-(...)
Affinity DataKi:  6.70nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254364((+/-)-3-[3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-(4...)
Affinity DataKi:  7nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50253952(3-{(S)-3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-[3-(...)
Affinity DataKi:  10nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254314((+/-)-3-[3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-(4...)
Affinity DataKi:  10nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254312((+/-)-3-[3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-(2...)
Affinity DataKi:  11nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254366((+/-)-3-[3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-(4...)
Affinity DataKi:  12nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254409((+/-)-3-{3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-[3...)
Affinity DataKi:  13nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254314((+/-)-3-[3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-(4...)
Affinity DataKi:  26nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPlasminogen(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50253952(3-{(S)-3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-[3-(...)
Affinity DataKi:  28nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50253953(CHEMBL513007 | US8569313, 20 | 3-{(S)-3-[4-(2-Amin...)
Affinity DataKi:  28nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254312((+/-)-3-[3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-(2...)
Affinity DataKi:  29nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254368((+/-)-3-[3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-(4...)
Affinity DataKi:  33nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254364((+/-)-3-[3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-(4...)
Affinity DataKi:  40nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254275({3-[(S)-2-[4-(2-Amino-ethyl)-piperidin-1-yl]-1-(3-...)
Affinity DataKi:  41nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254408((+/-)-3-[3-[4-(2-Amino-ethyl)-piperidin-1-yl]-3-ox...)
Affinity DataKi:  47nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254313((+/-)-3-[3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-(3...)
Affinity DataKi:  51nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50253954(CHEMBL459525 | US8569313, 61 | 3-Amino-N-{3-[(S)-2...)
Affinity DataKi:  56nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254276((+/-)-3-[3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-(b...)
Affinity DataKi:  56nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254407((+/-)-3-[3-[4-(2-Amino-ethyl)-piperidin-1-yl]-3-ox...)
Affinity DataKi:  60nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPlasminogen(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254366((+/-)-3-[3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-(4...)
Affinity DataKi:  80nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPlasminogen(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254312((+/-)-3-[3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-(2...)
Affinity DataKi:  85nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254313((+/-)-3-[3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-(3...)
Affinity DataKi:  91nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254410(3-{(S)-3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-[3-(...)
Affinity DataKi:  110nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254276((+/-)-3-[3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-(b...)
Affinity DataKi:  110nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPlasminogen(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254407((+/-)-3-[3-[4-(2-Amino-ethyl)-piperidin-1-yl]-3-ox...)
Affinity DataKi:  110nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254220(US8569313, 68 | CHEMBL513339 | N-{3-[(S)-2-[4-(2-A...)
Affinity DataKi:  120nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPlasminogen(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254364((+/-)-3-[3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-(4...)
Affinity DataKi:  120nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254024((+/-)-4'-Methoxy-biphenyl-3-sulfonic acid [2-[4-(2...)
Affinity DataKi:  145nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254408((+/-)-3-[3-[4-(2-Amino-ethyl)-piperidin-1-yl]-3-ox...)
Affinity DataKi:  150nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254409((+/-)-3-{3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-[3...)
Affinity DataKi:  150nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPlasminogen(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254365((+/-)-3-[3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-(4...)
Affinity DataKi:  150nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254407((+/-)-3-[3-[4-(2-Amino-ethyl)-piperidin-1-yl]-3-ox...)
Affinity DataKi:  160nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254274(N-{3-[(S)-2-[4-(2-Amino-ethyl)-piperidin-1-yl]-1-(...)
Affinity DataKi:  180nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPlasminogen(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254314((+/-)-3-[3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-(4...)
Affinity DataKi:  183nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254409((+/-)-3-{3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-[3...)
Affinity DataKi:  190nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPlasminogen(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM104908(CHEMBL468270 | US8569313, Inhibitor 16)
Affinity DataKi:  200nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPlasminogen(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50253953(CHEMBL513007 | US8569313, 20 | 3-{(S)-3-[4-(2-Amin...)
Affinity DataKi:  210nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPlasminogen(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254368((+/-)-3-[3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-(4...)
Affinity DataKi:  214nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPlasminogen(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254410(3-{(S)-3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-[3-(...)
Affinity DataKi:  230nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPlasminogen(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254367((+/-)-3-[3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-(3...)
Affinity DataKi:  230nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254366((+/-)-3-[3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-(4...)
Affinity DataKi:  240nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254410(3-{(S)-3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-[3-(...)
Affinity DataKi:  250nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
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