Compile Data Set for Download or QSAR
Report error Found 54 Enz. Inhib. hit(s) with all data for entry = 50027531
TargetThyroid hormone receptor beta(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM18869(2-{3,5-dichloro-4-[4-hydroxy-3-(propan-2-yl)phenox...)
Affinity DataKi:  0.240nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetThyroid hormone receptor beta(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50115668([4-(4-Hydroxy-3-isopropyl-benzyl)-3,5-dimethyl-phe...)
Affinity DataKi:  0.320nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetThyroid hormone receptor alpha(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM18860(triothyrone | (2S)-2-amino-3-[4-(4-hydroxy-3-iodop...)
Affinity DataKi:  0.330nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine from His-tagged human recombinant TRalpha1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50036402(N-[3,5-dimethyl-4-(4'-hydroxy-3'-isopropylphenoxy)...)
Affinity DataKi:  0.470nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50036402(N-[3,5-dimethyl-4-(4'-hydroxy-3'-isopropylphenoxy)...)
Affinity DataKi:  0.510nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine from His-tagged human recombinant TRalpha1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM18860(triothyrone | (2S)-2-amino-3-[4-(4-hydroxy-3-iodop...)
Affinity DataKi:  0.680nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50274809(3,5-Diiodo-4-(4'-hydroxy-3'-isopropylphenoxy)benzy...)
Affinity DataKi:  0.840nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50274812([3,5-Diiodo-4-(4'-hydroxy-3'-isopropylphenoxy)phen...)
Affinity DataKi:  0.970nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50115668([4-(4-Hydroxy-3-isopropyl-benzyl)-3,5-dimethyl-phe...)
Affinity DataKi:  1.09nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine from His-tagged human recombinant TRalpha1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetThyroid hormone receptor beta(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50274846([3,5-Dibromo-4-(4'-hydroxy-3'-isopropylphenoxy)phe...)
Affinity DataKi:  1.51nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50274809(3,5-Diiodo-4-(4'-hydroxy-3'-isopropylphenoxy)benzy...)
Affinity DataKi:  1.84nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine from His-tagged human recombinant TRalpha1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50275295(2-[3,5-Dibromo-4-(4'-hydroxy-3'-isopropylphenoxy)p...)
Affinity DataKi:  2.5nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50274811([3,5-Dibromo-4-(4'-hydroxy-3'-isopropylphenoxy)phe...)
Affinity DataKi:  2.51nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50242403([3,5-Dimethyl-4-(4'-hydroxy-3'-isopropylbenzyl)phe...)
Affinity DataKi:  2.95nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50274812([3,5-Diiodo-4-(4'-hydroxy-3'-isopropylphenoxy)phen...)
Affinity DataKi:  3.74nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine from His-tagged human recombinant TRalpha1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50275257([3,5-Dimethyl-4-(3'-sec-butyl-4'-hydroxybenzyl)phe...)
Affinity DataKi:  6.64nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM18869(2-{3,5-dichloro-4-[4-hydroxy-3-(propan-2-yl)phenox...)
Affinity DataKi:  7.79nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine from His-tagged human recombinant TRalpha1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetThyroid hormone receptor beta(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50275291([4-(4'-Hydroxy-3'-isopropylbenzyl)-3,5-dimethylphe...)
Affinity DataKi:  9.10nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50275228([3,5-Dimethyl-4-(3'-ethyl-4'-hydroxybenzyl)phenoxy...)
Affinity DataKi:  9.72nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50274846([3,5-Dibromo-4-(4'-hydroxy-3'-isopropylphenoxy)phe...)
Affinity DataKi:  10.3nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine from His-tagged human recombinant TRalpha1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50275294([3,5-Dibromo-4-(4'-hydroxy-3'-isopropylphenoxy)]be...)
Affinity DataKi:  15.5nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50274810(3,5-Diiodo-4-(4'-hydroxy-3'-iodophenoxy)benzylphos...)
Affinity DataKi:  16nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine from His-tagged human recombinant TRalpha1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50274811([3,5-Dibromo-4-(4'-hydroxy-3'-isopropylphenoxy)phe...)
Affinity DataKi:  18.6nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine from His-tagged human recombinant TRalpha1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50274813([3,5-Dimethyl-4-(4'-hydroxy-3'-isopropylphenoxy)ph...)
Affinity DataKi:  25.4nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50274810(3,5-Diiodo-4-(4'-hydroxy-3'-iodophenoxy)benzylphos...)
Affinity DataKi:  26nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50275291([4-(4'-Hydroxy-3'-isopropylbenzyl)-3,5-dimethylphe...)
Affinity DataKi:  28.4nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine from His-tagged human recombinant TRalpha1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50274814([3,5-Dichloro-4-(4'-hydroxy-3'-isopropylphenoxy)ph...)
Affinity DataKi:  30.5nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50275257([3,5-Dimethyl-4-(3'-sec-butyl-4'-hydroxybenzyl)phe...)
Affinity DataKi:  30.5nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine from His-tagged human recombinant TRalpha1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50275290(2-[3,5-Dimethoxy-4-(4'-hydroxy-3'-isopropylbenzyl)...)
Affinity DataKi:  31.3nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50242403([3,5-Dimethyl-4-(4'-hydroxy-3'-isopropylbenzyl)phe...)
Affinity DataKi:  35.2nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine from His-tagged human recombinant TRalpha1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50275226(N-[3,5-Dimethyl-4-(3'-isopropyl-4'-methoxyphenoxy)...)
Affinity DataKi:  36nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50275295(2-[3,5-Dibromo-4-(4'-hydroxy-3'-isopropylphenoxy)p...)
Affinity DataKi:  42.1nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine from His-tagged human recombinant TRalpha1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50275005([4-(4'-Hydroxy-3'-isopropylphenoxy)-3,5-dimethylph...)
Affinity DataKi:  42.1nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50275293([3,5-Dichloro-4-(4'-hydroxy-3'-isopropylphenoxy)]b...)
Affinity DataKi:  52.3nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50275228([3,5-Dimethyl-4-(3'-ethyl-4'-hydroxybenzyl)phenoxy...)
Affinity DataKi:  61.6nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine from His-tagged human recombinant TRalpha1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50275259([3,5-Dimethoxy-4-(4'-hydroxy-3'-isopropylbenzyl)ph...)
Affinity DataKi:  87nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50275227([3,5-Dimethyl-4-(4'-hydroxy-3'-methylbenzyl)phenox...)
Affinity DataKi:  89.7nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50275256([3,5-Dimethyl-4-(4'-hydroxy-3'-phenylbenzyl)phenox...)
Affinity DataKi:  106nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50275292([3,5-Dimethyl-4-(4'-hydroxy-3'-isopropylphenoxy)]b...)
Affinity DataKi:  128nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50275005([4-(4'-Hydroxy-3'-isopropylphenoxy)-3,5-dimethylph...)
Affinity DataKi:  143nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine from His-tagged human recombinant TRalpha1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50275258([3,5-Dimethoxy-4-(4'-hydroxy-3'-isopropylbenzyl)ph...)
Affinity DataKi:  146nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50274813([3,5-Dimethyl-4-(4'-hydroxy-3'-isopropylphenoxy)ph...)
Affinity DataKi:  183nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine from His-tagged human recombinant TRalpha1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50274814([3,5-Dichloro-4-(4'-hydroxy-3'-isopropylphenoxy)ph...)
Affinity DataKi:  186nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine from His-tagged human recombinant TRalpha1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50275294([3,5-Dibromo-4-(4'-hydroxy-3'-isopropylphenoxy)]be...)
Affinity DataKi:  235nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine from His-tagged human recombinant TRalpha1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50275225(1-Amino-2-[3,5-diiodo-4-(4'-hydroxy-3'-iodophenoxy...)
Affinity DataKi:  271nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50275226(N-[3,5-Dimethyl-4-(3'-isopropyl-4'-methoxyphenoxy)...)
Affinity DataKi:  285nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine from His-tagged human recombinant TRalpha1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50275293([3,5-Dichloro-4-(4'-hydroxy-3'-isopropylphenoxy)]b...)
Affinity DataKi:  303nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine from His-tagged human recombinant TRalpha1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50275290(2-[3,5-Dimethoxy-4-(4'-hydroxy-3'-isopropylbenzyl)...)
Affinity DataKi:  378nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine from His-tagged human recombinant TRalpha1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50275259([3,5-Dimethoxy-4-(4'-hydroxy-3'-isopropylbenzyl)ph...)
Affinity DataKi:  594nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine from His-tagged human recombinant TRalpha1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50275227([3,5-Dimethyl-4-(4'-hydroxy-3'-methylbenzyl)phenox...)
Affinity DataKi:  897nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine from His-tagged human recombinant TRalpha1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
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