Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50000772
TargetKappa-type opioid receptor(Guinea pig)
Case Western Reserve University

Curated by ChEMBL
LigandPNGBDBM224024(Dynorphin A (1-13) | YGGFLRRXRPKLK | BDBM50241435)
Affinity DataKi:  3.60nMAssay Description:The compound was tested for binding activity towards opioid receptor kappa in guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Case Western Reserve University

Curated by ChEMBL
LigandPNGBDBM224024(Dynorphin A (1-13) | YGGFLRRXRPKLK | BDBM50241435)
Affinity DataKi:  16nMAssay Description:The compound was tested for binding activity towards Opioid receptor delta 1 in guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Case Western Reserve University

Curated by ChEMBL
LigandPNGBDBM224024(Dynorphin A (1-13) | YGGFLRRXRPKLK | BDBM50241435)
Affinity DataKi:  50nMAssay Description:The compound was tested for binding activity towards opioid receptor mu in guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Case Western Reserve University

Curated by ChEMBL
LigandPNGBDBM50009674(4-Amino-N-[2-(4-amino-butyrylamino)-ethyl]-N-[2-((...)
Affinity DataKi:  3.73E+3nMAssay Description:The compound was tested for binding activity towards opioid receptor kappa in guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Case Western Reserve University

Curated by ChEMBL
LigandPNGBDBM50009677(CHEMBL94792 | 4-Amino-N-[3-(4-amino-butyrylamino)-...)
Affinity DataKi:  5.51E+3nMAssay Description:The compound was tested for binding activity towards opioid receptor kappa in guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Case Western Reserve University

Curated by ChEMBL
LigandPNGBDBM50009674(4-Amino-N-[2-(4-amino-butyrylamino)-ethyl]-N-[2-((...)
Affinity DataKi:  6.76E+3nMAssay Description:The compound was tested for binding activity towards opioid receptor mu in guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Case Western Reserve University

Curated by ChEMBL
LigandPNGBDBM50009677(CHEMBL94792 | 4-Amino-N-[3-(4-amino-butyrylamino)-...)
Affinity DataKi:  7.30E+3nMAssay Description:The compound was tested for binding activity towards opioid receptor mu in guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Case Western Reserve University

Curated by ChEMBL
LigandPNGBDBM50009677(CHEMBL94792 | 4-Amino-N-[3-(4-amino-butyrylamino)-...)
Affinity DataKi:  8.43E+3nMAssay Description:The compound was tested for binding activity towards Opioid receptor delta 1 in guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Case Western Reserve University

Curated by ChEMBL
LigandPNGBDBM50009678(CHEMBL98014 | 4-Amino-N-[2-(4-amino-butyrylamino)-...)
Affinity DataKi:  8.75E+3nMAssay Description:The compound was tested for binding activity towards opioid receptor kappa in guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Case Western Reserve University

Curated by ChEMBL
LigandPNGBDBM50009674(4-Amino-N-[2-(4-amino-butyrylamino)-ethyl]-N-[2-((...)
Affinity DataKi: >1.00E+4nMAssay Description:The compound was tested for binding activity towards Opioid receptor delta 1 in guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Case Western Reserve University

Curated by ChEMBL
LigandPNGBDBM50009676(CHEMBL412591 | 4-Amino-N-{2-[2-(2-{2-[2-amino-3-(4...)
Affinity DataKi:  1.01E+4nMAssay Description:The compound was tested for binding activity towards Opioid receptor delta 1 in guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Case Western Reserve University

Curated by ChEMBL
LigandPNGBDBM50009678(CHEMBL98014 | 4-Amino-N-[2-(4-amino-butyrylamino)-...)
Affinity DataKi:  1.44E+4nMAssay Description:The compound was tested for binding activity towards opioid receptor mu in guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Case Western Reserve University

Curated by ChEMBL
LigandPNGBDBM50009676(CHEMBL412591 | 4-Amino-N-{2-[2-(2-{2-[2-amino-3-(4...)
Affinity DataKi:  1.65E+4nMAssay Description:The compound was tested for binding activity towards opioid receptor mu in guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Case Western Reserve University

Curated by ChEMBL
LigandPNGBDBM50009678(CHEMBL98014 | 4-Amino-N-[2-(4-amino-butyrylamino)-...)
Affinity DataKi:  2.27E+4nMAssay Description:The compound was tested for binding activity towards Opioid receptor delta 1 in guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Case Western Reserve University

Curated by ChEMBL
LigandPNGBDBM50009676(CHEMBL412591 | 4-Amino-N-{2-[2-(2-{2-[2-amino-3-(4...)
Affinity DataKi:  3.67E+4nMAssay Description:The compound was tested for binding activity towards opioid receptor kappa in guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed