Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50027465
TargetGlucagon-like peptide 1 receptor(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50152769(GLP-1(7-36)-NH2 | NH2-HAEGTFTSDVSSYLEGQAAKEFIAWLVK...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human GLP1R expressed in CHO cells assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50275523(CHEMBL500187)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human GLP1R expressed in CHO cells assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50275524(CHEMBL499397)
Affinity DataEC50:  375nMAssay Description:Agonist activity at human GLP1R expressed in CHO cells assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50275522(CHEMBL525224)
Affinity DataEC50:  73nMAssay Description:Agonist activity at human GLP1R expressed in CHO cells assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50275527(CHEMBL524875)
Affinity DataEC50:  3.60nMAssay Description:Agonist activity at human GLP1R expressed in CHO cells assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50275528(CHEMBL525608)
Affinity DataEC50:  2.40nMAssay Description:Agonist activity at human GLP1R expressed in CHO cells assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50275525(CHEMBL527058)
Affinity DataEC50:  67nMAssay Description:Agonist activity at human GLP1R expressed in CHO cells assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50275526(CHEMBL506368)
Affinity DataEC50:  5.40nMAssay Description:Agonist activity at human GLP1R expressed in CHO cells assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50152769(GLP-1(7-36)-NH2 | NH2-HAEGTFTSDVSSYLEGQAAKEFIAWLVK...)
Affinity DataIC50: 1.90nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50275523(CHEMBL500187)
Affinity DataIC50: 5.10nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50275527(CHEMBL524875)
Affinity DataIC50: 13nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50275526(CHEMBL506368)
Affinity DataIC50: 19nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50275522(CHEMBL525224)
Affinity DataIC50: 52nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50275528(CHEMBL525608)
Affinity DataIC50: 57nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50275524(CHEMBL499397)
Affinity DataIC50: 107nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50275525(CHEMBL527058)
Affinity DataIC50: 113nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed