Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 3277
LigandPNGBDBM30322(Pyrrolo-pyrimidone, 15)
Affinity DataIC50: 42nMpH: 7.5 T: 2°CAssay Description:For MK2 inhibition, reactions contained compound or vehicle control, hsp27 peptide substrate and activated MK2 mix containing ATP. After incubation, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2009
Entry Details Article
PubMed
LigandPNGBDBM30323(Pyrrolo-pyrimidone, 16)
Affinity DataIC50: 51nMpH: 7.5 T: 2°CAssay Description:For MK2 inhibition, reactions contained compound or vehicle control, hsp27 peptide substrate and activated MK2 mix containing ATP. After incubation, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2009
Entry Details Article
PubMed
LigandPNGBDBM30324(Pyrrolo-pyrimidone, 17)
Affinity DataIC50: 82nMpH: 7.5 T: 2°CAssay Description:For MK2 inhibition, reactions contained compound or vehicle control, hsp27 peptide substrate and activated MK2 mix containing ATP. After incubation, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2009
Entry Details Article
PubMed
LigandPNGBDBM30325(Pyrrolo-pyrimidone, 18)
Affinity DataIC50: 150nMpH: 7.5 T: 2°CAssay Description:For MK2 inhibition, reactions contained compound or vehicle control, hsp27 peptide substrate and activated MK2 mix containing ATP. After incubation, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2009
Entry Details Article
PubMed
LigandPNGBDBM30315(Pyrrolo-pyrimidone, 8)
Affinity DataIC50: 170nMpH: 7.5 T: 2°CAssay Description:For MK2 inhibition, reactions contained compound or vehicle control, hsp27 peptide substrate and activated MK2 mix containing ATP. After incubation, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2009
Entry Details Article
PubMed
LigandPNGBDBM30314(Pyrrolo-pyrimidone, 7)
Affinity DataIC50: 190nMpH: 7.5 T: 2°CAssay Description:For MK2 inhibition, reactions contained compound or vehicle control, hsp27 peptide substrate and activated MK2 mix containing ATP. After incubation, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2009
Entry Details Article
PubMed
LigandPNGBDBM30316(Pyrrolo-pyrimidone, 9)
Affinity DataIC50: 200nMpH: 7.5 T: 2°CAssay Description:For MK2 inhibition, reactions contained compound or vehicle control, hsp27 peptide substrate and activated MK2 mix containing ATP. After incubation, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2009
Entry Details Article
PubMed
LigandPNGBDBM30317(Pyrrolo-pyrimidone, 10)
Affinity DataIC50: 290nMpH: 7.5 T: 2°CAssay Description:For MK2 inhibition, reactions contained compound or vehicle control, hsp27 peptide substrate and activated MK2 mix containing ATP. After incubation, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2009
Entry Details Article
PubMed
LigandPNGBDBM30321(Pyrrolo-pyrimidone, 14)
Affinity DataIC50: 340nMpH: 7.5 T: 2°CAssay Description:For MK2 inhibition, reactions contained compound or vehicle control, hsp27 peptide substrate and activated MK2 mix containing ATP. After incubation, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2009
Entry Details Article
PubMed
LigandPNGBDBM30319(Pyrrolo-pyrimidone, 12)
Affinity DataIC50: 350nMpH: 7.5 T: 2°CAssay Description:For MK2 inhibition, reactions contained compound or vehicle control, hsp27 peptide substrate and activated MK2 mix containing ATP. After incubation, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2009
Entry Details Article
PubMed
LigandPNGBDBM30311(Pyrrolo-pyrimidone, 4)
Affinity DataIC50: 550nMpH: 7.5 T: 2°CAssay Description:For MK2 inhibition, reactions contained compound or vehicle control, hsp27 peptide substrate and activated MK2 mix containing ATP. After incubation, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2009
Entry Details Article
PubMed
LigandPNGBDBM30310(Pyrrolo-pyrimidone, 3)
Affinity DataIC50: 1.23E+3nMpH: 7.5 T: 2°CAssay Description:For MK2 inhibition, reactions contained compound or vehicle control, hsp27 peptide substrate and activated MK2 mix containing ATP. After incubation, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2009
Entry Details Article
PubMed
LigandPNGBDBM30320(Pyrrolo-pyrimidone, 13)
Affinity DataIC50: 1.26E+3nMpH: 7.5 T: 2°CAssay Description:For MK2 inhibition, reactions contained compound or vehicle control, hsp27 peptide substrate and activated MK2 mix containing ATP. After incubation, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2009
Entry Details Article
PubMed
LigandPNGBDBM30309(Pyrrolo-pyrimidone, 2)
Affinity DataIC50: 1.30E+3nMpH: 7.5 T: 2°CAssay Description:For MK2 inhibition, reactions contained compound or vehicle control, hsp27 peptide substrate and activated MK2 mix containing ATP. After incubation, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2009
Entry Details Article
PubMed
LigandPNGBDBM30313(Pyrrolo-pyrimidone, 6)
Affinity DataIC50: 1.45E+3nMpH: 7.5 T: 2°CAssay Description:For MK2 inhibition, reactions contained compound or vehicle control, hsp27 peptide substrate and activated MK2 mix containing ATP. After incubation, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2009
Entry Details Article
PubMed
LigandPNGBDBM30318(Pyrrolo-pyrimidone, 11)
Affinity DataIC50: 1.70E+3nMpH: 7.5 T: 2°CAssay Description:For MK2 inhibition, reactions contained compound or vehicle control, hsp27 peptide substrate and activated MK2 mix containing ATP. After incubation, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2009
Entry Details Article
PubMed
LigandPNGBDBM30312(Pyrrolo-pyrimidone, 5)
Affinity DataIC50: 5.20E+3nMpH: 7.5 T: 2°CAssay Description:For MK2 inhibition, reactions contained compound or vehicle control, hsp27 peptide substrate and activated MK2 mix containing ATP. After incubation, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2009
Entry Details Article
PubMed