Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50030261
TargetGlycogen synthase kinase-3 beta(Human)
Sterling Road

Curated by ChEMBL
LigandPNGBDBM50293306(3-(5-methoxybenzofuran-7-yl)-4-(1-(2-(4-methylpipe...)
Affinity DataIC50: 0.140nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sterling Road

Curated by ChEMBL
LigandPNGBDBM50150699(3-(9-fluoro-2-(piperidine-1-carbonyl)-1,2,3,4-tetr...)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sterling Road

Curated by ChEMBL
LigandPNGBDBM50150701(7-(4-Imidazo[1,2-a]pyridin-3-yl-2,5-dioxo-2,5-dihy...)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sterling Road

Curated by ChEMBL
LigandPNGBDBM50293307(N-(4-(ethylsulfonamido)phenethyl)-2-(2-chloro-4-fl...)
Affinity DataIC50: 2nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sterling Road

Curated by ChEMBL
LigandPNGBDBM3175(Bisindolylmaleimide 11b | Ro 31-8220 | CHEMBL6291 ...)
Affinity DataIC50: 2.80nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sterling Road

Curated by ChEMBL
LigandPNGBDBM8579(N-[6-(pyridin-3-yl)furo[2,3-d]pyrimidin-4-yl]cyclo...)
Affinity DataIC50: 5nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sterling Road

Curated by ChEMBL
LigandPNGBDBM50132317(17,23-dimethyl-20-oxa-4,14,17,23,26-pentaazahexacy...)
Affinity DataIC50: 6nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sterling Road

Curated by ChEMBL
LigandPNGBDBM50293308(3-(2,5-dichlorophenyl)-4-(1-methyl-1H-indol-3-yl)-...)
Affinity DataIC50: 7nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sterling Road

Curated by ChEMBL
LigandPNGBDBM7492(3-[(2Z,3E)-3-(hydroxyimino)-2,3-dihydro-1H-indol-2...)
Affinity DataIC50: 9nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sterling Road

Curated by ChEMBL
LigandPNGBDBM7491(4-[2-Amino-5-oxo-1,5-dihydro-imidazol-(4Z)-ylidene...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sterling Road

Curated by ChEMBL
LigandPNGBDBM50059889(3-methoxy-2-methyl-4-methylamino-(2S,3S,4S,6R)-29-...)
Affinity DataIC50: 15nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sterling Road

Curated by ChEMBL
LigandPNGBDBM7393(Indirubin-3 -monoxime | 3-[(2Z,3E)-3-(hydroxyimino...)
Affinity DataIC50: 22nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sterling Road

Curated by ChEMBL
LigandPNGBDBM50293309(N-(4-(ethylsulfonamido)phenethyl)-2-(2,4-dichlorop...)
Affinity DataIC50: 30nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sterling Road

Curated by ChEMBL
LigandPNGBDBM8296(CHEMBL102714 | cid_176158 | 3-(2,4-dichlorophenyl)...)
Affinity DataIC50: 34nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sterling Road

Curated by ChEMBL
LigandPNGBDBM50293310(6-(2-(butylamino)pyrimidin-4-yl)-3-oxo-N-(3-(pyrid...)
Affinity DataIC50: 36nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sterling Road

Curated by ChEMBL
LigandPNGBDBM50293311(N-(4-chlorobenzyl)-6-(3-fluoro-4-hydroxyphenyl)-3-...)
Affinity DataIC50: 39nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sterling Road

Curated by ChEMBL
LigandPNGBDBM50293312(N-(4-(2-morpholinoacetamido)phenethyl)-2-(4-fluoro...)
Affinity DataIC50: 40nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sterling Road

Curated by ChEMBL
LigandPNGBDBM50293313(N-(2,4-difluorobenzyl)-3-oxo-6-(pyridin-4-yl)-2,3-...)
Affinity DataIC50: 65nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sterling Road

Curated by ChEMBL
LigandPNGBDBM50130725(SB-415286 | cid_4210951 | 3-(3-chloro-4-hydroxyphe...)
Affinity DataIC50: 78nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sterling Road

Curated by ChEMBL
LigandPNGBDBM50293314(2-(2,4-dichlorophenyl)-7-hydroxy-N-(4-(2-(methylsu...)
Affinity DataIC50: 80nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sterling Road

Curated by ChEMBL
LigandPNGBDBM50229962(N-(4-METHOXYBENZYL)-N'-(5-NITRO-1,3-THIAZOL-2-YL)U...)
Affinity DataIC50: 100nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlycogen synthase kinase-3 beta(Human)
Sterling Road

Curated by ChEMBL
LigandPNGBDBM50130724(cid_4565878 | CHEMBL325353 | 1-(4-Amino-furazan-3-...)
Affinity DataIC50: 100nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sterling Road

Curated by ChEMBL
LigandPNGBDBM50293315(4-(1H-benzo[d]imidazol-2-yl)-6-(1-methyl-6-oxo-1,6...)
Affinity DataIC50: 160nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sterling Road

Curated by ChEMBL
LigandPNGBDBM10840(4-(5-bromo-1H-indol-3-yl)pyrimidin-2-amine | Merid...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sterling Road

Curated by ChEMBL
LigandPNGBDBM50293316((4-amino-2-(phenylamino)thiazol-5-yl)(cyclopropyl)...)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sterling Road

Curated by ChEMBL
LigandPNGBDBM50293317(4-benzyl-2-phenethyl-1,2,4-thiadiazolidine-3,5-dio...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sterling Road

Curated by ChEMBL
LigandPNGBDBM50293318(N-(4-(4-benzylpiperazin-1-yl)phenyl)-4-(4-methyl-2...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sterling Road

Curated by ChEMBL
LigandPNGBDBM11429(4-({5-[(4-aminocyclohexyl)amino]-3-cyclopentylpyra...)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sterling Road

Curated by ChEMBL
LigandPNGBDBM7348(6-(3,5-dimethoxyphenyl)-5H-pyrrolo[2,3-b]pyrazine ...)
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sterling Road

Curated by ChEMBL
LigandPNGBDBM10844(4-(1H-indol-3-yl)pyrimidin-2-amine | Meridianin G)
Affinity DataIC50: 3.50E+5nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sterling Road

Curated by ChEMBL
LigandPNGBDBM10846(4-(1H-indol-2-yl)pyrimidin-2-amine | isomeridianin...)
Affinity DataIC50: 4.20E+5nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sterling Road

Curated by ChEMBL
LigandPNGBDBM50293305(CT-98014 | N1-(4-(2,4-dichlorophenyl)-5-(1H-imidaz...)
Affinity DataKi:  0.0900nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed