Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50038688
TargetNeurotensin receptor type 1(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50240845(2-{(S)-2-[2-({(S)-1-[(S)-2-((S)-2-Amino-5-guanidin...)
Affinity DataKd:  0.630nMAssay Description:Displacement of [3H]NT(8-13) from wild type human NTR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50248034(CHEMBL506981 | SR 48692 | 2-{[1-(7-Chloro-quinolin...)
Affinity DataKd:  8.90nMAssay Description:Displacement of [3H]SR48692 from wild type human NTR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNeurotensin receptor type 1(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50263386(H-Arg-N-Me-Arg-Pro-Tyr-Ile-Leu-OH | CHEMBL443967)
Affinity DataKi:  0.510nMAssay Description:Displacement of [3H]NT(8-13) from wild type human NTR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50240845(2-{(S)-2-[2-({(S)-1-[(S)-2-((S)-2-Amino-5-guanidin...)
Affinity DataKi:  0.630nMAssay Description:Displacement of [3H]NT(8-13) from wild type human NTR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50130880(pGlu-Leu-Tyr-Glu-Asn-Lys-Pro-Arg-Arg-Pro-Tyr-Ile-L...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]NT(8-13) from wild type human NTR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50263388(H-Arg-Arg-Pro-Tyr-Ile-Aac-OH | CHEMBL507382)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]NT(8-13) from wild type human NTR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50263387(H-Arg-Arg-Pro-Tyr-N-Me-Ile-Leu-OH | CHEMBL503059)
Affinity DataKi:  160nMAssay Description:Displacement of [3H]NT(8-13) from wild type human NTR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50263385(H-Arg-Arg-Pro-Tyr-Ile-N-Me-Leu-OH | CHEMBL508130)
Affinity DataKi:  190nMAssay Description:Displacement of [3H]NT(8-13) from wild type human NTR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed