Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50027228
TargetPeroxisome proliferator-activated receptor gamma(Human)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50225835((2s,5s)-2-methyl-5-(4-(5-methyl-2-p-tolyloxazol-4-...)
Affinity DataEC50:  7.00E+3nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in human HepG2 cells co-transfected with PPRE3-TK-luc assessed as induction of be...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50275488(cis-2-methyl-5-(4-(4-(methylsulfonyloxy)phenyl)but...)
Affinity DataEC50:  2.00E+4nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells co-transfected with PPRE3-TK-luc assessed as induction of be...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM28798((2S)-2-ethoxy-3-(4-{2-[4-(methanesulfonyloxy)pheny...)
Affinity DataEC50:  820nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells co-transfected with PPRE3-TK-luc assessed as induction of be...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50225835((2s,5s)-2-methyl-5-(4-(5-methyl-2-p-tolyloxazol-4-...)
Affinity DataEC50:  7.00E+3nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells co-transfected with PPRE3-TK-luc assessed as induction of be...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50275537(cis-2-methyl-5-(6-(4-(methylsulfonyloxy)phenyl)hex...)
Affinity DataEC50:  1.50E+4nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells co-transfected with PPRE3-TK-luc assessed as induction of be...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50275536(cis-2-methyl-5-(5-(4-(methylsulfonyloxy)phenyl)pen...)
Affinity DataEC50:  2.50E+3nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells co-transfected with PPRE3-TK-luc assessed as induction of be...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM28798((2S)-2-ethoxy-3-(4-{2-[4-(methanesulfonyloxy)pheny...)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in human HepG2 cells co-transfected with PPRE3-TK-luc assessed as induction of be...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50275537(cis-2-methyl-5-(6-(4-(methylsulfonyloxy)phenyl)hex...)
Affinity DataEC50:  1.50E+4nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in human HepG2 cells co-transfected with PPRE3-TK-luc assessed as induction of be...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed