Compile Data Set for Download or QSAR
Report error Found 96 Enz. Inhib. hit(s) with all data for entry = 50038728
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253203BDBM50253203((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-(2-bromob...)
Affinity DataIC50: 38nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252672BDBM50252672((S)-1-(4-Methanesulfonamidephenoxy)-3-(3,4-dichlor...)
Affinity DataIC50: 50nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253241BDBM50253241((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-(2,3,4-tr...)
Affinity DataIC50: 51nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252889BDBM50252889((S)-1-(4-Methanesulfonamidophenoxy)-3-(3-fluoro-4-...)
Affinity DataIC50: 68nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253032BDBM50253032((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-butyl-3,4...)
Affinity DataIC50: 70nMAssay Description:Displacement of [3H]astemizole from human ERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252673BDBM50252673((S)-1-(4-Methanesulfonamido-2-fluorophenoxy)-3-(3,...)
Affinity DataIC50: 72nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007674BDBM50007674((+)-erythro 4-[2-(4-Benzyl-piperidin-1-yl)-1-hydro...)
Affinity DataIC50: 73nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253204BDBM50253204((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-(2-fluoro...)
Affinity DataIC50: 80nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253003BDBM50253003((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-ethyl-3,4...)
Affinity DataIC50: 96nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252886BDBM50252886((S)-1-(4-Methanesulfonamidophenoxy)-3-(4-chlorophe...)
Affinity DataIC50: 101nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253078BDBM50253078((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-(4-hydrox...)
Affinity DataIC50: 113nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253030BDBM50253030((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-(2-hydrox...)
Affinity DataIC50: 122nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253002BDBM50253002((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-methyl-3,...)
Affinity DataIC50: 130nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253031BDBM50253031((S)-1-(4-Methanesulfonamidophenoxy)3-(N-propyl-3,4...)
Affinity DataIC50: 130nMAssay Description:Displacement of [3H]astemizole from human ERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253120BDBM50253120((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-(2,4-dihy...)
Affinity DataIC50: 146nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253003BDBM50253003((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-ethyl-3,4...)
Affinity DataIC50: 170nMAssay Description:Displacement of [3H]astemizole from human ERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252846BDBM50252846((R)-1-(4-Methanesulfonamidophenoxy)-3-(N-(2-hydrox...)
Affinity DataIC50: 173nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253057BDBM50253057((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-benzyl-3,...)
Affinity DataIC50: 177nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252812BDBM50252812((R)-1-(4-Methanesulfonamidophenoxy)-3-(3,4-dichlor...)
Affinity DataIC50: 188nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252999BDBM50252999((S)-1-(4-Methanesulfonamidophenoxy)-3-(3,4-dimethy...)
Affinity DataIC50: 207nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253077BDBM50253077((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-(3-hydrox...)
Affinity DataIC50: 238nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253238BDBM50253238((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-(3-fluoro...)
Affinity DataIC50: 249nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252813BDBM50252813((R)-1-(4-Methanesulfonamidophenoxy)3-(N-methyl-3,4...)
Affinity DataIC50: 253nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253239BDBM50253239((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-(4-fluoro...)
Affinity DataIC50: 275nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252680BDBM50252680((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-(3-pridyl...)
Affinity DataIC50: 278nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253240BDBM50253240((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-(2,6-difl...)
Affinity DataIC50: 281nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252936BDBM50252936((S)-1-(4-Methanesulfonamidophenoxy)-3-(3,4-difluor...)
Affinity DataIC50: 357nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253054BDBM50253054((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-isobutyl-...)
Affinity DataIC50: 370nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253002BDBM50253002((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-methyl-3,...)
Affinity DataIC50: 370nMAssay Description:Displacement of [3H]astemizole from human ERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252888BDBM50252888((S)-1-(4-Methanesulfonamidophenoxy)-3-(3-chloro-4-...)
Affinity DataIC50: 397nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252849BDBM50252849((R)-1-(4-Methanesulfonamidophenoxy)-3-(N-(3-hydrox...)
Affinity DataIC50: 409nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253032BDBM50253032((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-butyl-3,4...)
Affinity DataIC50: 421nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252674BDBM50252674((S)-1-(4-Methanesulfonamido-3-fluorophenoxy)-3-(3,...)
Affinity DataIC50: 427nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252845BDBM50252845((S)-1-(4-Methanesulfonamidophenoxy)-3-(2-chlorophe...)
Affinity DataIC50: 429nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253057BDBM50253057((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-benzyl-3,...)
Affinity DataIC50: 430nMAssay Description:Displacement of [3H]astemizole from human ERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252848BDBM50252848((R)-1-(4-Methanesulfonamidophenoxy)-3-(N-(2-hydrox...)
Affinity DataIC50: 433nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253202BDBM50253202((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-(2-chloro...)
Affinity DataIC50: 479nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252678BDBM50252678((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-(2-acetyl...)
Affinity DataIC50: 500nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252672BDBM50252672((S)-1-(4-Methanesulfonamidephenoxy)-3-(3,4-dichlor...)
Affinity DataIC50: 500nMAssay Description:Binding affinity to dopamine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252672BDBM50252672((S)-1-(4-Methanesulfonamidephenoxy)-3-(3,4-dichlor...)
Affinity DataIC50: 500nMAssay Description:Binding affinity to norepinephrine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253277BDBM50253277((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-(2,3,4,5,...)
Affinity DataIC50: 524nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252676BDBM50252676((S)-1-(3-Methanesulfonamidophenoxy)-3-(3,4-dichlor...)
Affinity DataIC50: 530nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252933BDBM50252933((S)-1-(4-Methanesulfonamidophenoxy)-3-(2-fluorophe...)
Affinity DataIC50: 573nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252805BDBM50252805((S)-1-(4-ethylsulphonamidophenoxy)-3-(3,4-dichloro...)
Affinity DataIC50: 587nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252677BDBM50252677((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-(2-nitrob...)
Affinity DataIC50: 589nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253056BDBM50253056((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-isopropyl...)
Affinity DataIC50: 603nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252885BDBM50252885((S)-1-(4-Methanesulfonamidophenoxy)-3-(3-chlorophe...)
Affinity DataIC50: 628nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253031BDBM50253031((S)-1-(4-Methanesulfonamidophenoxy)3-(N-propyl-3,4...)
Affinity DataIC50: 635nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253033BDBM50253033((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-pentyl-3,...)
Affinity DataIC50: 659nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253076BDBM50253076((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-(2-hydrox...)
Affinity DataIC50: 662nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
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