Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50027014
TargetTrace amine-associated receptor 1(Rat)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM18959(CHEMBL1598 | Di-N-desethylamiodarone | L 33530 | 3...)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at rat TAAR1 expressed in HEK293 cells assessed as intracellular cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Rat)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50247087((2-butylbenzofuran-3-yl)(3-ethyl-4-(2-(ethylamino)...)
Affinity DataEC50:  33nMAssay Description:Antagonist activity at rat TAAR1 expressed in HEK293 cells assessed as intracellular cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Rat)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50247119((2-butylbenzofuran-3-yl)(4-(2-(ethylamino)ethoxy)-...)
Affinity DataEC50:  33nMAssay Description:Antagonist activity at rat TAAR1 expressed in HEK293 cells assessed as intracellular cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Rat)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM18958(DEA | (2-{4-[(2-butyl-1-benzofuran-3-yl)carbonyl]-...)
Affinity DataEC50:  33nMAssay Description:Antagonist activity at rat TAAR1 expressed in HEK293 cells assessed as intracellular cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Rat)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM18961(DDIA | L 3937 | CHEMBL461546 | (2-{4-[(2-butyl-1-b...)
Affinity DataEC50:  33nMAssay Description:Antagonist activity at rat TAAR1 expressed in HEK293 cells assessed as intracellular cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Rat)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM18960(MIA | (2-{4-[(2-butyl-1-benzofuran-3-yl)carbonyl]-...)
Affinity DataEC50:  33nMAssay Description:Antagonist activity at rat TAAR1 expressed in HEK293 cells assessed as intracellular cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed