Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50026714
LigandPNGBDBM50174298(3-(4-(3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl)bicy...)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of human 11beta-HSD1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50239401(MERCK-544 | 3-Adamantan-1-yl-6,7,8,9-tetrahydro-5H...)
Affinity DataIC50: 7.5nMAssay Description:Inhibition of 11beta-HSD1 expressed in CHO-K1 cells assessed as conversion of [3H]cortisone to cortisol by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50241490(N-(3-((4aR,8aS)-decahydroquinoline-1-carbonyl)phen...)
Affinity DataIC50: 14nMAssay Description:Inhibition of human recombinant 11beta-HSD1 expressed in Pichia pastorisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50117901(2-[2-(3-Chloro-2-methyl-benzenesulfonylamino)-thia...)
Affinity DataIC50: 52nMAssay Description:Inhibition of human 11beta-HSD1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50117900(CHEMBL463978 | CHEMBL553071 | 3-Chloro-2-methyl-N-...)
Affinity DataIC50: 96nMAssay Description:Inhibition of human 11beta-HSD2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50117901(2-[2-(3-Chloro-2-methyl-benzenesulfonylamino)-thia...)
Affinity DataIC50: 284nMAssay Description:Inhibition of human 11beta-HSD2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50174298(3-(4-(3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl)bicy...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human 11beta-HSD2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50239401(MERCK-544 | 3-Adamantan-1-yl-6,7,8,9-tetrahydro-5H...)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of 11beta-HSD2 expressed in CHO-K1 cells assessed as conversion of [3H]cortisol to cortisone by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50117900(CHEMBL463978 | CHEMBL553071 | 3-Chloro-2-methyl-N-...)
Affinity DataIC50: 3.34E+3nMAssay Description:Inhibition of human 11beta-HSD1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50117901(2-[2-(3-Chloro-2-methyl-benzenesulfonylamino)-thia...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human 11beta-HSD2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50117900(CHEMBL463978 | CHEMBL553071 | 3-Chloro-2-methyl-N-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human 11beta-HSD2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed