Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50026705
TargetExcitatory amino acid transporter 3(Human)
The University of Montana

Curated by ChEMBL
LigandPNGBDBM50273238((S,S)-beta-3 Fluoro-Benzylaspartate | CHEMBL457411)
Affinity DataIC50: 2.46E+3nMAssay Description:Displacement of [3H]D-aspartate from human EAAT3 expressed in mouse C17.2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 3(Human)
The University of Montana

Curated by ChEMBL
LigandPNGBDBM50273197(L-threo-beta-(1-naphthyl)methyloxaspartate | CHEMB...)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of [14C]glutamate uptake at human EAAT3 expressed in african green monkey COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 3(Human)
The University of Montana

Curated by ChEMBL
LigandPNGBDBM50273237(L-threo-beta-(2-naphthyl)methyloxaspartate | CHEMB...)
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of [14C]glutamate uptake at human EAAT3 expressed in african green monkey COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 3(Human)
The University of Montana

Curated by ChEMBL
LigandPNGBDBM50093753(DL-TBOA | (2S,3S)-2-amino-3-(benzyloxy)succinic ac...)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of [14C]glutamate uptake at human EAAT3 expressed in african green monkey COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 3(Human)
The University of Montana

Curated by ChEMBL
LigandPNGBDBM50273239((S,R)-beta-3 Fluoro-Benzylaspartate | CHEMBL457412)
Affinity DataIC50: 2.11E+4nMAssay Description:Displacement of [3H]D-aspartate from human EAAT3 expressed in mouse C17.2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed