Compile Data Set for Download or QSAR
Report error Found 88 Enz. Inhib. hit(s) with all data for entry = 50026703
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 59087BDBM59087(CHEMBL258765 | Fascaplysin | Fasca-plysi)
Affinity DataIC50: 550nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50188071BDBM50188071(biphenyl-4-carboxylic acid [2-(1H-indol-3-yl)-ethy...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273105BDBM50273105((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(4'-me...)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272870BDBM50272870(N-(2-(1H-Indol-3-yl)ethyl)-4'-tert-butylbiphenyl-4...)
Affinity DataIC50: 9.20E+3nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273041BDBM50273041((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(3'-me...)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272800BDBM50272800(N-(2-(1H-Indol-3-yl)ethyl)-4'-tert-butyl-N-methylb...)
Affinity DataIC50: 1.12E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273074BDBM50273074((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(4'-fl...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272837BDBM50272837(N-(2-(1H-Indol-3-yl)ethyl)-4'-fluorobiphenyl-4-car...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272919BDBM50272919(N-(2-(1H-Indol-3-yl)ethyl)-3'-methylbiphenyl-2-car...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272836BDBM50272836(N-(2-(1H-Indol-3-yl)ethyl)biphenyl-4-carboxamide |...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273076BDBM50273076((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(2'-fl...)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272838BDBM50272838(N-(2-(1H-Indol-3-yl)ethyl)-4'-methylbiphenyl-4-car...)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273039BDBM50273039((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(2'-fl...)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272997BDBM50272997((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(2'-fl...)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272918BDBM50272918(N-(2-(1H-Indol-3-yl)ethyl)-3'-fluorobiphenyl-2-car...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272798BDBM50272798(N-(2-(1H-Indol-3-yl)ethyl)-4'-fluoro-N-methylbiphe...)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273075BDBM50273075((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(3'-fl...)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273109BDBM50273109((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(2'-me...)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272995BDBM50272995((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(4'-fl...)
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272799BDBM50272799(N-(2-(1H-Indol-3-yl)ethyl)-N,4'-dimethylbiphenyl-4...)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273040BDBM50273040((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(4'-me...)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272999BDBM50272999((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(4'-fl...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273106BDBM50273106((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(3'-me...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273141BDBM50273141(N-(2-(1H-Indol-3-yl)ethyl)-N-methyl-4-(pyridin-4-y...)
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272917BDBM50272917(N-(2-(1H-Indol-3-yl)ethyl)-2'-methoxybiphenyl-2-ca...)
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272998BDBM50272998((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(3'-me...)
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273038BDBM50273038((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(3'-fl...)
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273108BDBM50273108((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(3'-me...)
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273142BDBM50273142(N-(2-(1H-Indol-3-yl)ethyl)-3-(pyridin-3-yl)benzami...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273107BDBM50273107((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(2'-me...)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273072BDBM50273072((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(3'-me...)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272996BDBM50272996((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(3'-fl...)
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272835BDBM50272835(N-(2-(1H-Indol-3-yl)ethyl)-4'-phenyl-N-methylbiphe...)
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273144BDBM50273144((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(2-(py...)
Affinity DataIC50: 3.60E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272873BDBM50272873(N-(2-(1H-Indol-3-yl)ethyl)-4'-fluorobiphenyl-2-car...)
Affinity DataIC50: 3.80E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272874BDBM50272874(N-(2-(1H-Indol-3-yl)ethyl)-4'-tert-butylbiphenyl-2...)
Affinity DataIC50: 3.80E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273143BDBM50273143((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(2-(py...)
Affinity DataIC50: 3.90E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272871BDBM50272871(N-(2-(1H-Indol-3-yl)ethyl)-4'-methoxybiphenyl-4-ca...)
Affinity DataIC50: 4.80E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272834BDBM50272834(N-(2-(1H-Indol-3-yl)ethyl)-4'-methoxy-N-methylbiph...)
Affinity DataIC50: 4.90E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272916BDBM50272916(N-(2-(1H-Indol-3-yl)ethyl)-3'-methoxybiphenyl-2-ca...)
Affinity DataIC50: 5.30E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272799BDBM50272799(N-(2-(1H-Indol-3-yl)ethyl)-N,4'-dimethylbiphenyl-4...)
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibition of human CDK2/GST-cyclin A expressed in Sf9 cells assessed as histone phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273042BDBM50273042((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(2'-me...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272915BDBM50272915(N-(2-(1H-Indol-3-yl)ethyl)-4'-methoxybiphenyl-2-ca...)
Affinity DataIC50: 7.90E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273073BDBM50273073(Biphenyl-3-yl(3,4-dihydro-1H-pyrido[3,4-b]indol-2(...)
Affinity DataIC50: 7.90E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272872BDBM50272872(N-(2-(1H-Indol-3-yl)ethyl)biphenyl-3-carboxamide |...)
Affinity DataIC50: 8.60E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272835BDBM50272835(N-(2-(1H-Indol-3-yl)ethyl)-4'-phenyl-N-methylbiphe...)
Affinity DataIC50: 9.10E+4nMAssay Description:Inhibition of human CDK2/GST-cyclin A expressed in Sf9 cells assessed as histone phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273141BDBM50273141(N-(2-(1H-Indol-3-yl)ethyl)-N-methyl-4-(pyridin-4-y...)
Affinity DataIC50: 9.20E+4nMAssay Description:Inhibition of human CDK2/GST-cyclin A expressed in Sf9 cells assessed as histone phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273142BDBM50273142(N-(2-(1H-Indol-3-yl)ethyl)-3-(pyridin-3-yl)benzami...)
Affinity DataIC50: 1.50E+5nMAssay Description:Inhibition of human CDK2/GST-cyclin A expressed in Sf9 cells assessed as histone phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272874BDBM50272874(N-(2-(1H-Indol-3-yl)ethyl)-4'-tert-butylbiphenyl-2...)
Affinity DataIC50: 2.62E+5nMAssay Description:Inhibition of human CDK2/GST-cyclin A expressed in Sf9 cells assessed as histone phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
University of Leicester

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272834BDBM50272834(N-(2-(1H-Indol-3-yl)ethyl)-4'-methoxy-N-methylbiph...)
Affinity DataIC50: 2.89E+5nMAssay Description:Inhibition of human CDK2/GST-cyclin A expressed in Sf9 cells assessed as histone phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
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