Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50026618
TargetTyrosine-protein kinase ABL1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50262718(N-(5-(4-methoxybenzyl)thiazol-2-yl)thiophene-2-car...)
Affinity DataKi:  16nMAssay Description:Inhibition of Abl kinase by cell free assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50262723(N-(5-(2,5-dichlorobenzyl)thiazol-2-yl)thiophene-2-...)
Affinity DataKi:  50nMAssay Description:Inhibition of Abl kinase by cell free assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50262722(Thiophene-2-carboxylic acid [5-(3-methyl-benzyl)-t...)
Affinity DataKi:  59nMAssay Description:Inhibition of Abl kinase by cell free assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50262667(cid_889490 | CHEMBL477139 | N-(6-methoxy-8H-indeno...)
Affinity DataKi:  68nMAssay Description:Inhibition of Abl kinase by cell free assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50262664(CHEMBL504598 | cid_644846 | N-(5-benzylthiazol-2-y...)
Affinity DataKi:  90nMAssay Description:Inhibition of Abl kinase by cell free assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50262715(CHEMBL518430 | cid_1113641 | N-(5-(3-chlorobenzyl)...)
Affinity DataKi:  97nMAssay Description:Inhibition of Abl kinase by cell free assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50262665(N-(5-(4-fluorobenzyl)thiazol-2-yl)thiophene-2-carb...)
Affinity DataKi:  130nMAssay Description:Inhibition of Abl kinase by cell free assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50262669(N-(5-(3-(trifluoromethyl)benzyl)thiazol-2-yl)thiop...)
Affinity DataKi:  136nMAssay Description:Inhibition of Abl kinase by cell free assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50262671(N-(5-(2-fluorobenzyl)thiazol-2-yl)thiophene-2-carb...)
Affinity DataKi:  170nMAssay Description:Inhibition of Abl kinase by cell free assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50262670(N-(5-(2-chlorobenzyl)thiazol-2-yl)thiophene-2-carb...)
Affinity DataKi:  245nMAssay Description:Inhibition of Abl kinase by cell free assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50262719(CHEMBL476513 | cid_1113642 | Thiophene-2-carboxyli...)
Affinity DataKi:  249nMAssay Description:Inhibition of Abl kinase by cell free assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50262668(N-(5-(phenoxymethyl)-1,3,4-thiadiazol-2-yl)thiophe...)
Affinity DataKi:  278nMAssay Description:Inhibition of Abl kinase by cell free assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50262724(N-(5-benzyl-1,3,4-thiadiazol-2-yl)thiophene-2-carb...)
Affinity DataKi:  360nMAssay Description:Inhibition of Abl kinase by cell free assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50262714(N-(5-(4-chlorobenzyl)thiazol-2-yl)thiophene-2-carb...)
Affinity DataKi:  624nMAssay Description:Inhibition of Abl kinase by cell free assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50262721(N-(5-(4-chlorophenyl)thiazol-2-yl)thiophene-2-carb...)
Affinity DataKi:  791nMAssay Description:Inhibition of Abl kinase by cell free assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50262716(N-(5-(2-chloro-5-(trifluoromethyl)benzyl)thiazol-2...)
Affinity DataKi:  845nMAssay Description:Inhibition of Abl kinase by cell free assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50262720(N-(5-(4-fluorophenyl)thiazol-2-yl)thiophene-2-carb...)
Affinity DataKi:  1.65E+3nMAssay Description:Inhibition of Abl kinase by cell free assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50262717(N-(5-(2,4-dichlorobenzyl)thiazol-2-yl)thiophene-2-...)
Affinity DataKi:  3.47E+3nMAssay Description:Inhibition of Abl kinase by cell free assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed