Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50038634
TargetHistamine H3 receptor(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50263096(N-cyclohexyl-6-(1-isopropylpiperidin-4-yloxy)-2-na...)
Affinity DataEC50:  21nMAssay Description:Inverse agonist activity at human histamine H3 receptor expressed in CHO cells by GTPgammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50110288([4-(3-Piperidin-1-yl-propoxy)-phenyl]-quinolin-4-y...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]RAMH from human histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50263054((6-(3-(piperidin-1-yl)propoxy)naphthalen-2-yl)(pyr...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]RAMH from human histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50139391((R)-4-(2-(2-(2-methylpyrrolidin-1-yl)ethyl)benzofu...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]RAMH from human histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50370569(A-349821 | A-349,821)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]RAMH from human histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50263055((6-(1-isopropylpiperidin-4-yloxy)naphthalen-2-yl)(...)
Affinity DataKi:  57nMAssay Description:Displacement of [3H]RAMH from human histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50263096(N-cyclohexyl-6-(1-isopropylpiperidin-4-yloxy)-2-na...)
Affinity DataKi:  87nMAssay Description:Displacement of [3H]RAMH from human histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed