Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 3231
TargetEstrogen-related receptor gamma(Human)
Kyushu University

LigandPNGBDBM20608([3H]4-OHT | cid_449459 | CHEMBL489 | AFIMOXIFENE |...)
Affinity DataIC50: 10.3nMpH: 7.4 T: 2°CAssay Description:The receptor-binding assay was conducted using [3H]4-hydroxytamoxifen (4-OHT) as the radioligand. To estimate the binding affinity, the IC50 values (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEstrogen-related receptor gamma(Human)
Kyushu University

LigandPNGBDBM29608(Diphenylolpropane | Bisphenol A (BPA) | US9688816,...)
Affinity DataIC50: 13.1nMpH: 7.4 T: 2°CAssay Description:The receptor-binding assay was conducted using [3H]4-hydroxytamoxifen (4-OHT) as the radioligand. To estimate the binding affinity, the IC50 values (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEstrogen-related receptor gamma(Human)
Kyushu University

LigandPNGBDBM29609(4-cumylphenol | 4-alpha-Cumylphenol | US9688816, B)
Affinity DataIC50: 13.9nMpH: 7.4 T: 2°CAssay Description:The receptor-binding assay was conducted using [3H]4-hydroxytamoxifen (4-OHT) as the radioligand. To estimate the binding affinity, the IC50 values (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEstrogen-related receptor gamma(Human)
Kyushu University

LigandPNGBDBM29610(2,2-Diphenylpropane)
Affinity DataIC50: 1.00E+4nMpH: 7.4 T: 2°CAssay Description:The receptor-binding assay was conducted using [3H]4-hydroxytamoxifen (4-OHT) as the radioligand. To estimate the binding affinity, the IC50 values (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed