Compile Data Set for Download or QSAR
Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 50038630
TargetCannabinoid receptor 1(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM21279(N-(piperidin-1-yl)-1-(2,4-dichlorophenyl)-5-(4-iod...)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50180022(5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1...)
Affinity DataKi:  5.40nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50263033(N-(3,3-Diphenyl)propyl-2,2-diphenylacetamide | CHE...)
Affinity DataKi:  58nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM21279(N-(piperidin-1-yl)-1-(2,4-dichlorophenyl)-5-(4-iod...)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50263074(2-(4-Bromophenyl)-2-phenyl-N-(3,3-diphenylpropyl)-...)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50263032(N-(3,3-Diphenyl)propyl-2-chloro-2,2-diphenylacetam...)
Affinity DataKi:  280nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50263034(N-(3,3-Diphenyl)propyl-2-methyl-2,2-diphenylacetam...)
Affinity DataKi:  290nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50263116(2-(4-Hydroxyphenyl)-2-phenyl-N-(3,3-diphenylpropyl...)
Affinity DataKi:  560nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50263034(N-(3,3-Diphenyl)propyl-2-methyl-2,2-diphenylacetam...)
Affinity DataKi:  560nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50263073(2-(4-Chlorophenyl)-2-phenyl-N-(3,3-diphenylpropyl)...)
Affinity DataKi:  560nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50263075(2-(4-Methoxyphenyl)-2-phenyl-N-(3,3-diphenylpropyl...)
Affinity DataKi:  560nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50263114(2-(4-Methylphenyl)-2-phenyl-N-(3,3-diphenylpropyl)...)
Affinity DataKi:  560nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50263115(2-(4-Nitrophenyl)-2-phenyl-N-(3,3-diphenylpropyl)-...)
Affinity DataKi:  560nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50263154(N-(3,3-Diphenyl)propyl-2-phenylacetamide | CHEMBL5...)
Affinity DataKi:  560nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50263114(2-(4-Methylphenyl)-2-phenyl-N-(3,3-diphenylpropyl)...)
Affinity DataKi:  650nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50263115(2-(4-Nitrophenyl)-2-phenyl-N-(3,3-diphenylpropyl)-...)
Affinity DataKi:  790nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50263075(2-(4-Methoxyphenyl)-2-phenyl-N-(3,3-diphenylpropyl...)
Affinity DataKi:  790nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataKi:  790nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50263197(N-(3,3-Diphenyl)propyl-2-(4-bromophenyl) acetamide...)
Affinity DataKi:  800nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50263117(2-(4-Aminophenyl)-2-phenyl-N-(3,3-diphenylpropyl)-...)
Affinity DataKi:  900nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50263116(2-(4-Hydroxyphenyl)-2-phenyl-N-(3,3-diphenylpropyl...)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50263117(2-(4-Aminophenyl)-2-phenyl-N-(3,3-diphenylpropyl)-...)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50263197(N-(3,3-Diphenyl)propyl-2-(4-bromophenyl) acetamide...)
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50263032(N-(3,3-Diphenyl)propyl-2-chloro-2,2-diphenylacetam...)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50263155(N-(3,3-Diphenyl)propyl-2-(4-chlorophenyl)acetamide...)
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50263153(N-(3-Phenyl)propyl-2-(4-bromophenylacetamide) | CH...)
Affinity DataKi:  1.80E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50263153(N-(3-Phenyl)propyl-2-(4-bromophenylacetamide) | CH...)
Affinity DataKi:  1.90E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50263035(N-(3,3-Diphenyl)propyl-2-hydroxy-2,2-diphenylaceta...)
Affinity DataKi:  2.20E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50263152(N-(3-Phenyl)propyl-2-(4-chlorophenyl)-2-phenylacet...)
Affinity DataKi:  2.20E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50263035(N-(3,3-Diphenyl)propyl-2-hydroxy-2,2-diphenylaceta...)
Affinity DataKi:  2.30E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50263155(N-(3,3-Diphenyl)propyl-2-(4-chlorophenyl)acetamide...)
Affinity DataKi:  2.40E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50263152(N-(3-Phenyl)propyl-2-(4-chlorophenyl)-2-phenylacet...)
Affinity DataKi:  2.40E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50263151(N-(3-Phenyl)propyl-2,2-diphenylacetamide | CHEMBL4...)
Affinity DataKi:  3.40E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50180022(5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1...)
Affinity DataKi: >5.60E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50263154(N-(3,3-Diphenyl)propyl-2-phenylacetamide | CHEMBL5...)
Affinity DataKi: >7.90E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50263151(N-(3-Phenyl)propyl-2,2-diphenylacetamide | CHEMBL4...)
Affinity DataKi: >7.90E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50263074(2-(4-Bromophenyl)-2-phenyl-N-(3,3-diphenylpropyl)-...)
Affinity DataKi: >7.90E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50263073(2-(4-Chlorophenyl)-2-phenyl-N-(3,3-diphenylpropyl)...)
Affinity DataKi: >7.90E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50263033(N-(3,3-Diphenyl)propyl-2,2-diphenylacetamide | CHE...)
Affinity DataKi:  7.90E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed