Compile Data Set for Download or QSAR
Report error Found 77 Enz. Inhib. hit(s) with all data for entry = 50038624
TargetExcitatory amino acid transporter 2(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50247191((2S,3S)-2-Amino-3-benzyloxy-succinic acid | DL-thr...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT2 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 1(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50247191((2S,3S)-2-Amino-3-benzyloxy-succinic acid | DL-thr...)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT1 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 3(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50247191((2S,3S)-2-Amino-3-benzyloxy-succinic acid | DL-thr...)
Affinity DataIC50: 9.30E+3nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT3 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 2(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50251894((2S,4R)-4-(2,2-Diphenylethylamino-3-oxopropyl)glut...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT2 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 2(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50240399(dihydrokainic acid | Dihydrokainate | (2R,3R,4S)-3...)
Affinity DataIC50: 8.90E+4nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT2 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 2(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50252046((2S,4S)-2-amino-4-(benzyloxymethyl)pentanedioic ac...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT2 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 2(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50251951((2S,4S)-2-amino-4-(hydroxymethyl)pentanedioic acid...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT2 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 2(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50252048((2S,4R)-2-amino-4-(3-methoxy-3-oxopropyl)pentanedi...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT2 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 2(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50251893((2S,4R)-2-amino-4-(3-(benzylamino)-3-oxopropyl)pen...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT2 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 1(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50252051((2S,4R)-2-amino-4-(3-(methylamino)-3-oxopropyl)pen...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT1 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 1(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50252046((2S,4S)-2-amino-4-(benzyloxymethyl)pentanedioic ac...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT1 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 1(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50252662((2S,4R)-4-(3-Propylamino-3-oxopropyl)glutamic acid...)
Affinity DataIC50: 3.00E+6nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT1 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 1(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50251893((2S,4R)-2-amino-4-(3-(benzylamino)-3-oxopropyl)pen...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT1 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 1(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50251894((2S,4R)-4-(2,2-Diphenylethylamino-3-oxopropyl)glut...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT1 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 1(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50240399(dihydrokainic acid | Dihydrokainate | (2R,3R,4S)-3...)
Affinity DataIC50: 3.00E+6nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT1 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 3(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50251951((2S,4S)-2-amino-4-(hydroxymethyl)pentanedioic acid...)
Affinity DataIC50: 3.00E+6nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT3 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 1(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50251951((2S,4S)-2-amino-4-(hydroxymethyl)pentanedioic acid...)
Affinity DataIC50: 3.00E+6nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT1 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 3(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50251894((2S,4R)-4-(2,2-Diphenylethylamino-3-oxopropyl)glut...)
Affinity DataIC50: 1.00E+6nMAssay Description:Binding affinity to human cloned mGluR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50251894((2S,4R)-4-(2,2-Diphenylethylamino-3-oxopropyl)glut...)
Affinity DataIC50: 1.00E+6nMAssay Description:Binding affinity to human cloned mGluR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 1(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50252050((2S,4R)-2-amino-4-(3-amino-3-oxopropyl)pentanedioi...)
Affinity DataIC50: 3.00E+6nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT1 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 1(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50252048((2S,4R)-2-amino-4-(3-methoxy-3-oxopropyl)pentanedi...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT1 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 1(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50252049((2S,4R)-4-(3-Hydroxy-3-oxopropyl)glutamic Acid | (...)
Affinity DataIC50: 3.00E+6nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT1 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 1(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50252047((2S,4S)-4-aminobutane-1,2,4-tricarboxylic acid | (...)
Affinity DataIC50: 3.00E+6nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT1 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 3(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50252662((2S,4R)-4-(3-Propylamino-3-oxopropyl)glutamic acid...)
Affinity DataIC50: 3.00E+6nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT3 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 2(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50252662((2S,4R)-4-(3-Propylamino-3-oxopropyl)glutamic acid...)
Affinity DataIC50: 3.00E+6nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT2 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 2(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50252051((2S,4R)-2-amino-4-(3-(methylamino)-3-oxopropyl)pen...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT2 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 2(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50252050((2S,4R)-2-amino-4-(3-amino-3-oxopropyl)pentanedioi...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT2 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 2(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50252049((2S,4R)-4-(3-Hydroxy-3-oxopropyl)glutamic Acid | (...)
Affinity DataIC50: 3.00E+6nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT2 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 2(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50252047((2S,4S)-4-aminobutane-1,2,4-tricarboxylic acid | (...)
Affinity DataIC50: 3.00E+6nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT2 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 3(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50240399(dihydrokainic acid | Dihydrokainate | (2R,3R,4S)-3...)
Affinity DataIC50: 3.00E+6nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT3 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 3(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50251894((2S,4R)-4-(2,2-Diphenylethylamino-3-oxopropyl)glut...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT3 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 3(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50251893((2S,4R)-2-amino-4-(3-(benzylamino)-3-oxopropyl)pen...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT3 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 3(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50252051((2S,4R)-2-amino-4-(3-(methylamino)-3-oxopropyl)pen...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT3 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 3(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50252050((2S,4R)-2-amino-4-(3-amino-3-oxopropyl)pentanedioi...)
Affinity DataIC50: 3.00E+6nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT3 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 3(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50252048((2S,4R)-2-amino-4-(3-methoxy-3-oxopropyl)pentanedi...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT3 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 3(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50252049((2S,4R)-4-(3-Hydroxy-3-oxopropyl)glutamic Acid | (...)
Affinity DataIC50: 3.00E+6nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT3 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 3(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50252047((2S,4S)-4-aminobutane-1,2,4-tricarboxylic acid | (...)
Affinity DataIC50: 3.00E+6nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT3 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 3(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50252046((2S,4S)-2-amino-4-(benzyloxymethyl)pentanedioic ac...)
Affinity DataIC50: 3.00E+6nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT3 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 3(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM17657(L-Glutamic acid | L-Glu | (2S)-2-aminopentanedioic...)
Affinity DataKi:  51nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT3 in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50240399(dihydrokainic acid | Dihydrokainate | (2R,3R,4S)-3...)
Affinity DataKi:  376nMAssay Description:Displacement of [3H]SYM2081 from rat cloned iGluR7More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 3(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50252046((2S,4S)-2-amino-4-(benzyloxymethyl)pentanedioic ac...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT3 in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 3(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50251893((2S,4R)-2-amino-4-(3-(benzylamino)-3-oxopropyl)pen...)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT3 in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 3(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50251894((2S,4R)-4-(2,2-Diphenylethylamino-3-oxopropyl)glut...)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT3 in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 3(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50252662((2S,4R)-4-(3-Propylamino-3-oxopropyl)glutamic acid...)
Affinity DataKi: >3.00E+3nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT3 in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 3(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50252051((2S,4R)-2-amino-4-(3-(methylamino)-3-oxopropyl)pen...)
Affinity DataKi: >3.00E+3nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT3 in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 3(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50252050((2S,4R)-2-amino-4-(3-amino-3-oxopropyl)pentanedioi...)
Affinity DataKi: >3.00E+3nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT3 in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 3(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50252048((2S,4R)-2-amino-4-(3-methoxy-3-oxopropyl)pentanedi...)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT3 in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 3(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50252049((2S,4R)-4-(3-Hydroxy-3-oxopropyl)glutamic Acid | (...)
Affinity DataKi: >3.00E+3nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT3 in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 3(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50252047((2S,4S)-4-aminobutane-1,2,4-tricarboxylic acid | (...)
Affinity DataKi: >3.00E+3nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT3 in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 3(Human)
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50251951((2S,4S)-2-amino-4-(hydroxymethyl)pentanedioic acid...)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT3 in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
Displayed 1 to 50 (of 77 total ) | Next | Last >>
Jump to: