Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50026444
TargetAminopeptidase N(Pig)
Shandong University

Curated by ChEMBL
LigandPNGBDBM23971(CHEMBL29292 | (2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-...)
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibition of pig kidney microsomes aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM23971(CHEMBL29292 | (2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-...)
Affinity DataIC50: 9.50E+3nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50252583((2R)-N-[5-(4-Methoxyphenyl)-1,3,4-thiadiazol-2-yl]...)
Affinity DataIC50: 3.14E+4nMAssay Description:Inhibition of pig kidney microsomes aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50252587((2R)-N-[5-(4-Bromophenyl)-1,3,4-thiadiazol-2-yl]-2...)
Affinity DataIC50: 3.53E+4nMAssay Description:Inhibition of pig kidney microsomes aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50251877((2R)-N-[5-(4-Nitrorophenyl)-1,3,4-thiadiazol-2-yl]...)
Affinity DataIC50: 4.46E+4nMAssay Description:Inhibition of pig kidney microsomes aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50252640((2R)-N-[5-(4-Nitrorophenyl)-1,3,4-thiadiazol-2-yl]...)
Affinity DataIC50: 5.41E+4nMAssay Description:Inhibition of pig kidney microsomes aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50252642((2R)-N-[5-(4-Methoxyphenyl)-1,3,4-thiadiazol-2-yl]...)
Affinity DataIC50: 6.88E+4nMAssay Description:Inhibition of pig kidney microsomes aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50252023((2R)-N-[5-(4-Methoxyphenyl)-1,3,4-thiadiazol-2-yl]...)
Affinity DataIC50: 7.85E+4nMAssay Description:Inhibition of pig kidney microsomes aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50252532((2R)-N-[5-(4-Nitrorophenyl)-1,3,4-thiadiazol-2-yl]...)
Affinity DataIC50: 8.47E+4nMAssay Description:Inhibition of pig kidney microsomes aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50251874((2R)-N-[5-(4-Fluorophenyl)-1,3,4-thiadiazol-2-yl]-...)
Affinity DataIC50: 9.07E+4nMAssay Description:Inhibition of pig kidney microsomes aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50252586((2R)-N-[5-(4-Chlorophenyl)-1,3,4-thiadiazol-2-yl]-...)
Affinity DataIC50: 1.05E+5nMAssay Description:Inhibition of pig kidney microsomes aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50251876((2R)-N-[5-(4-Bromophenyl)-1,3,4-thiadiazol-2-yl]-2...)
Affinity DataIC50: 1.08E+5nMAssay Description:Inhibition of pig kidney microsomes aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50252531((2R)-N-[5-(4-Bromophenyl)-1,3,4-thiadiazol-2-yl]-2...)
Affinity DataIC50: 1.15E+5nMAssay Description:Inhibition of pig kidney microsomes aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50252585((2R)-N-[5-(4-Fluorophenyl)-1,3,4-thiadiazol-2-yl]-...)
Affinity DataIC50: 1.15E+5nMAssay Description:Inhibition of pig kidney microsomes aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50252584((2R)-N-[5-Phenyl-1,3,4-thiadiazol-2-yl]-2-[(p-coum...)
Affinity DataIC50: 1.24E+5nMAssay Description:Inhibition of pig kidney microsomes aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50252641((2R)-N-[5-(4-Methylphenyl)-1,3,4-thiadiazol-2-yl]-...)
Affinity DataIC50: 1.27E+5nMAssay Description:Inhibition of pig kidney microsomes aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50252643((2R)-N-[5-Phenyl-1,3,4-thiadiazol-2-yl]-2-[(pmetho...)
Affinity DataIC50: 1.31E+5nMAssay Description:Inhibition of pig kidney microsomes aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50251875((2R)-N-[5-(4-Chlorophenyl)-1,3,4-thiadiazol-2-yl]-...)
Affinity DataIC50: 1.35E+5nMAssay Description:Inhibition of pig kidney microsomes aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50251922((2R)-N-[5-(4-Methylphenyl)-1,3,4-thiadiazol-2-yl]-...)
Affinity DataIC50: 1.41E+5nMAssay Description:Inhibition of pig kidney microsomes aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50252530((2R)-N-[5-(4-Chlorophenyl)-1,3,4-thiadiazol-2-yl]-...)
Affinity DataIC50: 1.53E+5nMAssay Description:Inhibition of pig kidney microsomes aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50252529((2R)-N-[5-(4-Fluorophenyl)-1,3,4-thiadiazol-2-yl]-...)
Affinity DataIC50: 1.83E+5nMAssay Description:Inhibition of pig kidney microsomes aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50252533((2R)-N-[5-(4-Methylphenyl)-1,3,4-thiadiazol-2-yl]-...)
Affinity DataIC50: 2.06E+5nMAssay Description:Inhibition of pig kidney microsomes aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50252490((2R)-N-[5-phenyl-1,3,4-thiadiazol-2-yl]-2-[(cinnam...)
Affinity DataIC50: 2.16E+5nMAssay Description:Inhibition of pig kidney microsomes aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50251877((2R)-N-[5-(4-Nitrorophenyl)-1,3,4-thiadiazol-2-yl]...)
Affinity DataIC50: 2.97E+5nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed