Compile Data Set for Download or QSAR
Report error Found 149 Enz. Inhib. hit(s) with all data for entry = 50026258
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244318BDBM50244318(2-(4-ethoxybenzyl)-1-(cyclohexylmethyl)-N,N-diethy...)
Affinity DataEC50:  0.520nMAssay Description:Agonist activity at cloned human CB2 receptor in Sf9 cells assessed as stimulation of [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244317BDBM50244317(2-(4-ethoxybenzyl)-1-(cyclopentylmethyl)-N,N-dieth...)
Affinity DataEC50:  0.700nMAssay Description:Agonist activity at cloned human CB2 receptor in Sf9 cells assessed as stimulation of [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50243706BDBM50243706(2-(4-ethoxybenzyl)-N,N-diethyl-1-((tetrahydro-2H-p...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at cloned human CB2 receptor in Sf9 cells assessed as stimulation of [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244317BDBM50244317(2-(4-ethoxybenzyl)-1-(cyclopentylmethyl)-N,N-dieth...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244351BDBM50244351(2-(4-ethoxybenzyl)-1-benzyl-N,N-diethyl-1H-benzo[d...)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at cloned human CB2 receptor in Sf9 cells assessed as stimulation of [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244319BDBM50244319(1-adamantan-1-ylmethyl-2-(4-ethoxy-benzyl)-1H-benz...)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at cloned human CB2 receptor in Sf9 cells assessed as stimulation of [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244316BDBM50244316(2-(4-ethoxybenzyl)-1-(cyclobutylmethyl)-N,N-diethy...)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at cloned human CB2 receptor in Sf9 cells assessed as stimulation of [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 60994BDBM60994((10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tet...)
Affinity DataEC50:  1.5nMAssay Description:Agonist activity at cloned human CB2 receptor in Sf9 cells assessed as stimulation of [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244316BDBM50244316(2-(4-ethoxybenzyl)-1-(cyclobutylmethyl)-N,N-diethy...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244180BDBM50244180(1-(2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-1H-ben...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at cloned human CB2 receptor in Sf9 cells assessed as stimulation of [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244098BDBM50244098(2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-N,N-bis(2...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at cloned human CB2 receptor in Sf9 cells assessed as stimulation of [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244060BDBM50244060(2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-N,N-dipro...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at cloned human CB2 receptor in Sf9 cells assessed as stimulation of [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244277BDBM50244277(2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-N,N-dieth...)
Affinity DataEC50:  2.10nMAssay Description:Agonist activity at cloned human CB2 receptor in Sf9 cells assessed as stimulation of [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50243861BDBM50243861((R)-2-(4-ethoxybenzyl)-N,N-diethyl-1-((1-methylpip...)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at cloned human CB2 receptor in Sf9 cells assessed as stimulation of [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50243961BDBM50243961(2-(4-isopropoxybenzyl)-N,N-diethyl-1-isopentyl-1H-...)
Affinity DataEC50:  2.40nMAssay Description:Agonist activity at cloned human CB2 receptor in Sf9 cells assessed as stimulation of [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244178BDBM50244178(N-(2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-1H-ben...)
Affinity DataEC50:  2.60nMAssay Description:Agonist activity at cloned human CB2 receptor in Sf9 cells assessed as stimulation of [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244140BDBM50244140(N-(2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-1H-ben...)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at cloned human CB2 receptor in Sf9 cells assessed as stimulation of [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244319BDBM50244319(1-adamantan-1-ylmethyl-2-(4-ethoxy-benzyl)-1H-benz...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244060BDBM50244060(2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-N,N-dipro...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244276BDBM50244276(2-(4-ethoxybenzyl)-N,N-diethyl-1-isopentyl-1H-benz...)
Affinity DataEC50:  2.90nMAssay Description:Agonist activity at cloned human CB2 receptor in Sf9 cells assessed as stimulation of [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 60994BDBM60994((10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tet...)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244096BDBM50244096((2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-1H-benzo...)
Affinity DataEC50:  3nMAssay Description:Agonist activity at cloned human CB2 receptor in Sf9 cells assessed as stimulation of [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244059BDBM50244059(2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-N-methyl-...)
Affinity DataEC50:  3.20nMAssay Description:Agonist activity at cloned human CB2 receptor in Sf9 cells assessed as stimulation of [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244010BDBM50244010(2-(4-phenoxybenzyl)-N,N-diethyl-1-isopentyl-1H-ben...)
Affinity DataEC50:  3.20nMAssay Description:Agonist activity at cloned human CB2 receptor in Sf9 cells assessed as stimulation of [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50243705BDBM50243705(2-(4-ethoxybenzyl)-N,N-diethyl-1-(furan-2-ylmethyl...)
Affinity DataEC50:  3.30nMAssay Description:Agonist activity at cloned human CB2 receptor in Sf9 cells assessed as stimulation of [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244214BDBM50244214(N-(2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-1H-ben...)
Affinity DataEC50:  3.30nMAssay Description:Agonist activity at cloned human CB2 receptor in Sf9 cells assessed as stimulation of [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50243862BDBM50243862((S)-2-(4-ethoxybenzyl)-N,N-diethyl-1-((1-methylpyr...)
Affinity DataEC50:  3.40nMAssay Description:Agonist activity at cloned human CB2 receptor in Sf9 cells assessed as stimulation of [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244318BDBM50244318(2-(4-ethoxybenzyl)-1-(cyclohexylmethyl)-N,N-diethy...)
Affinity DataKi:  3.70nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50243706BDBM50243706(2-(4-ethoxybenzyl)-N,N-diethyl-1-((tetrahydro-2H-p...)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244140BDBM50244140(N-(2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-1H-ben...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244214BDBM50244214(N-(2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-1H-ben...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244277BDBM50244277(2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-N,N-dieth...)
Affinity DataKi:  4.10nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244097BDBM50244097(2-(4-ethoxybenzyl)-N-cyclohexyl-1-(cyclopropylmeth...)
Affinity DataEC50:  4.20nMAssay Description:Agonist activity at cloned human CB2 receptor in Sf9 cells assessed as stimulation of [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50243961BDBM50243961(2-(4-isopropoxybenzyl)-N,N-diethyl-1-isopentyl-1H-...)
Affinity DataKi:  4.5nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244276BDBM50244276(2-(4-ethoxybenzyl)-N,N-diethyl-1-isopentyl-1H-benz...)
Affinity DataKi:  4.5nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50243707BDBM50243707((S)-2-(4-ethoxybenzyl)-N,N-diethyl-1-((tetrahydrof...)
Affinity DataEC50:  4.80nMAssay Description:Agonist activity at cloned human CB2 receptor in Sf9 cells assessed as stimulation of [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244010BDBM50244010(2-(4-phenoxybenzyl)-N,N-diethyl-1-isopentyl-1H-ben...)
Affinity DataKi:  4.90nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244353BDBM50244353(2-(4-ethoxybenzyl)-N,N-diethyl-1-(pyridin-4-ylmeth...)
Affinity DataEC50:  5nMAssay Description:Agonist activity at cloned human CB2 receptor in Sf9 cells assessed as stimulation of [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244178BDBM50244178(N-(2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-1H-ben...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244098BDBM50244098(2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-N,N-bis(2...)
Affinity DataKi:  5.60nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244181BDBM50244181(1-(2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-1H-ben...)
Affinity DataKi:  5.70nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244180BDBM50244180(1-(2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-1H-ben...)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244061BDBM50244061((2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-1H-benzo...)
Affinity DataEC50:  6.20nMAssay Description:Agonist activity at cloned human CB2 receptor in Sf9 cells assessed as stimulation of [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244181BDBM50244181(1-(2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-1H-ben...)
Affinity DataEC50:  6.40nMAssay Description:Agonist activity at cloned human CB2 receptor in Sf9 cells assessed as stimulation of [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244096BDBM50244096((2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-1H-benzo...)
Affinity DataKi:  6.90nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50243913BDBM50243913(2-(4-methoxybenzyl)-N,N-diethyl-1-isopentyl-1H-ben...)
Affinity DataEC50:  7.30nMAssay Description:Agonist activity at cloned human CB2 receptor in Sf9 cells assessed as stimulation of [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50244059BDBM50244059(2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-N-methyl-...)
Affinity DataKi:  7.60nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50243708BDBM50243708((R)-2-(4-ethoxybenzyl)-N,N-diethyl-1-((tetrahydrof...)
Affinity DataEC50:  8.30nMAssay Description:Agonist activity at cloned human CB2 receptor in Sf9 cells assessed as stimulation of [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50243861BDBM50243861((R)-2-(4-ethoxybenzyl)-N,N-diethyl-1-((1-methylpip...)
Affinity DataKi:  8.90nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50243705BDBM50243705(2-(4-ethoxybenzyl)-N,N-diethyl-1-(furan-2-ylmethyl...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
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