Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50026178
TargetMitogen-activated protein kinase 8(Human)
Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50270672(N1-(1-(4-(1H-Indazol-3-yl)phenyl)-16-methyl-1,7,10...)
Affinity DataIC50: 20nMAssay Description:Displacement of biotin-labeled pep-JIP1 from GST fused JNK1 by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50270672(N1-(1-(4-(1H-Indazol-3-yl)phenyl)-16-methyl-1,7,10...)
Affinity DataIC50: 295nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50270641(N-(4-(1-Oxo-2,2,6,6-tetramethylpiperidin-4-ylamino...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50270670(4-(4-(1H-Indazol-3-yl)benzamido)butanoic acid | CH...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50270671(Ac-RPTTLNL-OH | CHEMBL504550)
Affinity DataIC50: 5.30E+4nMAssay Description:Displacement of biotin-labeled pep-JIP1 from GST fused JNK1 by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed