Compile Data Set for Download or QSAR
Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 50038569
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261673((3R,6S,9S,12R,15S)-12-benzyl-9-(3-carbamimidamidop...)
Affinity DataEC50:  810nMAssay Description:Agonist activity at human melanocortin 1 receptor expressed in HEK293 cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261672((3R,6S,9S,12R,15S)-12-benzyl-9-(3-carbamimidamidop...)
Affinity DataEC50:  76nMAssay Description:Agonist activity at human melanocortin 1 receptor expressed in HEK293 cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261681((3R,6R,9S,12R,15S)-12-benzyl-9-(3-carbamimidamidop...)
Affinity DataEC50:  330nMAssay Description:Agonist activity at human melanocortin 3 receptor expressed in HEK293 cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261670((3R,6S,9S,12R,15S)-12-benzyl-9-(3-carbamimidamidop...)
Affinity DataEC50:  37nMAssay Description:Agonist activity at human melanocortin 4 receptor expressed in HEK293 cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261670((3R,6S,9S,12R,15S)-12-benzyl-9-(3-carbamimidamidop...)
Affinity DataEC50:  44nMAssay Description:Agonist activity at human melanocortin 5 receptor expressed in HEK293 cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261677((3R,6S,9S,12S,15S)-9-(3-carbamimidamidopropyl)-15-...)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human melanocortin 3 receptor expressed in HEK293 cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261678((3R,6S,9S,12S,15S)-12-[(4-aminophenyl)methyl]-9-(3...)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human melanocortin 1 receptor expressed in HEK293 cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261670((3R,6S,9S,12R,15S)-12-benzyl-9-(3-carbamimidamidop...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human melanocortin 1 receptor expressed in HEK293 cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261676((3R,6S,9S,12R,15S)-9-(3-carbamimidamidopropyl)-15-...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human melanocortin 1 receptor expressed in HEK293 cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261671((3R,6S,9S,12R)-12-benzyl-9-(3-carbamimidamidopropy...)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human melanocortin 1 receptor expressed in HEK293 cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261682((3R,6S,9S,12R,15S)-12-benzyl-9-(3-carbamimidamidop...)
Affinity DataEC50:  71nMAssay Description:Agonist activity at human melanocortin 1 receptor expressed in HEK293 cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261678((3R,6S,9S,12S,15S)-12-[(4-aminophenyl)methyl]-9-(3...)
Affinity DataEC50:  150nMAssay Description:Agonist activity at human melanocortin 3 receptor expressed in HEK293 cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50377916(CHEMBL552520 | CHEMBL553202)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human melanocortin 3 receptor expressed in HEK293 cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261671((3R,6S,9S,12R)-12-benzyl-9-(3-carbamimidamidopropy...)
Affinity DataEC50: >5.00E+3nMAssay Description:Agonist activity at human melanocortin 3 receptor expressed in HEK293 cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261670((3R,6S,9S,12R,15S)-12-benzyl-9-(3-carbamimidamidop...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human melanocortin 3 receptor expressed in HEK293 cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261684((3R,6R,9S,12R,15S)-12-benzyl-9-(3-carbamimidamidop...)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human melanocortin 1 receptor expressed in HEK293 cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261673((3R,6S,9S,12R,15S)-12-benzyl-9-(3-carbamimidamidop...)
Affinity DataEC50: >4.00E+3nMAssay Description:Agonist activity at human melanocortin 3 receptor expressed in HEK293 cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261682((3R,6S,9S,12R,15S)-12-benzyl-9-(3-carbamimidamidop...)
Affinity DataEC50:  56nMAssay Description:Agonist activity at human melanocortin 3 receptor expressed in HEK293 cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261670((3R,6S,9S,12R,15S)-12-benzyl-9-(3-carbamimidamidop...)
Affinity DataIC50: 3.70nMAssay Description:Displacement of [125I]-[Nle4, D-Phe7]alpha-MSH from human melanocortin 1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261673((3R,6S,9S,12R,15S)-12-benzyl-9-(3-carbamimidamidop...)
Affinity DataIC50: 38nMAssay Description:Displacement of [125I]-[Nle4, D-Phe7]alpha-MSH from human melanocortin 5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261670((3R,6S,9S,12R,15S)-12-benzyl-9-(3-carbamimidamidop...)
Affinity DataIC50: 40nMAssay Description:Displacement of [125I]-[Nle4, D-Phe7]alpha-MSH from human melanocortin 3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261670((3R,6S,9S,12R,15S)-12-benzyl-9-(3-carbamimidamidop...)
Affinity DataIC50: 47nMAssay Description:Displacement of [125I]-[Nle4, D-Phe7]alpha-MSH from human melanocortin 4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50377916(CHEMBL552520 | CHEMBL553202)
Affinity DataIC50: 58nMAssay Description:Displacement of [125I]-[Nle4, D-Phe7]alpha-MSH from human melanocortin 5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261677((3R,6S,9S,12S,15S)-9-(3-carbamimidamidopropyl)-15-...)
Affinity DataIC50: 130nMAssay Description:Displacement of [125I]-[Nle4, D-Phe7]alpha-MSH from human melanocortin 5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261682((3R,6S,9S,12R,15S)-12-benzyl-9-(3-carbamimidamidop...)
Affinity DataIC50: 180nMAssay Description:Displacement of [125I]-[Nle4, D-Phe7]alpha-MSH from human melanocortin 1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261670((3R,6S,9S,12R,15S)-12-benzyl-9-(3-carbamimidamidop...)
Affinity DataIC50: 190nMAssay Description:Displacement of [125I]-[Nle4, D-Phe7]alpha-MSH from human melanocortin 5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261676((3R,6S,9S,12R,15S)-9-(3-carbamimidamidopropyl)-15-...)
Affinity DataIC50: 190nMAssay Description:Displacement of [125I]-[Nle4, D-Phe7]alpha-MSH from human melanocortin 3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261682((3R,6S,9S,12R,15S)-12-benzyl-9-(3-carbamimidamidop...)
Affinity DataIC50: 340nMAssay Description:Displacement of [125I]-[Nle4, D-Phe7]alpha-MSH from human melanocortin 5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50377916(CHEMBL552520 | CHEMBL553202)
Affinity DataIC50: 380nMAssay Description:Displacement of [125I]-[Nle4, D-Phe7]alpha-MSH from human melanocortin 3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261671((3R,6S,9S,12R)-12-benzyl-9-(3-carbamimidamidopropy...)
Affinity DataIC50: 560nMAssay Description:Displacement of [125I]-[Nle4, D-Phe7]alpha-MSH from human melanocortin 5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261682((3R,6S,9S,12R,15S)-12-benzyl-9-(3-carbamimidamidop...)
Affinity DataIC50: 610nMAssay Description:Displacement of [125I]-[Nle4, D-Phe7]alpha-MSH from human melanocortin 3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261676((3R,6S,9S,12R,15S)-9-(3-carbamimidamidopropyl)-15-...)
Affinity DataIC50: 760nMAssay Description:Displacement of [125I]-[Nle4, D-Phe7]alpha-MSH from human melanocortin 5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261676((3R,6S,9S,12R,15S)-9-(3-carbamimidamidopropyl)-15-...)
Affinity DataIC50: 760nMAssay Description:Displacement of [125I]-[Nle4, D-Phe7]alpha-MSH from human melanocortin 1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261682((3R,6S,9S,12R,15S)-12-benzyl-9-(3-carbamimidamidop...)
Affinity DataIC50: 1.00E+3nMAssay Description:Agonist activity at human melanocortin 4 receptor expressed in HEK293 cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261673((3R,6S,9S,12R,15S)-12-benzyl-9-(3-carbamimidamidop...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]-[Nle4, D-Phe7]alpha-MSH from human melanocortin 3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50377916(CHEMBL552520 | CHEMBL553202)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]-[Nle4, D-Phe7]alpha-MSH from human melanocortin 1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50377916(CHEMBL552520 | CHEMBL553202)
Affinity DataIC50: 1.00E+3nMAssay Description:Agonist activity at human melanocortin 4 receptor expressed in HEK293 cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261677((3R,6S,9S,12S,15S)-9-(3-carbamimidamidopropyl)-15-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]-[Nle4, D-Phe7]alpha-MSH from human melanocortin 3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261678((3R,6S,9S,12S,15S)-12-[(4-aminophenyl)methyl]-9-(3...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]-[Nle4, D-Phe7]alpha-MSH from human melanocortin 3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261683((3R,6S,9S,12R,15S)-6,12-dibenzyl-9-(3-carbamimidam...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]-[Nle4, D-Phe7]alpha-MSH from human melanocortin 1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261684((3R,6R,9S,12R,15S)-12-benzyl-9-(3-carbamimidamidop...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]-[Nle4, D-Phe7]alpha-MSH from human melanocortin 1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261671((3R,6S,9S,12R)-12-benzyl-9-(3-carbamimidamidopropy...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]-[Nle4, D-Phe7]alpha-MSH from human melanocortin 1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261679((3R,6S,9S,12R,15S)-9-(4-aminobutyl)-12-benzyl-15-(...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]-[Nle4, D-Phe7]alpha-MSH from human melanocortin 3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261684((3R,6R,9S,12R,15S)-12-benzyl-9-(3-carbamimidamidop...)
Affinity DataIC50: 1.00E+3nMAssay Description:Agonist activity at human melanocortin 4 receptor expressed in HEK293 cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50377916(CHEMBL552520 | CHEMBL553202)
Affinity DataIC50: 1.50E+3nMAssay Description:Displacement of [125I]-[Nle4, D-Phe7]alpha-MSH from human melanocortin 1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261677((3R,6S,9S,12S,15S)-9-(3-carbamimidamidopropyl)-15-...)
Affinity DataIC50: 2.00E+3nMAssay Description:Displacement of [125I]-[Nle4, D-Phe7]alpha-MSH from human melanocortin 1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261673((3R,6S,9S,12R,15S)-12-benzyl-9-(3-carbamimidamidop...)
Affinity DataIC50: 2.00E+3nMAssay Description:Displacement of [125I]-[Nle4, D-Phe7]alpha-MSH from human melanocortin 1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261684((3R,6R,9S,12R,15S)-12-benzyl-9-(3-carbamimidamidop...)
Affinity DataIC50: 2.00E+3nMAssay Description:Displacement of [125I]-[Nle4, D-Phe7]alpha-MSH from human melanocortin 5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261677((3R,6S,9S,12S,15S)-9-(3-carbamimidamidopropyl)-15-...)
Affinity DataIC50: 5.00E+3nMAssay Description:Agonist activity at human melanocortin 4 receptor expressed in HEK293 cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50261681((3R,6R,9S,12R,15S)-12-benzyl-9-(3-carbamimidamidop...)
Affinity DataIC50: 8.00E+3nMAssay Description:Displacement of [125I]-[Nle4, D-Phe7]alpha-MSH from human melanocortin 3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
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