Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50025959
TargetThyrotropin-releasing hormone receptor(Rat)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50072394(PROTIRELIN | ABBOTT-38579 | A-38579 | 1-[3-(1H-4-i...)
Affinity DataIC50: 23nMAssay Description:Displacement of [3H]3-methylhistidyl-TRH from rat recombinant TRHR2 expressed in HEK2935 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyrotropin-releasing hormone receptor(Rat)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50261331(20-Acetoxy-19-hydroxyspongia-13(16),14-diene | CHE...)
Affinity DataIC50: 2.30E+4nMAssay Description:Displacement of [3H]3-methylhistidyl-TRH from rat recombinant TRHR2 expressed in HEK2935 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyrotropin-releasing hormone receptor(Rat)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50261332(19-Acetoxy-20-hydroxyspongia-13(16),14-diene | CHE...)
Affinity DataIC50: 7.00E+4nMAssay Description:Displacement of [3H]3-methylhistidyl-TRH from rat recombinant TRHR2 expressed in HEK2935 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyrotropin-releasing hormone receptor(Rat)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50261333(19,20-Diacetoxyspongia-13(16),14-diene | CHEMBL466...)
Affinity DataIC50: 4.00E+5nMAssay Description:Displacement of [3H]3-methylhistidyl-TRH from rat recombinant TRHR2 expressed in HEK2935 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyrotropin-releasing hormone receptor(Rat)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50261358(19,20-Dihydroxyspongia-13(16),14-diene | CHEMBL512...)
Affinity DataIC50: 6.00E+5nMAssay Description:Displacement of [3H]3-methylhistidyl-TRH from rat recombinant TRHR2 expressed in HEK2935 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetThyrotropin-releasing hormone receptor(Rat)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50261359(spongia-13(16),14-diene | (3bR,5aS,9aS,9bR)-3b,6,6...)
Affinity DataIC50: 1.00E+6nMAssay Description:Displacement of [3H]3-methylhistidyl-TRH from rat recombinant TRHR2 expressed in HEK2935 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed