Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 3437
LigandPNGBDBM34017(CHEMBL104850 | phenylpropanoic acid derivative, 7)
Affinity DataIC50: 29nM EC50:  26nMpH: 7.4 T: 2°CAssay Description:Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2009
Entry Details Article
PubMed
LigandPNGBDBM33284(BMC164883 Compound 53 | phenylpropanoic acid deriv...)
Affinity DataIC50: 185nM EC50:  140nMpH: 7.4 T: 2°CAssay Description:Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2009
Entry Details Article
PubMed
LigandPNGBDBM34025(phenylpropanoic acid derivative, 40)
Affinity DataIC50: 255nM EC50:  102nMpH: 7.4 T: 2°CAssay Description:Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2009
Entry Details Article
PubMed
LigandPNGBDBM34018(phenylpropanoic acid derivative, 28)
Affinity DataIC50: 293nM EC50:  173nMpH: 7.4 T: 2°CAssay Description:Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2009
Entry Details Article
PubMed
LigandPNGBDBM34030(racemic | phenylpropanoic acid derivative, 56)
Affinity DataIC50: 587nM EC50:  1.80E+3nMpH: 7.4 T: 2°CAssay Description:Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2009
Entry Details Article
PubMed
LigandPNGBDBM34034(phenylpropanoic acid derivative, 66)
Affinity DataIC50: 1.60E+3nM EC50:  480nMpH: 7.4 T: 2°CAssay Description:Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2009
Entry Details Article
PubMed
LigandPNGBDBM34027(phenylpropanoic acid derivative, 44)
Affinity DataIC50: 2.00E+3nM EC50:  3.70E+3nMpH: 7.4 T: 2°CAssay Description:Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2009
Entry Details Article
PubMed
LigandPNGBDBM34020(racemic | phenylpropanoic acid derivative, 30)
Affinity DataIC50: 2.20E+3nM EC50:  2.50E+3nMpH: 7.4 T: 2°CAssay Description:Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2009
Entry Details Article
PubMed
LigandPNGBDBM34026(phenylpropanoic acid derivative, 41)
Affinity DataIC50: 2.60E+3nM EC50:  2.60E+3nMpH: 7.4 T: 2°CAssay Description:Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2009
Entry Details Article
PubMed
LigandPNGBDBM34021(racemic | phenylpropanoic acid derivative, 31)
Affinity DataIC50: 2.80E+3nM EC50:  1.30E+4nMpH: 7.4 T: 2°CAssay Description:Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2009
Entry Details Article
PubMed
LigandPNGBDBM34031(racemic | phenylpropanoic acid derivative, 57)
Affinity DataIC50: 2.80E+3nM EC50:  4.00E+3nMpH: 7.4 T: 2°CAssay Description:Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2009
Entry Details Article
PubMed
LigandPNGBDBM34028(phenylpropanoic acid derivative, 54)
Affinity DataIC50: 3.10E+3nM EC50:  2.30E+3nMpH: 7.4 T: 2°CAssay Description:Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2009
Entry Details Article
PubMed
LigandPNGBDBM33296(BMC164883 Compound 58 | racemic | phenylpropanoic ...)
Affinity DataIC50: 4.00E+3nM EC50:  3.90E+3nMpH: 7.4 T: 2°CAssay Description:Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2009
Entry Details Article
PubMed
LigandPNGBDBM34033(phenylpropanoic acid derivative, 60)
Affinity DataIC50: 1.10E+4nM EC50:  3.60E+3nMpH: 7.4 T: 2°CAssay Description:Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2009
Entry Details Article
PubMed
LigandPNGBDBM34024(phenylpropanoic acid derivative, 36)
Affinity DataIC50: 1.20E+4nM EC50:  492nMpH: 7.4 T: 2°CAssay Description:Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2009
Entry Details Article
PubMed
LigandPNGBDBM34023(phenylpropanoic acid derivative, 33)
Affinity DataIC50: 1.20E+4nM EC50:  2.00E+3nMpH: 7.4 T: 2°CAssay Description:Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2009
Entry Details Article
PubMed
LigandPNGBDBM34029(racemic | phenylpropanoic acid derivative, 55)
Affinity DataIC50: 2.20E+4nM EC50:  3.90E+3nMpH: 7.4 T: 2°CAssay Description:Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2009
Entry Details Article
PubMed
LigandPNGBDBM34019(racemic | phenylpropanoic acid derivative, 29)
Affinity DataIC50: 2.60E+4nM EC50:  4.50E+3nMpH: 7.4 T: 2°CAssay Description:Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2009
Entry Details Article
PubMed
LigandPNGBDBM34032(phenylpropanoic acid derivative, 59)
Affinity DataIC50: 2.80E+4nM EC50:  1.20E+3nMpH: 7.4 T: 2°CAssay Description:Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2009
Entry Details Article
PubMed
LigandPNGBDBM34035(phenylpropanoic acid derivative, 74)
Affinity DataIC50: 5.00E+4nM EC50:  9.00E+3nMpH: 7.4 T: 2°CAssay Description:Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2009
Entry Details Article
PubMed
LigandPNGBDBM34022(racemic | phenylpropanoic acid derivative, 32)
Affinity DataIC50: 5.30E+4nM EC50:  9.00E+3nMpH: 7.4 T: 2°CAssay Description:Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2009
Entry Details Article
PubMed
LigandPNGBDBM34036(phenylpropanoic acid derivative, 75)
Affinity DataIC50: 1.00E+5nM EC50:  7.00E+3nMpH: 7.4 T: 2°CAssay Description:Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2009
Entry Details Article
PubMed
LigandPNGBDBM34037(phenylpropanoic acid derivative, 76)
Affinity DataIC50: 1.00E+5nM EC50: >3.00E+4nMpH: 7.4 T: 2°CAssay Description:Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2009
Entry Details Article
PubMed