Compile Data Set for Download or QSAR
Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 50025806
TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266569(Methyl 7-(2-(5-methyl-2-m-tolyloxazol-4-yl)ethoxy)...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266531(Methyl 7-(2-(2-(4-methoxyphenyl)-5-methyloxazol-4-...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266532(Methyl 7-(2-(2-(4-methoxyphenyl)-5-methyloxazol-4-...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266533(Methyl 7-(2-(2-(3-methoxyphenyl)-5-methyloxazol-4-...)
Affinity DataEC50:  350nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266534(Methyl 7-(2-(2-(3-methoxyphenyl)-5-methyloxazol-4-...)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266548(Methyl 7-(2-(2-(4-tert-butylphenyl)-5-methyloxazol...)
Affinity DataEC50:  1.74E+3nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266549(Methyl 7-(2-(2-(4-tert-butylphenyl)-5-methyloxazol...)
Affinity DataEC50:  250nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266550(Methyl 7-(2-(5-methyl-2-p-tolyloxazol-4-yl)ethoxy)...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266551(Methyl 7-(2-(5-methyl-2-p-tolyloxazol-4-yl)ethoxy)...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266568(Methyl 7-(2-(5-methyl-2-m-tolyloxazol-4-yl)ethoxy)...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266501(Methyl 7-(2-(2-(biphenyl-4-yl)-5-methyloxazol-4-yl...)
Affinity DataEC50:  1.12E+3nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266570(Methyl 7-(2-(5-methyl-2-(3-(trifluoromethyl)phenyl...)
Affinity DataEC50:  420nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266571(Methyl 7-(2-(5-methyl-2-(3-(trifluoromethyl)phenyl...)
Affinity DataEC50:  160nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266595(Methyl 7-(2-(2-(4-fluorophenyl)-5-methyloxazol-4-y...)
Affinity DataEC50:  1.62E+3nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266596(Methyl 7-(2-(2-(4-fluorophenyl)-5-methyloxazol-4-y...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266597(Methyl 7-(2-(2-(3-fluorophenyl)-5-methyloxazol-4-y...)
Affinity DataEC50:  960nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266598(Methyl 7-(2-(2-(3-fluorophenyl)-5-methyloxazol-4-y...)
Affinity DataEC50:  170nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266609(Methyl 7-(2-(5-methyl-2-(3-nitrophenyl)oxazol-4-yl...)
Affinity DataEC50:  3.55E+3nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50240768(methyl 7-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-...)
Affinity DataEC50:  130nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM28681(cid_5281055 | [3H]rosiglitazone | CHEMBL121 | ROSI...)
Affinity DataEC50:  20nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266569(Methyl 7-(2-(5-methyl-2-m-tolyloxazol-4-yl)ethoxy)...)
Affinity DataEC50:  1.55E+3nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266501(Methyl 7-(2-(2-(biphenyl-4-yl)-5-methyloxazol-4-yl...)
Affinity DataEC50:  910nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266531(Methyl 7-(2-(2-(4-methoxyphenyl)-5-methyloxazol-4-...)
Affinity DataEC50:  5.25E+3nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266532(Methyl 7-(2-(2-(4-methoxyphenyl)-5-methyloxazol-4-...)
Affinity DataEC50:  1.74E+3nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266533(Methyl 7-(2-(2-(3-methoxyphenyl)-5-methyloxazol-4-...)
Affinity DataEC50:  1.62E+3nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266534(Methyl 7-(2-(2-(3-methoxyphenyl)-5-methyloxazol-4-...)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266548(Methyl 7-(2-(2-(4-tert-butylphenyl)-5-methyloxazol...)
Affinity DataEC50:  2.29E+3nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266549(Methyl 7-(2-(2-(4-tert-butylphenyl)-5-methyloxazol...)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266550(Methyl 7-(2-(5-methyl-2-p-tolyloxazol-4-yl)ethoxy)...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266551(Methyl 7-(2-(5-methyl-2-p-tolyloxazol-4-yl)ethoxy)...)
Affinity DataEC50:  910nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266500(Methyl 7-(2-(2-(biphenyl-4-yl)-5-methyloxazol-4-yl...)
Affinity DataEC50:  1.23E+3nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266570(Methyl 7-(2-(5-methyl-2-(3-(trifluoromethyl)phenyl...)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266571(Methyl 7-(2-(5-methyl-2-(3-(trifluoromethyl)phenyl...)
Affinity DataEC50:  170nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266595(Methyl 7-(2-(2-(4-fluorophenyl)-5-methyloxazol-4-y...)
Affinity DataEC50:  70nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266596(Methyl 7-(2-(2-(4-fluorophenyl)-5-methyloxazol-4-y...)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266597(Methyl 7-(2-(2-(3-fluorophenyl)-5-methyloxazol-4-y...)
Affinity DataEC50:  1.29E+3nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266598(Methyl 7-(2-(2-(3-fluorophenyl)-5-methyloxazol-4-y...)
Affinity DataEC50:  720nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50240768(methyl 7-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-...)
Affinity DataEC50:  140nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM24566(JMC515449 Compound 1 | Wyeth 14,643 | 2-({4-chloro...)
Affinity DataEC50:  1.20E+4nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266500(Methyl 7-(2-(2-(biphenyl-4-yl)-5-methyloxazol-4-yl...)
Affinity DataEC50:  1.26E+3nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed