Compile Data Set for Download or QSAR
Report error Found 136 Enz. Inhib. hit(s) with all data for entry = 50038322
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374829(CHEMBL255629)
Affinity DataIC50: 30nMAssay Description:Antagonist activity at human CCR1 receptor expressed in THP1 cells assessed as human MIP-1-alpha-stimulated intracellular calcium level by FLIPR assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374816(CHEMBL256404)
Affinity DataIC50: 30nMAssay Description:Antagonist activity at human CCR1 receptor expressed in THP1 cells assessed as human MIP-1-alpha-stimulated intracellular calcium level by FLIPR assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374831(CHEMBL429419)
Affinity DataIC50: 40nMAssay Description:Antagonist activity at human CCR1 receptor expressed in THP1 cells assessed as human MIP-1-alpha-stimulated intracellular calcium level by FLIPR assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374806(CHEMBL269957)
Affinity DataIC50: 40nMAssay Description:Antagonist activity at human CCR1 receptor expressed in THP1 cells assessed as human MIP-1-alpha-stimulated intracellular calcium level by FLIPR assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374818(CHEMBL258065)
Affinity DataIC50: 50nMAssay Description:Antagonist activity at human CCR1 receptor expressed in THP1 cells assessed as human MIP-1-alpha-stimulated intracellular calcium level by FLIPR assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374807(CHEMBL272097)
Affinity DataIC50: 70nMAssay Description:Antagonist activity at human CCR1 receptor expressed in THP1 cells assessed as human MIP-1-alpha-stimulated intracellular calcium level by FLIPR assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374829(CHEMBL255629)
Affinity DataIC50: 80nMAssay Description:Displacement of [125I]MIP1-alpha from human CCR1 receptor expressed in THP1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374814(CHEMBL256888)
Affinity DataIC50: 80nMAssay Description:Antagonist activity at human CCR1 receptor expressed in THP1 cells assessed as human MIP-1-alpha-stimulated intracellular calcium level by FLIPR assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374808(CHEMBL272523)
Affinity DataIC50: 84nMAssay Description:Antagonist activity at human CCR1 receptor expressed in THP1 cells assessed as human MIP-1-alpha-stimulated intracellular calcium level by FLIPR assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374831(CHEMBL429419)
Affinity DataIC50: 90nMAssay Description:Displacement of [125I]MIP1-alpha from human CCR1 receptor expressed in THP1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374837(CHEMBL403728)
Affinity DataIC50: 90nMAssay Description:Displacement of [125I]MIP1-alpha from human CCR1 receptor expressed in THP1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374837(CHEMBL403728)
Affinity DataIC50: 90nMAssay Description:Antagonist activity at human CCR1 receptor expressed in THP1 cells assessed as human MIP-1-alpha-stimulated intracellular calcium level by FLIPR assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374804(CHEMBL270631)
Affinity DataIC50: 90nMAssay Description:Antagonist activity at human CCR1 receptor expressed in THP1 cells assessed as human MIP-1-alpha-stimulated intracellular calcium level by FLIPR assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374812(CHEMBL256821)
Affinity DataIC50: 100nMAssay Description:Antagonist activity at human CCR1 receptor expressed in THP1 cells assessed as human MIP-1-alpha-stimulated intracellular calcium level by FLIPR assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374830(CHEMBL257509)
Affinity DataIC50: 100nMAssay Description:Antagonist activity at human CCR1 receptor expressed in THP1 cells assessed as human MIP-1-alpha-stimulated intracellular calcium level by FLIPR assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374806(CHEMBL269957)
Affinity DataIC50: 110nMAssay Description:Displacement of [125I]MIP1-alpha from human CCR1 receptor expressed in THP1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374823(CHEMBL255338)
Affinity DataIC50: 110nMAssay Description:Antagonist activity at human CCR1 receptor expressed in THP1 cells assessed as human MIP-1-alpha-stimulated intracellular calcium level by FLIPR assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374846(CHEMBL256272)
Affinity DataIC50: 120nMAssay Description:Antagonist activity at human CCR1 receptor expressed in THP1 cells assessed as human MIP-1-alpha-stimulated intracellular calcium level by FLIPR assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374817(CHEMBL258064)
Affinity DataIC50: 120nMAssay Description:Antagonist activity at human CCR1 receptor expressed in THP1 cells assessed as human MIP-1-alpha-stimulated intracellular calcium level by FLIPR assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374855(CHEMBL404465)
Affinity DataIC50: 130nMAssay Description:Antagonist activity at human CCR1 receptor expressed in THP1 cells assessed as human MIP-1-alpha-stimulated intracellular calcium level by FLIPR assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374833(CHEMBL270253)
Affinity DataIC50: 130nMAssay Description:Antagonist activity at human CCR1 receptor expressed in THP1 cells assessed as human MIP-1-alpha-stimulated intracellular calcium level by FLIPR assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374805(CHEMBL429591)
Affinity DataIC50: 140nMAssay Description:Displacement of [125I]MIP1-alpha from human CCR1 receptor expressed in THP1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374816(CHEMBL256404)
Affinity DataIC50: 150nMAssay Description:Displacement of [125I]MIP1-alpha from human CCR1 receptor expressed in THP1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374807(CHEMBL272097)
Affinity DataIC50: 160nMAssay Description:Displacement of [125I]MIP1-alpha from human CCR1 receptor expressed in THP1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374860(CHEMBL258359)
Affinity DataIC50: 180nMAssay Description:Antagonist activity at human CCR1 receptor expressed in THP1 cells assessed as human MIP-1-alpha-stimulated intracellular calcium level by FLIPR assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374858(CHEMBL271903)
Affinity DataIC50: 180nMAssay Description:Antagonist activity at human CCR1 receptor expressed in THP1 cells assessed as human MIP-1-alpha-stimulated intracellular calcium level by FLIPR assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374835(CHEMBL404033)
Affinity DataIC50: 180nMAssay Description:Antagonist activity at human CCR1 receptor expressed in THP1 cells assessed as human MIP-1-alpha-stimulated intracellular calcium level by FLIPR assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374866(CHEMBL270433)
Affinity DataIC50: 180nMAssay Description:Antagonist activity at human CCR1 receptor expressed in THP1 cells assessed as human MIP-1-alpha-stimulated intracellular calcium level by FLIPR assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374819(CHEMBL258361)
Affinity DataIC50: 190nMAssay Description:Antagonist activity at human CCR1 receptor expressed in THP1 cells assessed as human MIP-1-alpha-stimulated intracellular calcium level by FLIPR assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374833(CHEMBL270253)
Affinity DataIC50: 200nMAssay Description:Displacement of [125I]MIP1-alpha from human CCR1 receptor expressed in THP1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374815(CHEMBL256889)
Affinity DataIC50: 210nMAssay Description:Antagonist activity at human CCR1 receptor expressed in THP1 cells assessed as human MIP-1-alpha-stimulated intracellular calcium level by FLIPR assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374846(CHEMBL256272)
Affinity DataIC50: 220nMAssay Description:Displacement of [125I]MIP1-alpha from human CCR1 receptor expressed in THP1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374822(CHEMBL257452)
Affinity DataIC50: 230nMAssay Description:Antagonist activity at human CCR1 receptor expressed in THP1 cells assessed as human MIP-1-alpha-stimulated intracellular calcium level by FLIPR assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374822(CHEMBL257452)
Affinity DataIC50: 240nMAssay Description:Displacement of [125I]MIP1-alpha from human CCR1 receptor expressed in THP1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374818(CHEMBL258065)
Affinity DataIC50: 250nMAssay Description:Displacement of [125I]MIP1-alpha from human CCR1 receptor expressed in THP1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374847(CHEMBL402827)
Affinity DataIC50: 270nMAssay Description:Antagonist activity at human CCR1 receptor expressed in THP1 cells assessed as human MIP-1-alpha-stimulated intracellular calcium level by FLIPR assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374845(CHEMBL256271)
Affinity DataIC50: 280nMAssay Description:Antagonist activity at human CCR1 receptor expressed in THP1 cells assessed as human MIP-1-alpha-stimulated intracellular calcium level by FLIPR assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374826(CHEMBL270863)
Affinity DataIC50: 280nMAssay Description:Antagonist activity at human CCR1 receptor expressed in THP1 cells assessed as human MIP-1-alpha-stimulated intracellular calcium level by FLIPR assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374804(CHEMBL270631)
Affinity DataIC50: 300nMAssay Description:Displacement of [125I]MIP1-alpha from human CCR1 receptor expressed in THP1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374845(CHEMBL256271)
Affinity DataIC50: 320nMAssay Description:Displacement of [125I]MIP1-alpha from human CCR1 receptor expressed in THP1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374838(CHEMBL256887)
Affinity DataIC50: 330nMAssay Description:Antagonist activity at human CCR1 receptor expressed in THP1 cells assessed as human MIP-1-alpha-stimulated intracellular calcium level by FLIPR assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374819(CHEMBL258361)
Affinity DataIC50: 350nMAssay Description:Displacement of [125I]MIP1-alpha from human CCR1 receptor expressed in THP1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374823(CHEMBL255338)
Affinity DataIC50: 350nMAssay Description:Displacement of [125I]MIP1-alpha from human CCR1 receptor expressed in THP1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374824(CHEMBL258360)
Affinity DataIC50: 350nMAssay Description:Antagonist activity at human CCR1 receptor expressed in THP1 cells assessed as human MIP-1-alpha-stimulated intracellular calcium level by FLIPR assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374830(CHEMBL257509)
Affinity DataIC50: 360nMAssay Description:Displacement of [125I]MIP1-alpha from human CCR1 receptor expressed in THP1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374825(CHEMBL411477)
Affinity DataIC50: 360nMAssay Description:Antagonist activity at human CCR1 receptor expressed in THP1 cells assessed as human MIP-1-alpha-stimulated intracellular calcium level by FLIPR assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374836(CHEMBL269956)
Affinity DataIC50: 370nMAssay Description:Displacement of [125I]MIP1-alpha from human CCR1 receptor expressed in THP1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374813(CHEMBL404732)
Affinity DataIC50: 370nMAssay Description:Antagonist activity at human CCR1 receptor expressed in THP1 cells assessed as human MIP-1-alpha-stimulated intracellular calcium level by FLIPR assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374812(CHEMBL256821)
Affinity DataIC50: 380nMAssay Description:Displacement of [125I]MIP1-alpha from human CCR1 receptor expressed in THP1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50374821(CHEMBL270564)
Affinity DataIC50: 385nMAssay Description:Antagonist activity at human CCR1 receptor expressed in THP1 cells assessed as human MIP-1-alpha-stimulated intracellular calcium level by FLIPR assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
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