Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50025773
TargetBaculoviral IAP repeat-containing protein 2(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50251287(N-[(R)-3-Hydroxycarbamoyl-2-pentylpropanoyl]-L-ala...)
Affinity DataIC50: 530nMAssay Description:Promotion of flag-tagged cIAP1 degradation in human HT1080 cells assessed as decrease in cIAPI production after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 2(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50251279((S)-methyl 2-((2S,3R)-3-amino-2-hydroxy-4-phenylbu...)
Affinity DataIC50: 690nMAssay Description:Promotion of flag-tagged cIAP1 degradation in human HT1080 cells assessed as decrease in cIAPI production after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 2(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50251296(N-[(R)-3-Hydroxycarbamoyl-2-pentylpropanoyl]-L-phe...)
Affinity DataIC50: 840nMAssay Description:Promotion of flag-tagged cIAP1 degradation in human HT1080 cells assessed as decrease in cIAPI production after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 2(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50251280(N-[(R)-3-Hydroxycarbamoyl-2-pentylpropanoyl]-L-leu...)
Affinity DataIC50: 1.06E+3nMAssay Description:Promotion of flag-tagged cIAP1 degradation in human HT1080 cells assessed as decrease in cIAPI production after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 2(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50251288(N-[(R)-3-Hydroxycarbamoyl-2-pentylpropanoyl]-L-val...)
Affinity DataIC50: 1.25E+3nMAssay Description:Promotion of flag-tagged cIAP1 degradation in human HT1080 cells assessed as decrease in cIAPI production after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 2(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50251286(N-[(R)-3-Hydroxycarbamoyl-2-pentylpropanoyl]glycin...)
Affinity DataIC50: 1.54E+3nMAssay Description:Promotion of flag-tagged cIAP1 degradation in human HT1080 cells assessed as decrease in cIAPI production after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 2(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50251297(N-[(R)-3-Hydroxycarbamoyl-2-butylaminopropanoyl]-L...)
Affinity DataIC50: 4.69E+3nMAssay Description:Promotion of flag-tagged cIAP1 degradation in human HT1080 cells assessed as decrease in cIAPI production after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 2(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50251298(N-[(R)-3-Hydroxycarbamoyl-2-dibutylaminopropanyl]-...)
Affinity DataIC50: 9.20E+3nMAssay Description:Promotion of flag-tagged cIAP1 degradation in human HT1080 cells assessed as decrease in cIAPI production after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 2(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50251282(N-[(S)-3-Hydroxycarbamoyl-2-pentylpropanoyl]-L-leu...)
Affinity DataIC50: 1.21E+4nMAssay Description:Promotion of flag-tagged cIAP1 degradation in human HT1080 cells assessed as decrease in cIAPI production after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 2(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50251285(N-[N-Hydroxysuccinamiyl]-L-leucine methylester | C...)
Affinity DataIC50: 1.99E+4nMAssay Description:Promotion of flag-tagged cIAP1 degradation in human HT1080 cells assessed as decrease in cIAPI production after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 2(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50251295(N-[(R)-3-Hydroxycarbamoyl-2-pentylpropanoyl]-L-ter...)
Affinity DataIC50: 2.00E+4nMAssay Description:Promotion of flag-tagged cIAP1 degradation in human HT1080 cells assessed as decrease in cIAPI production after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 2(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50251283(N-[(R)-3-Hydroxycarbamoyl-2-ethylpropanoyl]-L-leuc...)
Affinity DataIC50: 2.41E+4nMAssay Description:Promotion of flag-tagged cIAP1 degradation in human HT1080 cells assessed as decrease in cIAPI production after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 2(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50251284(N-[(R)-3-Hydroxycarbamoyl-2-benzylpropanyl]-L-leuc...)
Affinity DataIC50: 4.52E+4nMAssay Description:Promotion of flag-tagged cIAP1 degradation in human HT1080 cells assessed as decrease in cIAPI production after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed