Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50038383
TargetMu-type opioid receptor(Guinea pig)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50375696(CHEMBL269842)
Affinity DataIC50: 50.6nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig assessed as inhibition of electrically evoked-contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50375694(CHEMBL244265)
Affinity DataIC50: 1.92E+3nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig assessed as inhibition of electrically evoked-contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50375696(CHEMBL269842)
Affinity DataIC50: 5.18E+3nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically evoked-contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50375695(CHEMBL270984)
Affinity DataIC50: 1.00E+4nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig assessed as inhibition of electrically evoked-contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50375695(CHEMBL270984)
Affinity DataKi:  0.0190nMAssay Description:Displacement of [3H]deltorphin2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50375694(CHEMBL244265)
Affinity DataKi:  0.172nMAssay Description:Displacement of [3H]deltorphin2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50375696(CHEMBL269842)
Affinity DataKi:  0.248nMAssay Description:Displacement of [3H]deltorphin2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50375695(CHEMBL270984)
Affinity DataKi:  2.75nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50375696(CHEMBL269842)
Affinity DataKi:  13.2nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50375694(CHEMBL244265)
Affinity DataKi:  41.2nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed