Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50000699
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50008790(CHEMBL299224 | 5-[Pyridin-4-yl-(3-trifluoromethyl-...)
Affinity DataIC50: 3nMAssay Description:In vitro inhibition of Thromboxane synthase using [14C]arachidonic acid as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50008798(CHEMBL301280 | 7-(3-Pyridin-3-yl-bicyclo[2.2.1]hep...)
Affinity DataIC50: 7nMAssay Description:In vitro inhibition of thromboxane synthase using [14C]arachidonic acidMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM7962(CHEMBL537708 | 4-[2-(1H-imidazol-1-yl)ethoxy]benzo...)
Affinity DataIC50: 28nMAssay Description:In vitro inhibition of Thromboxane synthase using [14C]arachidonic acid as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50008794(CHEMBL50916 | 6-(3-Pyridin-3-yl-bicyclo[2.2.1]hept...)
Affinity DataIC50: 29nMAssay Description:In vitro inhibition of thromboxane synthase using [14C]arachidonic acidMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50008800(CHEMBL430965 | 7-(3-Pyridin-3-yl-bicyclo[2.2.1]hep...)
Affinity DataIC50: 50nMAssay Description:In vitro inhibition of thromboxane synthase using [14C]arachidonic acidMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50008797(CHEMBL51526 | 7-(3-Pyridin-3-yl-bicyclo[2.2.1]hept...)
Affinity DataIC50: 54nMAssay Description:In vitro inhibition of thromboxane synthase using [14C]arachidonic acidMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50008801(CHEMBL51158 | 7-(3-Pyridin-3-yl-bicyclo[2.2.1]hept...)
Affinity DataIC50: 54nMAssay Description:In vitro inhibition of thromboxane synthase using [14C]arachidonic acidMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50008793(CHEMBL298130 | 6-(3-Pyridin-3-yl-bicyclo[2.2.1]hep...)
Affinity DataIC50: 78nMAssay Description:In vitro inhibition of thromboxane synthase using [14C]arachidonic acidMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50008792(CHEMBL297712 | 7-[3-(Biphenyl-4-yloxymethyl)-2-pyr...)
Affinity DataIC50: 120nMAssay Description:In vitro inhibition of thromboxane synthase using [14C]arachidonic acidMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50008795(CHEMBL299878 | 7-(3-Pyridin-3-yl-bicyclo[2.2.1]hep...)
Affinity DataIC50: 125nMAssay Description:In vitro inhibition of thromboxane synthase using [14C]arachidonic acidMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50008796(CHEMBL51949 | 8-(3-Pyridin-3-yl-bicyclo[2.2.1]hept...)
Affinity DataIC50: 165nMAssay Description:In vitro inhibition of Thromboxane synthase using [14C]arachidonic acid as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50008799(CHEMBL51875 | 6-{3-[(4-Chloro-benzenesulfonylamino...)
Affinity DataIC50: 340nMAssay Description:In vitro inhibition of thromboxane synthase using [14C]arachidonic acidMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50008803(CHEMBL51618 | 7-(3-Pyridin-3-yl-7-oxa-bicyclo[2.2....)
Affinity DataIC50: 500nMAssay Description:In vitro inhibition of thromboxane synthase using [14C]arachidonic acidMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50008802(CHEMBL301520 | 7-[3-(5-Phenyl-pentyl)-3-pyridin-3-...)
Affinity DataIC50: 790nMAssay Description:In vitro inhibition of thromboxane synthase using [14C]arachidonic acidMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50008791(CHEMBL52344 | 7-(3-Pyridin-3-yl-7-oxa-bicyclo[2.2....)
Affinity DataIC50: 2.00E+3nMAssay Description:In vitro inhibition of thromboxane synthase using [14C]arachidonic acidMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed