Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50025744
TargetD(3) dopamine receptor(Rat)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50251027(CHEMBL458579 | CHEMBL517028 | (R)-(-)-2-(4-Hydroxy...)
Affinity DataIC50: 3.70nMAssay Description:Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in SF9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50251026(CHEMBL465054 | CHEMBL458397 | (R)-(-)-2-Phenyl-apo...)
Affinity DataIC50: 15nMAssay Description:Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in SF9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50251026(CHEMBL465054 | CHEMBL458397 | (R)-(-)-2-Phenyl-apo...)
Affinity DataIC50: 23nMAssay Description:Displacement of [3H]spiperone from rat dopamine D2 receptor in brain striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50251028(CHEMBL507567 | CHEMBL557547 | (R)-(-)-2-Methyl-apo...)
Affinity DataIC50: 43nMAssay Description:Displacement of [3H]spiperone from rat dopamine D2 receptor in brain striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM29644(APOMORPHINE HYDROCHLORIDE | SMR000059235 | APOMORP...)
Affinity DataIC50: 87nMAssay Description:Displacement of [3H]spiperone from rat dopamine D2 receptor in brain striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50251029((R)-(-)-2-(4-N,N-Dimethylaminophenyl)-apomorphine ...)
Affinity DataIC50: 484nMAssay Description:Displacement of [3H]spiperone from rat dopamine D2 receptor in brain striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50251027(CHEMBL458579 | CHEMBL517028 | (R)-(-)-2-(4-Hydroxy...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in SF9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50251027(CHEMBL458579 | CHEMBL517028 | (R)-(-)-2-(4-Hydroxy...)
Affinity DataKi:  4.10nMAssay Description:Displacement of [3H]spiperone from rat dopamine D2 receptor in brain striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50251027(CHEMBL458579 | CHEMBL517028 | (R)-(-)-2-(4-Hydroxy...)
Affinity DataKi:  4.10nMAssay Description:Displacement of [3H]spiperone from rat dopamine D2 receptor in brain striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50251026(CHEMBL465054 | CHEMBL458397 | (R)-(-)-2-Phenyl-apo...)
Affinity DataKi:  7.70nMAssay Description:Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in SF9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50251026(CHEMBL465054 | CHEMBL458397 | (R)-(-)-2-Phenyl-apo...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]spiperone from rat dopamine D2 receptor in brain striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50251028(CHEMBL507567 | CHEMBL557547 | (R)-(-)-2-Methyl-apo...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]spiperone from rat dopamine D2 receptor in brain striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50251034((R)-(-)-2-(4-dibenzo-furanyl)-apomorphine hydrochl...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in SF9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50251034((R)-(-)-2-(4-dibenzo-furanyl)-apomorphine hydrochl...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in SF9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM29644(APOMORPHINE HYDROCHLORIDE | SMR000059235 | APOMORP...)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in SF9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM29644(APOMORPHINE HYDROCHLORIDE | SMR000059235 | APOMORP...)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in SF9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50251028(CHEMBL507567 | CHEMBL557547 | (R)-(-)-2-Methyl-apo...)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in SF9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50251028(CHEMBL507567 | CHEMBL557547 | (R)-(-)-2-Methyl-apo...)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in SF9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM29644(APOMORPHINE HYDROCHLORIDE | SMR000059235 | APOMORP...)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]spiperone from rat dopamine D2 receptor in brain striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50251029((R)-(-)-2-(4-N,N-Dimethylaminophenyl)-apomorphine ...)
Affinity DataKi:  78nMAssay Description:Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in SF9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50251029((R)-(-)-2-(4-N,N-Dimethylaminophenyl)-apomorphine ...)
Affinity DataKi:  78nMAssay Description:Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in SF9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50251029((R)-(-)-2-(4-N,N-Dimethylaminophenyl)-apomorphine ...)
Affinity DataKi:  242nMAssay Description:Displacement of [3H]spiperone from rat dopamine D2 receptor in brain striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50251034((R)-(-)-2-(4-dibenzo-furanyl)-apomorphine hydrochl...)
Affinity DataKi:  1.63E+3nMAssay Description:Displacement of [3H]spiperone from rat dopamine D2 receptor in brain striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50251034((R)-(-)-2-(4-dibenzo-furanyl)-apomorphine hydrochl...)
Affinity DataKi:  1.63E+3nMAssay Description:Displacement of [3H]spiperone from rat dopamine D2 receptor in brain striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed