Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50038264
TargetEstrogen receptor beta(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50234790((E)-2-chloro-3,4'-dihydroxybiphenyl-4-carbaldehyde...)
Affinity DataEC50:  11nMAssay Description:Agonist activity at full length human ERbeta receptor expressed in human HEC-1 cells assessed as (ERE)2-pS2-luc reporter gene transcriptional activit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50234790((E)-2-chloro-3,4'-dihydroxybiphenyl-4-carbaldehyde...)
Affinity DataEC50:  26nMAssay Description:Agonist activity at full length human ERalpha receptor expressed in human HEC-1 cells assessed as (ERE)2-pS2-luc reporter gene transcriptional activi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50234790((E)-2-chloro-3,4'-dihydroxybiphenyl-4-carbaldehyde...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]estradiol from purified full length human ERbeta receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50234790((E)-2-chloro-3,4'-dihydroxybiphenyl-4-carbaldehyde...)
Affinity DataKi:  310nMAssay Description:Displacement of [3H]estradiol from purified full length human ERalpha receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed