Compile Data Set for Download or QSAR
Report error Found 93 Enz. Inhib. hit(s) with all data for entry = 2473
LigandPNGBDBM21034((1R,3R,5S,6S,18S)-6-hydroxy-18-(methoxymethyl)-1,5...)
Affinity DataIC50: 2.70nMpH: 7.5 T: 2°CAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21042((2R,3S,6E,14S,15S,17R)-6-({[2-(dimethylamino)ethyl...)
Affinity DataIC50: 5nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21036((2R,3S,6Z,14S,15S,17R)-6-({[3-(dimethylamino)propy...)
Affinity DataIC50: 6.40nMpH: 7.5 T: 2°CAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21036((2R,3S,6Z,14S,15S,17R)-6-({[3-(dimethylamino)propy...)
Affinity DataIC50: 8nMpH: 7.5 T: 2°CAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21041((2R,3S,6E,14S,15S,17R)-6-({[2-(dimethylamino)ethyl...)
Affinity DataIC50: 8.40nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21039((2R,3S,6Z,14S,15S,17R)-6-({tert-butyl[2-(dimethyla...)
Affinity DataIC50: 9.60nMpH: 7.5 T: 2°CAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21047((2R,3S,6E,14S,15S,17R)-8,14-dihydroxy-3-(methoxyme...)
Affinity DataIC50: 10nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21036((2R,3S,6Z,14S,15S,17R)-6-({[3-(dimethylamino)propy...)
Affinity DataIC50: 11nMpH: 7.5 T: 2°CAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21043((2R,3S,6E,14S,15S,17R)-6-({[3-(dimethylamino)propy...)
Affinity DataIC50: 12nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21036((2R,3S,6Z,14S,15S,17R)-6-({[3-(dimethylamino)propy...)
Affinity DataIC50: 13nMpH: 7.5 T: 2°CAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21049((2R,3S,6E,14S,15S,17R)-8,14-dihydroxy-3-(methoxyme...)
Affinity DataIC50: 15nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21046((2R,3S,6E,14S,15S,17R)-6-({bis[3-(dimethylamino)pr...)
Affinity DataIC50: 22nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21045((2R,3S,6E,14S,15S,17R)-6-({[2-(diethylamino)ethyl]...)
Affinity DataIC50: 24nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21048((2R,3S,6E,14S,15S,17R)-8,14-dihydroxy-3-(methoxyme...)
Affinity DataIC50: 24nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21065(methyl 1-{[(2R,3S,6E,14S,15S,17R)-17-(acetyloxy)-8...)
Affinity DataIC50: 31nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21066(1-{[(2R,3S,6E,14S,15S,17R)-17-(acetyloxy)-8,14-dih...)
Affinity DataIC50: 33nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21068((2R,3S,6E,14S,15S,17R)-8,14-dihydroxy-3-(methoxyme...)
Affinity DataIC50: 37nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21061((2R,3S,6E,14S,15S,17R)-6-({4-[3-(dimethylamino)pro...)
Affinity DataIC50: 38nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21057((2R,3S,6E,14S,15S,17R)-6-[(4-cyclohexylpiperazin-1...)
Affinity DataIC50: 43nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21063((2R,3S,6E,14S,15S,17R)-8,14-dihydroxy-3-(methoxyme...)
Affinity DataIC50: 45nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21044((2R,3S,6E,14S,15S,17R)-6-({[2-(diethylamino)ethyl]...)
Affinity DataIC50: 50nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21059((2R,3S,6E,14S,15S,17R)-8,14-dihydroxy-3-(methoxyme...)
Affinity DataIC50: 56nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21069((2R,3S,6E,14S,15S,17R)-8,14-dihydroxy-3-(methoxyme...)
Affinity DataIC50: 60nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21067((2R,3S,6E,14S,15S,17R)-8,14-dihydroxy-3-(methoxyme...)
Affinity DataIC50: 63nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21040((2R,3S,6Z,14S,15S,17R)-6-({benzyl[2-(dimethylamino...)
Affinity DataIC50: 66nMpH: 7.5 T: 2°CAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21062((2R,3S,6E,14S,15S,17R)-8,14-dihydroxy-3-(methoxyme...)
Affinity DataIC50: 78nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21058((2R,3S,6E,14S,15S,17R)-6-[(4-benzylpiperazin-1-yl)...)
Affinity DataIC50: 87nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21035(PX-866 | (2R,3S,6E,15S,17R)-6-{[bis(prop-2-en-1-yl...)
Affinity DataIC50: 88nMpH: 7.5 T: 2°CAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21060((2R,3S,6E,14S,15S,17R)-8,14-dihydroxy-3-(methoxyme...)
Affinity DataIC50: 90nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21056((2R,3S,6E,14S,15S,17R)-8,14-dihydroxy-3-(methoxyme...)
Affinity DataIC50: 91nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21070((2R,3S,6E,14S,15S,17R)-8,14-dihydroxy-3-(methoxyme...)
Affinity DataIC50: 104nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21050((2R,3S,6E,14S,15S,17R)-8,14-dihydroxy-3-(methoxyme...)
Affinity DataIC50: 127nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21064((2R,3S,6E,14S,15S,17R)-8,14-dihydroxy-3-(methoxyme...)
Affinity DataIC50: 172nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21052(4-({[(2R,3S,6E,14S,15S,17R)-17-(acetyloxy)-8,14-di...)
Affinity DataIC50: 193nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

LigandPNGBDBM21034((1R,3R,5S,6S,18S)-6-hydroxy-18-(methoxymethyl)-1,5...)
Affinity DataIC50: 193nMpH: 7.4 T: 2°CAssay Description:The enzyme was assayed in DELFIA format using purified FLAG-TOR in kinase buffer containing ATP and His6-S6K in the presence of inhibitor compounds. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21054((2R,3S,6E,14S,15S,17R)-6-{[(2,3-dihydroxypropyl)(m...)
Affinity DataIC50: 199nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

LigandPNGBDBM21061((2R,3S,6E,14S,15S,17R)-6-({4-[3-(dimethylamino)pro...)
Affinity DataIC50: 249nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21026((2R,3S,6Z,14S,15S,17R)-6-[(diethylamino)methyliden...)
Affinity DataIC50: 382nMpH: 7.5 T: 2°CAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21030((2R,3S,6Z,14S,15S,17R)-6-{[tert-butyl(methyl)amino...)
Affinity DataIC50: 440nMpH: 7.5 T: 2°CAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21055((2R,3S,6E,14S,15S,17R)-6-{[benzyl(2-cyanoethyl)ami...)
Affinity DataIC50: 444nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21033((2R,3S,6Z,14S,15S,17R)-8,14-dihydroxy-3-(methoxyme...)
Affinity DataIC50: 496nMpH: 7.5 T: 2°CAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

LigandPNGBDBM21067((2R,3S,6E,14S,15S,17R)-8,14-dihydroxy-3-(methoxyme...)
Affinity DataIC50: 568nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

LigandPNGBDBM21062((2R,3S,6E,14S,15S,17R)-8,14-dihydroxy-3-(methoxyme...)
Affinity DataIC50: 619nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21032((2R,3S,6Z,14S,15S,17R)-6-{[butyl(methyl)amino]meth...)
Affinity DataIC50: 635nMpH: 7.5 T: 2°CAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
LigandPNGBDBM21038((2R,3S,6Z,14S,15S,17R)-6-({[3-(dimethylamino)propy...)
Affinity DataIC50: 638nMpH: 7.5 T: 2°CAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

LigandPNGBDBM21059((2R,3S,6E,14S,15S,17R)-8,14-dihydroxy-3-(methoxyme...)
Affinity DataIC50: 692nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

LigandPNGBDBM21044((2R,3S,6E,14S,15S,17R)-6-({[2-(diethylamino)ethyl]...)
Affinity DataIC50: 767nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

LigandPNGBDBM21039((2R,3S,6Z,14S,15S,17R)-6-({tert-butyl[2-(dimethyla...)
Affinity DataIC50: 816nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

LigandPNGBDBM21057((2R,3S,6E,14S,15S,17R)-6-[(4-cyclohexylpiperazin-1...)
Affinity DataIC50: 820nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

LigandPNGBDBM21066(1-{[(2R,3S,6E,14S,15S,17R)-17-(acetyloxy)-8,14-dih...)
Affinity DataIC50: 822nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
Displayed 1 to 50 (of 93 total ) | Next | Last >>
Jump to: