Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 50022256
TargetC-C chemokine receptor type 2(Human)
National Institute of Pharmaceutical Education and Research (NIPER)

Curated by ChEMBL
LigandPNGBDBM50091438((E)-3-(3,4-dichlorophenyl)-N-(5-(4-(5-hydroxy-1H-i...)
Affinity DataKi:  50nMAssay Description:Antagonist activity at human CCR2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
National Institute of Pharmaceutical Education and Research (NIPER)

Curated by ChEMBL
LigandPNGBDBM50233075(3-(3,4-dichlorophenyl)-N-((1s,4s)-4-((4-(5-hydroxy...)
Affinity DataKi:  79nMAssay Description:Antagonist activity at human CCR2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
National Institute of Pharmaceutical Education and Research (NIPER)

Curated by ChEMBL
LigandPNGBDBM50233073(N-((1s,4s)-4-((4-(1H-indol-3-yl)piperidin-1-yl)met...)
Affinity DataKi:  126nMAssay Description:Antagonist activity at human CCR2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
National Institute of Pharmaceutical Education and Research (NIPER)

Curated by ChEMBL
LigandPNGBDBM50233071(3-(3,4-dichlorophenyl)-N-((1r,4r)-4-((4-(5-hydroxy...)
Affinity DataKi:  316nMAssay Description:Antagonist activity at human CCR2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
National Institute of Pharmaceutical Education and Research (NIPER)

Curated by ChEMBL
LigandPNGBDBM50091454((E)-3-(4-Bromo-phenyl)-N-{5-[4-(1H-indol-3-yl)-pip...)
Affinity DataKi:  350nMAssay Description:Antagonist activity at human CCR2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
National Institute of Pharmaceutical Education and Research (NIPER)

Curated by ChEMBL
LigandPNGBDBM50091458((E)-N-(5-(4-(1H-indol-3-yl)piperidin-1-yl)pentyl)-...)
Affinity DataKi:  420nMAssay Description:Antagonist activity at human CCR2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
National Institute of Pharmaceutical Education and Research (NIPER)

Curated by ChEMBL
LigandPNGBDBM50091465((E)-N-(5-(4-(1H-indol-3-yl)piperidin-1-yl)pentyl)-...)
Affinity DataKi:  460nMAssay Description:Antagonist activity at human CCR2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
National Institute of Pharmaceutical Education and Research (NIPER)

Curated by ChEMBL
LigandPNGBDBM50091445((E)-3-(4-Chloro-phenyl)-N-{5-[4-(1H-indol-3-yl)-pi...)
Affinity DataKi:  520nMAssay Description:Antagonist activity at human CCR2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
National Institute of Pharmaceutical Education and Research (NIPER)

Curated by ChEMBL
LigandPNGBDBM50091471(TCMDC-139236 | (E)-N-{5-[4-(1H-Indol-3-yl)-piperid...)
Affinity DataKi:  550nMAssay Description:Antagonist activity at human CCR2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
National Institute of Pharmaceutical Education and Research (NIPER)

Curated by ChEMBL
LigandPNGBDBM50091460((E)-3-(3-Chloro-phenyl)-N-{5-[4-(1H-indol-3-yl)-pi...)
Affinity DataKi:  560nMAssay Description:Antagonist activity at human CCR2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
National Institute of Pharmaceutical Education and Research (NIPER)

Curated by ChEMBL
LigandPNGBDBM50233072(N-((1r,4r)-4-((4-(1H-indol-3-yl)piperidin-1-yl)met...)
Affinity DataKi:  631nMAssay Description:Antagonist activity at human CCR2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
National Institute of Pharmaceutical Education and Research (NIPER)

Curated by ChEMBL
LigandPNGBDBM50091442(TCMDC-139333 | (E)-3-(3,4-Dichloro-phenyl)-N-{4-[4...)
Affinity DataKi:  660nMAssay Description:Antagonist activity at human CCR2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
National Institute of Pharmaceutical Education and Research (NIPER)

Curated by ChEMBL
LigandPNGBDBM50091448((E)-N-{5-[4-(1H-Indol-3-yl)-piperidin-1-yl]-pentyl...)
Affinity DataKi:  790nMAssay Description:Antagonist activity at human CCR2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
National Institute of Pharmaceutical Education and Research (NIPER)

Curated by ChEMBL
LigandPNGBDBM50091467((E)-N-{5-[4-(1H-Indol-3-yl)-piperidin-1-yl]-pentyl...)
Affinity DataKi:  790nMAssay Description:Antagonist activity at human CCR2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
National Institute of Pharmaceutical Education and Research (NIPER)

Curated by ChEMBL
LigandPNGBDBM50091439((E)-N-(5-(4-(1H-indol-3-yl)piperidin-1-yl)pentyl)c...)
Affinity DataKi:  870nMAssay Description:Antagonist activity at human CCR2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
National Institute of Pharmaceutical Education and Research (NIPER)

Curated by ChEMBL
LigandPNGBDBM50091468((E)-N-(5-(4-(1H-indol-3-yl)piperidin-1-yl)pentyl)-...)
Affinity DataKi:  1.20E+3nMAssay Description:Antagonist activity at human CCR2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
National Institute of Pharmaceutical Education and Research (NIPER)

Curated by ChEMBL
LigandPNGBDBM50091443((E)-3-Biphenyl-4-yl-N-{5-[4-(1H-indol-3-yl)-piperi...)
Affinity DataKi:  1.45E+3nMAssay Description:Antagonist activity at human CCR2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
National Institute of Pharmaceutical Education and Research (NIPER)

Curated by ChEMBL
LigandPNGBDBM50091441(1-(5-(4-(1H-indol-3-yl)piperidin-1-yl)pentyl)-3-(3...)
Affinity DataKi:  1.60E+3nMAssay Description:Antagonist activity at human CCR2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
National Institute of Pharmaceutical Education and Research (NIPER)

Curated by ChEMBL
LigandPNGBDBM50233074((E)-N-(5-(4-(1H-indol-3-yl)piperidin-1-yl)pentyl)-...)
Affinity DataKi:  1.70E+3nMAssay Description:Antagonist activity at human CCR2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
National Institute of Pharmaceutical Education and Research (NIPER)

Curated by ChEMBL
LigandPNGBDBM50091453((E)-N-(3-(4-(1H-indol-3-yl)piperidin-1-yl)propyl)-...)
Affinity DataKi:  2.50E+3nMAssay Description:Antagonist activity at human CCR2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
National Institute of Pharmaceutical Education and Research (NIPER)

Curated by ChEMBL
LigandPNGBDBM50091446((E)-3-(4-Cyano-phenyl)-N-{5-[4-(1H-indol-3-yl)-pip...)
Affinity DataKi:  2.80E+3nMAssay Description:Antagonist activity at human CCR2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
National Institute of Pharmaceutical Education and Research (NIPER)

Curated by ChEMBL
LigandPNGBDBM50091464(2-(3,4-Dichloro-phenyl)-N-{5-[4-(1H-indol-3-yl)-pi...)
Affinity DataKi:  4.40E+3nMAssay Description:Antagonist activity at human CCR2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
National Institute of Pharmaceutical Education and Research (NIPER)

Curated by ChEMBL
LigandPNGBDBM50091466((E)-N-(5-(4-(1H-indol-3-yl)piperidin-1-yl)pentyl)-...)
Affinity DataKi:  4.40E+3nMAssay Description:Antagonist activity at human CCR2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
National Institute of Pharmaceutical Education and Research (NIPER)

Curated by ChEMBL
LigandPNGBDBM50091459(TCMDC-139112 | N-(5-(4-(1H-indol-3-yl)piperidin-1-...)
Affinity DataKi:  5.10E+3nMAssay Description:Antagonist activity at human CCR2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
National Institute of Pharmaceutical Education and Research (NIPER)

Curated by ChEMBL
LigandPNGBDBM50091444(Biphenyl-4-carboxylic acid {5-[4-(1H-indol-3-yl)-p...)
Affinity DataKi:  5.40E+3nMAssay Description:Antagonist activity at human CCR2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
National Institute of Pharmaceutical Education and Research (NIPER)

Curated by ChEMBL
LigandPNGBDBM50091450(3-(3,4-Dichloro-phenyl)-N-{5-[4-(1H-indol-3-yl)-pi...)
Affinity DataKi:  5.90E+3nMAssay Description:Antagonist activity at human CCR2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
National Institute of Pharmaceutical Education and Research (NIPER)

Curated by ChEMBL
LigandPNGBDBM50091455((E)-N-(5-(4-(1H-indol-3-yl)piperidin-1-yl)pentyl)-...)
Affinity DataKi:  6.30E+3nMAssay Description:Antagonist activity at human CCR2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
National Institute of Pharmaceutical Education and Research (NIPER)

Curated by ChEMBL
LigandPNGBDBM50091472(N-(5-(4-(1H-indol-3-yl)piperidin-1-yl)pentyl)-4-br...)
Affinity DataKi:  7.10E+3nMAssay Description:Antagonist activity at human CCR2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
National Institute of Pharmaceutical Education and Research (NIPER)

Curated by ChEMBL
LigandPNGBDBM50091452((E)-3-(4-Acetylamino-phenyl)-N-{5-[4-(1H-indol-3-y...)
Affinity DataKi:  1.29E+4nMAssay Description:Antagonist activity at human CCR2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed