Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50038072
TargetSomatostatin receptor type 5(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50232821(CHEMBL252764 | L-817,818 | (S)-((S)-2-aminopropyl)...)
Affinity DataIC50: 0.400nMAssay Description:Binding affinity to sst5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50159392(SRIF-28 | (4R,7R,10S,13S,16S,19S,22S,25S,28S,31S,3...)
Affinity DataIC50: 1.60nMAssay Description:Displacement of [125I](Leu8,D-Trp22,Tyr25)-SRIF28 from human sst4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50159392(SRIF-28 | (4R,7R,10S,13S,16S,19S,22S,25S,28S,31S,3...)
Affinity DataIC50: 2.10nMAssay Description:Displacement of [125I](Leu8,D-Trp22,Tyr25)-SRIF28 from human sst5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50159392(SRIF-28 | (4R,7R,10S,13S,16S,19S,22S,25S,28S,31S,3...)
Affinity DataIC50: 2.30nMAssay Description:Displacement of [125I](Leu8,D-Trp22,Tyr25)-SRIF28 from human sst1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50159392(SRIF-28 | (4R,7R,10S,13S,16S,19S,22S,25S,28S,31S,3...)
Affinity DataIC50: 3nMAssay Description:Displacement of [125I](Leu8,D-Trp22,Tyr25)-SRIF28 from human sst2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50159392(SRIF-28 | (4R,7R,10S,13S,16S,19S,22S,25S,28S,31S,3...)
Affinity DataIC50: 3.60nMAssay Description:Displacement of [125I](Leu8,D-Trp22,Tyr25)-SRIF28 from human sst3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50232819((2S,5R,8S,11S,14S,16Z,19S)-19-[(2R)-2-amino-3-phen...)
Affinity DataIC50: 28nMAssay Description:Displacement of [125I](Leu8,D-Trp22,Tyr25)-SRIF28 from human sst5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50232819((2S,5R,8S,11S,14S,16Z,19S)-19-[(2R)-2-amino-3-phen...)
Affinity DataIC50: 44nMAssay Description:Displacement of [125I](Leu8,D-Trp22,Tyr25)-SRIF28 from human sst2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50232818((2S,5R,8S,11S,14S,19S)-19-[(2R)-2-amino-3-phenylpr...)
Affinity DataIC50: 49nMAssay Description:Displacement of [125I](Leu8,D-Trp22,Tyr25)-SRIF28 from human sst2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50232817((2S,5R,8S,11S,14S,16Z,19S)-19-[(2R)-2-amino-3-phen...)
Affinity DataIC50: 141nMAssay Description:Displacement of [125I](Leu8,D-Trp22,Tyr25)-SRIF28 from human sst4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50232818((2S,5R,8S,11S,14S,19S)-19-[(2R)-2-amino-3-phenylpr...)
Affinity DataIC50: 203nMAssay Description:Displacement of [125I](Leu8,D-Trp22,Tyr25)-SRIF28 from human sst5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50232817((2S,5R,8S,11S,14S,16Z,19S)-19-[(2R)-2-amino-3-phen...)
Affinity DataIC50: 206nMAssay Description:Displacement of [125I](Leu8,D-Trp22,Tyr25)-SRIF28 from human sst5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50232818((2S,5R,8S,11S,14S,19S)-19-[(2R)-2-amino-3-phenylpr...)
Affinity DataIC50: 214nMAssay Description:Displacement of [125I](Leu8,D-Trp22,Tyr25)-SRIF28 from human sst4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50232819((2S,5R,8S,11S,14S,16Z,19S)-19-[(2R)-2-amino-3-phen...)
Affinity DataIC50: 412nMAssay Description:Displacement of [125I](Leu8,D-Trp22,Tyr25)-SRIF28 from human sst4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50232817((2S,5R,8S,11S,14S,16Z,19S)-19-[(2R)-2-amino-3-phen...)
Affinity DataIC50: 961nMAssay Description:Displacement of [125I](Leu8,D-Trp22,Tyr25)-SRIF28 from human sst1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50232818((2S,5R,8S,11S,14S,19S)-19-[(2R)-2-amino-3-phenylpr...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I](Leu8,D-Trp22,Tyr25)-SRIF28 from human sst3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50232817((2S,5R,8S,11S,14S,16Z,19S)-19-[(2R)-2-amino-3-phen...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I](Leu8,D-Trp22,Tyr25)-SRIF28 from human sst3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50232818((2S,5R,8S,11S,14S,19S)-19-[(2R)-2-amino-3-phenylpr...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I](Leu8,D-Trp22,Tyr25)-SRIF28 from human sst1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50232819((2S,5R,8S,11S,14S,16Z,19S)-19-[(2R)-2-amino-3-phen...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I](Leu8,D-Trp22,Tyr25)-SRIF28 from human sst3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50232819((2S,5R,8S,11S,14S,16Z,19S)-19-[(2R)-2-amino-3-phen...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I](Leu8,D-Trp22,Tyr25)-SRIF28 from human sst1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50232817((2S,5R,8S,11S,14S,16Z,19S)-19-[(2R)-2-amino-3-phen...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I](Leu8,D-Trp22,Tyr25)-SRIF28 from human sst2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed