Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50022216
TargetCytochrome P450 2C9(Human)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50232748(6-(2-(methylsulfonyl)propan-2-yl)-8-(3-(pyridin-4-...)
Affinity DataIC50: 110nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50174022(L-454560 | 8-(3-methoxyphenyl)-6-(pyridin-4-ylmeth...)
Affinity DataIC50: 200nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50232743(8-(3'-methanesulfonyl-biphenyl-3-yl)-6-(1-methanes...)
Affinity DataIC50: 580nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50232730(6-(2-(methylsulfonyl)propan-2-yl)-8-(3-(pyridin-3-...)
Affinity DataIC50: 630nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50232737(8-(4'-methanesulfonyl-biphenyl-3-yl)-6-(1-methanes...)
Affinity DataIC50: 730nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50232733(1-isopropyl-3-(5-{3-[6-(1-methanesulfonyl-1-methyl...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50232740(8-(4'-methanesulfonylmethyl-biphenyl-3-yl)-6-(1-me...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50232727(3-{3'-[6-(1-methanesulfonyl-1-methyl-ethyl)-quinol...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50232744(8-(3-(1H-imidazo[4,5-b]pyridin-6-yl)phenyl)-6-(2-(...)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50232731(2-{3'-[6-(1-methanesulfonyl-1-methyl-ethyl)-quinol...)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50232731(2-{3'-[6-(1-methanesulfonyl-1-methyl-ethyl)-quinol...)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50232729(5-{3-[6-(1-methanesulfonyl-1-methyl-ethyl)-quinoli...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50232747(3-{3'-[6-(1-methanesulfonyl-1-methyl-ethyl)-quinol...)
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50232732(3-{3'-[6-(1-methanesulfonyl-1-methyl-ethyl)-quinol...)
Affinity DataIC50: 9.80E+3nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50232741(2-(5-{3-[6-(1-methanesulfonyl-1-methyl-ethyl)-quin...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50232752(3-{3'-[6-(1-methanesulfonyl-1-methyl-ethyl)-quinol...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50232745(6-(1-methanesulfonyl-1-methyl-ethyl)-8-[3-(6-methy...)
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50232736(6-(1-methanesulfonyl-1-methyl-ethyl)-8-[3-(1-oxy-p...)
Affinity DataIC50: 3.60E+4nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed