Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50021716
TargetPotassium voltage-gated channel subfamily H member 2(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50227131(N-(1-(4-chloro-3-ethoxybenzyl)piperidin-4-yl)-3-(m...)
Affinity DataIC50: 1.30E+3nMAssay Description:Binding affinity to human ERG channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50227129(N-(1-(4-chloro-3-ethoxybenzyl)piperidin-4-yl)-5-me...)
Affinity DataKi:  20nMAssay Description:Binding affinity to human SST5RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50227132(4-tert-butyl-N-(1-((1,4-dimethoxynaphthalen-2-yl)m...)
Affinity DataKi:  20nMAssay Description:Binding affinity to human SST5RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50227130(N-(1-((1,4-dimethoxynaphthalen-2-yl)methyl)piperid...)
Affinity DataKi:  40nMAssay Description:Binding affinity to human SST5RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50227131(N-(1-(4-chloro-3-ethoxybenzyl)piperidin-4-yl)-3-(m...)
Affinity DataKi:  60nMAssay Description:Binding affinity to human SST5RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50227128(N-(1-((1,4-dimethoxynaphthalen-2-yl)methyl)piperid...)
Affinity DataKi:  120nMAssay Description:Binding affinity to human SST5RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50227129(N-(1-(4-chloro-3-ethoxybenzyl)piperidin-4-yl)-5-me...)
Affinity DataKi:  270nMAssay Description:Binding affinity to human histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50227133(1'-[(1,4-dimethoxynaphthalen-2-yl)methyl]-3H-spiro...)
Affinity DataKi:  1.10E+3nMAssay Description:Binding affinity to human SST5RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50227131(N-(1-(4-chloro-3-ethoxybenzyl)piperidin-4-yl)-3-(m...)
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity to human histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50227129(N-(1-(4-chloro-3-ethoxybenzyl)piperidin-4-yl)-5-me...)
Affinity DataKi:  5.10E+3nMAssay Description:Binding affinity to human SST1RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50227129(N-(1-(4-chloro-3-ethoxybenzyl)piperidin-4-yl)-5-me...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human SST3RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50227129(N-(1-(4-chloro-3-ethoxybenzyl)piperidin-4-yl)-5-me...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human SST2RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed