Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50021597
TargetHistone deacetylase 1(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226108(N-(2-aminophenyl)-4-((4-oxo-4H-chromen-3-yl)methyl...)
Affinity DataIC50: 30nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226109(N-(2-aminophenyl)-4-((2,4-dioxo-1,2-dihydrothieno[...)
Affinity DataIC50: 60nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226111(N-(2-aminophenyl)-4-((2,4-dioxo-1,2-dihydroquinazo...)
Affinity DataIC50: 60nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226107(N-(2-aminophenyl)-4-((2-methyl-4-oxoquinazolin-3(4...)
Affinity DataIC50: 80nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226117(N-(2-aminophenyl)-4-((4-oxochroman-3-yl)methyl)ben...)
Affinity DataIC50: 90nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226115(N-(2-aminophenyl)-4-((1-oxoisoindolin-2-yl)methyl)...)
Affinity DataIC50: 100nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226116(4-((1-(4-methoxybenzyl)-2,4-dioxo-1,2-dihydroquina...)
Affinity DataIC50: 100nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226112(N-(2-aminophenyl)-4-((2,4-dioxo-2H-benzo[e][1,3]ox...)
Affinity DataIC50: 100nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226120(N-(2-aminophenyl)-4-((1-oxo-2,3-dihydro-1H-inden-2...)
Affinity DataIC50: 100nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226114(N-(2-aminophenyl)-4-((4-oxoquinazolin-3(4H)-yl)met...)
Affinity DataIC50: 100nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226118(N-(2-aminophenyl)-4-((1-methyl-2,4-dioxo-1,2-dihyd...)
Affinity DataIC50: 100nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226110(N-(2-aminophenyl)-4-((1,3-dioxoisoindolin-2-yl)met...)
Affinity DataIC50: 200nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226123(N-(2-aminophenyl)-4-((1-ethyl-2,4-dioxo-1,2-dihydr...)
Affinity DataIC50: 200nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226124(N-(2-aminophenyl)-4-((4-oxobenzo[d][1,2,3]triazin-...)
Affinity DataIC50: 200nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226106(N-(2-aminophenyl)-4-((4-oxothieno[3,2-d]pyrimidin-...)
Affinity DataIC50: 200nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226119(N-(2-aminophenyl)-4-((1-ethyl-2,4-dioxo-1,2-dihydr...)
Affinity DataIC50: 300nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226121(N-(2-aminophenyl)-4-((1-(2-(dimethylamino)ethyl)-2...)
Affinity DataIC50: 300nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226122(N-(2-aminophenyl)-4-((1-(2-morpholinoethyl)-2,4-di...)
Affinity DataIC50: 400nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226113(N-(2-aminophenyl)-4-(chroman-3-ylmethyl)benzamide ...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed