Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50038460
TargetTelomerase reverse transcriptase(Human)
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50339190(telomestatin | CHEMBL443683)
Affinity DataIC50: 0.640nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells treated before telomerase elongation by telomeric repeat amplification protocol assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50339190(telomestatin | CHEMBL443683)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells treated after telomerase elongation by telomeric repeat amplification protocol assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50376748(CHEMBL259739 | Phen-DC3)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells treated before telomerase elongation by telomeric repeat amplification protocol assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50376748(CHEMBL259739 | Phen-DC3)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells treated after telomerase elongation by telomeric repeat amplification protocol assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50134030(N,N'-(9-{[4-(dimethylamino)phenyl]amino}acridine-3...)
Affinity DataIC50: 45nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells treated before telomerase elongation by telomeric repeat amplification protocol assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50376747(CHEMBL409247)
Affinity DataIC50: 45nMAssay Description:Inhibition of human telomerase expressed in in HEK293T cells in presence of primer (T2AG3)4 by primer extension assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50376747(CHEMBL409247)
Affinity DataIC50: 52nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells treated before telomerase elongation by telomeric repeat amplification protocol assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50339190(telomestatin | CHEMBL443683)
Affinity DataIC50: 58nMAssay Description:Inhibition of human telomerase expressed in in HEK293T cells in presence of primer (T2AG3)4 by primer extension assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50376747(CHEMBL409247)
Affinity DataIC50: 63nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells treated after telomerase elongation by telomeric repeat amplification protocol assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50376748(CHEMBL259739 | Phen-DC3)
Affinity DataIC50: 63nMAssay Description:Inhibition of human telomerase expressed in in HEK293T cells in presence of primer (T2AG3)4 by primer extension assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50134030(N,N'-(9-{[4-(dimethylamino)phenyl]amino}acridine-3...)
Affinity DataIC50: 65nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells treated after telomerase elongation by telomeric repeat amplification protocol assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50107609(CHEMBL2170855 | CHEMBL337559 | TMPyP4 | 5,10,15,20...)
Affinity DataIC50: 550nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells treated before telomerase elongation by telomeric repeat amplification protocol assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50107609(CHEMBL2170855 | CHEMBL337559 | TMPyP4 | 5,10,15,20...)
Affinity DataIC50: 710nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells in presence of primer (T2AG3)3 by primer extension assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50107609(CHEMBL2170855 | CHEMBL337559 | TMPyP4 | 5,10,15,20...)
Affinity DataIC50: 740nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells treated after telomerase elongation by telomeric repeat amplification protocol assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50376748(CHEMBL259739 | Phen-DC3)
Affinity DataIC50: 790nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells in presence of primer (T2AG3)3 by primer extension assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50134030(N,N'-(9-{[4-(dimethylamino)phenyl]amino}acridine-3...)
Affinity DataIC50: 830nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells in presence of primer (T2AG3)3 by primer extension assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50339190(telomestatin | CHEMBL443683)
Affinity DataIC50: 900nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells in presence of primer (T2AG3)3 by primer extension assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50339190(telomestatin | CHEMBL443683)
Affinity DataIC50: 1.15E+3nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells in presence of primer TS by primer extension assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50376748(CHEMBL259739 | Phen-DC3)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells in presence of primer TS by primer extension assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50376747(CHEMBL409247)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells in presence of primer (T2AG3)3 by primer extension assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50376747(CHEMBL409247)
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells in presence of primer TS by primer extension assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed