Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50021302
TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM50223090(3-(4-(3-chloro-4-fluorophenylamino)quinazolin-6-yl...)
Affinity DataIC50: 14nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM5446(Erlotinib | OSI-774 | N-(3-ethynylphenyl)-6,7-bis(...)
Affinity DataIC50: 23nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM50095259(N-(3-ethynylphenyl)-6,7-dimethoxyquinazolin-4-amin...)
Affinity DataIC50: 29nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM5447(ZD1839 | N-(3-chloro-4-fluorophenyl)-7-methoxy-6-[...)
Affinity DataIC50: 39nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM50223084(N-(3-chloro-4-fluorophenyl)-6-(3-morpholinoprop-1-...)
Affinity DataIC50: 50nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM50223082(N-(3-chloro-4-fluorophenyl)-6-(3-(piperidin-1-yl)p...)
Affinity DataIC50: 89nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM50223095(4-(4-(3-chloro-4-fluorophenylamino)quinazolin-6-yl...)
Affinity DataIC50: 95nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM50223092(5-(4-(3-chloro-4-fluorophenylamino)quinazolin-6-yl...)
Affinity DataIC50: 114nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM50223085(N-(3-chloro-4-fluorophenyl)-6-ethynylquinazolin-4-...)
Affinity DataIC50: 127nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM50223093(4-(4-(3-chloro-4-fluorophenylamino)quinazolin-6-yl...)
Affinity DataIC50: 152nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM50223088(4-(4-(3-chloro-4-fluorophenylamino)quinazolin-6-yl...)
Affinity DataIC50: 186nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM50223086(4-(3-(6,7-dimethoxyquinazolin-4-ylamino)phenyl)-2-...)
Affinity DataIC50: 206nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM50223094(N-(3-chloro-4-fluorophenyl)-6-(2-phenylethynyl)qui...)
Affinity DataIC50: 331nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM50223091(4-(3-(6,7-dimethoxyquinazolin-4-ylamino)phenyl)but...)
Affinity DataIC50: 402nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM50223087(6,7-dimethoxy-N-(3-(2-phenylethynyl)phenyl)quinazo...)
Affinity DataIC50: 921nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM50223089(5-(3-(6,7-dimethoxyquinazolin-4-ylamino)phenyl)pen...)
Affinity DataIC50: 1.36E+3nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM50223096(N-(3-chloro-4-fluorophenyl)-6-(2-(thiophen-2-yl)et...)
Affinity DataIC50: 1.64E+3nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM50223083(3-(3-(6,7-dimethoxyquinazolin-4-ylamino)phenyl)pro...)
Affinity DataIC50: 1.64E+3nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed